Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 829 件

1X4T
DownloadVisualize
BU of 1x4t by Molmil
Solution structure of Isy1 domain in hypothetical protein
分子名称: hypothetical protein LOC57905
著者He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2005-05-14
公開日2005-11-14
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of Isy1 domain in hypothetical protein
To be Published
1X5O
DownloadVisualize
BU of 1x5o by Molmil
Solution structure of RRM domain in RNA binding motif, single-stranded interacting protein 1
分子名称: RNA binding motif, single-stranded interacting protein 1
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2005-05-16
公開日2005-11-16
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RRM domain in RNA binding motif, single-stranded interacting protein 1
To be Published
1WEM
DownloadVisualize
BU of 1wem by Molmil
Solution structure of PHD domain in death inducer-obliterator 1(DIO-1)
分子名称: Death associated transcription factor 1, ZINC ION
著者He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-05-25
公開日2004-11-25
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of PHD domain in death inducer-obliterator 1(DIO-1)
To be Published
1WF1
DownloadVisualize
BU of 1wf1 by Molmil
Solution structure of RRM domain in RNA-binding protein NP_057951
分子名称: RNA-binding protein Raly
著者He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-05-25
公開日2004-11-25
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RRM domain in RNA-binding protein NP_057951
To be Published
1WG6
DownloadVisualize
BU of 1wg6 by Molmil
Solution structure of PDZ domain in protein XP_110852
分子名称: HYPOTHETICAL PROTEIN (RIKEN cDNA 2810455B10)
著者He, F, Hanaki, K, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-05-27
公開日2004-11-27
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of PDZ domain in protein XP_110852
To be Published
1WHQ
DownloadVisualize
BU of 1whq by Molmil
Solution structure of the N-terminal dsRBD from hypothetical protein BAB28848
分子名称: RNA helicase A
著者Nagata, T, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-05-28
公開日2004-11-28
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the N-terminal dsRBD from hypothetical protein BAB28848
To be Published
5H09
DownloadVisualize
BU of 5h09 by Molmil
Crystal structure of HCK complexed with a pyrrolo-pyrimidine inhibitor (S)-ethyl2-(((1r,4S)-4-(4-amino-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclohexyl)amino)-4-methylpentanoate
分子名称: Tyrosine-protein kinase HCK, ethyl (2~{S})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methyl-pentanoate
著者Tomabechi, Y, Kukimoto-Niino, M, Shirouzu, M.
登録日2016-10-04
公開日2017-10-04
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.945 Å)
主引用文献Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen.
Bioorg. Med. Chem., 25, 2017
1X4J
DownloadVisualize
BU of 1x4j by Molmil
Solution structure of RING finger in RING finger protein 38
分子名称: RING finger protein 38, ZINC ION
著者He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2005-05-14
公開日2005-11-14
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RING finger in RING finger protein 38
To be Published
1WEZ
DownloadVisualize
BU of 1wez by Molmil
Solution structure of RRM domain in heterogeneous nuclear ribonucleoprotein H'
分子名称: Heterogeneous nuclear ribonucleoprotein H'
著者He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-05-25
公開日2004-11-25
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RRM domain in heterogeneous nuclear ribonucleoprotein H'
To be Published
1X4L
DownloadVisualize
BU of 1x4l by Molmil
Solution structure of LIM domain in Four and a half LIM domains protein 2
分子名称: Skeletal muscle LIM-protein 3, ZINC ION
著者He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2005-05-14
公開日2005-11-14
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of LIM domain in Four and a half LIM domains protein 2
To be Published
5H0B
DownloadVisualize
BU of 5h0b by Molmil
Crystal structure of HCK complexed with a pyrrolo-pyrimidine inhibitor (S)-2-(((1r,4S)-4-(4-amino-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclohexyl)amino)-4-methylpentanoic acid
分子名称: (2~{S})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]azaniumyl]-4-methyl-pentanoate, Tyrosine-protein kinase HCK
著者Tomabechi, Y, Kukimoto-Niino, M, Shirouzu, M.
登録日2016-10-04
公開日2017-10-11
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.651 Å)
主引用文献Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen.
Bioorg. Med. Chem., 25, 2017
1X5P
DownloadVisualize
BU of 1x5p by Molmil
Solution structure of RRM domain in Parp14
分子名称: Negative elongation factor E
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2005-05-16
公開日2005-11-16
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RRM domain in Parp14
To be Published
1WEU
DownloadVisualize
BU of 1weu by Molmil
Solution structure of PHD domain in ING1-like protein BAC25009
分子名称: ZINC ION, inhibitor of growth family, member 4
著者He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-05-25
公開日2004-11-25
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of PHD domain in ING1-like protein BAC25009
To be Published
1WZ7
DownloadVisualize
BU of 1wz7 by Molmil
Crystal structure of enhancer of rudimentary homologue (ERH)
分子名称: Enhancer of rudimentary homolog
著者Arai, R, Kukimoto-Niino, M, Uda-Tochio, H, Morita, S, Uchikubo-Kamo, T, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2005-02-26
公開日2005-05-03
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure of an enhancer of rudimentary homolog (ERH) at 2.1 Angstroms resolution.
