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PDB: 1 results

7E2E
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BU of 7e2e by Molmil
Crystal structure of the Estrogen-Related Receptor alpha (ERRalpha) ligand-binding domain (LBD) in complex with an agonist DS45500853 and a PGC-1alpha peptide
Descriptor: 1-[4-(3-tert-butyl-4-oxidanyl-phenoxy)phenyl]ethanone, IODIDE ION, Peroxisome proliferator-activated receptor gamma coactivator 1-alpha, ...
Authors:Ito, S, Shinozuka, T, Kimura, T, Izumi, M, Wakabayashi, K.
Deposit date:2021-02-05
Release date:2021-06-30
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Discovery of a Novel Class of ERR alpha Agonists.
Acs Med.Chem.Lett., 12, 2021

218853

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