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PDB: 1 results

8TUC
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BU of 8tuc by Molmil
Unphosphorylated CaMKK2 in complex with CC-8977
Descriptor: (4M)-2-cyclopentyl-4-(7-ethoxyquinazolin-4-yl)benzoic acid, 1,2-ETHANEDIOL, Calcium/calmodulin-dependent protein kinase kinase 2, ...
Authors:Bernard, S.M, Shanmugasundaram, V, D'Agostino, L.
Deposit date:2023-08-16
Release date:2023-12-13
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Identification of Small Molecule Inhibitors and Ligand Directed Degraders of Calcium/Calmodulin Dependent Protein Kinase Kinase 1 and 2 (CaMKK1/2).
J.Med.Chem., 66, 2023

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