Protein Sci., 14, 2005
1WHU
DownloadVisualize
BU of 1whu by Molmil
Solution structure of the alpha-helical domain from mouse hypothetical PNPase
分子名称: polynucleotide phosphorylase; 3'-5' RNA exonuclease
著者Nagata, T, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-05-28
公開日2004-11-28
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the alpha-helical domain from mouse hypothetical PNPase
To be Published
1X4D
DownloadVisualize
BU of 1x4d by Molmil
Solution structure of RRM domain in Matrin 3
分子名称: Matrin 3
著者He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2005-05-14
公開日2005-11-14
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RRM domain in Matrin 3
To be Published
5H0H
DownloadVisualize
BU of 5h0h by Molmil
Crystal structure of HCK complexed with a pyrrolo-pyrimidine inhibitor (S)-2-(((1r,4S)-4-(4-amino-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclohexyl)amino)-N,N,4-trimethylpentanamide
分子名称: (2~{S})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-~{N},~{N},4-trimethyl-pentanamide, Tyrosine-protein kinase HCK
著者Tomabechi, Y, Kukimoto-Niino, M, Shirouzu, M.
登録日2016-10-04
公開日2017-10-04
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen.
Bioorg. Med. Chem., 25, 2017
5H0G
DownloadVisualize
BU of 5h0g by Molmil
Crystal structure of HCK complexed with a pyrrolo-pyrimidine inhibitor (S)-2-(((1r,4S)-4-(4-amino-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclohexyl)amino)-N,4-dimethylpentanamide
分子名称: (2~{S})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-~{N},4-dimethyl-pentanamide, Tyrosine-protein kinase HCK
著者Tomabechi, Y, Kukimoto-Niino, M, Shirouzu, M.
登録日2016-10-04
公開日2017-10-04
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen.
Bioorg. Med. Chem., 25, 2017
5H0E
DownloadVisualize
BU of 5h0e by Molmil
Crystal structure of HCK complexed with a pyrrolo-pyrimidine inhibitor (S)-2-(((1r,4S)-4-(4-amino-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclohexyl)amino)-4-methylpentanamide
分子名称: (2~{S})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methyl-pentanamide, Tyrosine-protein kinase HCK
著者Tomabechi, Y, Kukimoto-Niino, M, Shirouzu, M.
登録日2016-10-04
公開日2017-10-04
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen.
Bioorg. Med. Chem., 25, 2017
8I94
DownloadVisualize
BU of 8i94 by Molmil
Structure of flavone 4'-O-glucoside 7-O-glucosyltransferase from Nemophila menziesii, complex with luteolin
分子名称: 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4-one, Glycosyltransferase, SULFATE ION
著者Murayama, K, Kato-Murayama, M, Shirouzu, M.
登録日2023-02-06
公開日2024-02-14
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.43 Å)
主引用文献Molecular basis of ligand recognition specificity of flavone glucosyltransferases in Nemophila menziesii.
Arch.Biochem.Biophys., 753, 2024
8I8Z
DownloadVisualize
BU of 8i8z by Molmil
Structure of flavone 4'-O-glucoside 7-O-glucosyltransferase from Nemophila menziesii, apo form
分子名称: Glycosyltransferase, SULFATE ION
著者Murayama, K, Kato-Murayama, M, Shirouzu, M.
登録日2023-02-06
公開日2024-02-14
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Molecular basis of ligand recognition specificity of flavone glucosyltransferases in Nemophila menziesii.
Arch.Biochem.Biophys., 753, 2024
4LM5
DownloadVisualize
BU of 4lm5 by Molmil
Crystal structure of Pim1 in complex with 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol (resulting from displacement of SKF86002)
分子名称: 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol, GLYCEROL, Serine/threonine-protein kinase pim-1
著者Parker, L.J, Tanaka, A, Handa, N, Honda, K, Tomabechi, Y, Shirouzu, M, Yokoyama, S.
登録日2013-07-10
公開日2014-02-12
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Kinase crystal identification and ATP-competitive inhibitor screening using the fluorescent ligand SKF86002.
Acta Crystallogr.,Sect.D, 70, 2014
4LL5
DownloadVisualize
BU of 4ll5 by Molmil
Crystal Structure of Pim-1 in complex with the fluorescent compound SKF86002
分子名称: 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole, CALCIUM ION, GLYCEROL, ...
著者Parker, L.J, Tanaka, A, Handa, N, Honda, K, Tomabechi, Y, Shirouzu, M, Yokoyama, S.
登録日2013-07-09
公開日2014-02-12
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Kinase crystal identification and ATP-competitive inhibitor screening using the fluorescent ligand SKF86002.
Acta Crystallogr.,Sect.D, 70, 2014
4LMU
DownloadVisualize
BU of 4lmu by Molmil
Crystal structure of Pim1 in complex with the inhibitor Quercetin (resulting from displacement of SKF86002)
分子名称: 3,5,7,3',4'-PENTAHYDROXYFLAVONE, GLYCEROL, Serine/threonine-protein kinase pim-1
著者Parker, L.J, Tanaka, A, Handa, N, Honda, K, Tomabechi, Y, Shirouzu, M, Yokoyama, S.
登録日2013-07-11
公開日2014-02-12
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Kinase crystal identification and ATP-competitive inhibitor screening using the fluorescent ligand SKF86002.
Acta Crystallogr.,Sect.D, 70, 2014
8I90
DownloadVisualize
BU of 8i90 by Molmil
Structure of flavone 4'-O-glucoside 7-O-glucosyltransferase from Nemophila menziesii, complex with UDP-glucose
分子名称: Glycosyltransferase, URIDINE-5'-DIPHOSPHATE-GLUCOSE
著者Murayama, K, Kato-Murayama, M, Shirouzu, M.
登録日2023-02-06
公開日2024-02-14
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Molecular basis of ligand recognition specificity of flavone glucosyltransferases in Nemophila menziesii.
Arch.Biochem.Biophys., 753, 2024

221051

件を2024-06-12に公開中

PDB statisticsPDBj update infoContact PDBjnumon