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PDB: 27265 件

6CNO
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Cryo-EM structure of the human SK4/calmodulin channel complex in the Ca2+ bound state II
分子名称: CALCIUM ION, Calmodulin-1, Intermediate conductance calcium-activated potassium channel protein 4
著者Lee, C.H, MacKinnon, R.
登録日2018-03-08
公開日2018-05-02
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (4.7 Å)
主引用文献Activation mechanism of a human SK-calmodulin channel complex elucidated by cryo-EM structures.
Science, 360, 2018
6COE
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AtHNL enantioselectivity mutant At-A9-H7 Apo Y13C,Y121L,P126F,L128W,C131T,F179L,A209I with benzaldehyde, MANDELIC ACID NITRILE
分子名称: (2R)-hydroxy(phenyl)ethanenitrile, (S)-MANDELIC ACID NITRILE, Alpha-hydroxynitrile lyase, ...
著者Jones, B.J, Kazlauskas, R.J, Desrouleaux, R.
登録日2018-03-12
公開日2019-03-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.844 Å)
主引用文献AtHNL enantioselectivity mutants
To be published
5HNH
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Crystal structure of pyrene- and phenanthrene-modified DNA in complex with the BpuJ1 endonuclease binding domain
分子名称: DNA (5'-D(*GP*(YPY)P*AP*CP*CP*CP*GP*TP*GP*GP*A)-3'), DNA (5'-D(*TP*CP*CP*AP*CP*GP*GP*GP*T*(YPY)*(YPY)*C)-3'), Restriction endonuclease R.BpuJI
著者Probst, M, Aeschimann, W, Chau, T.-T.-H, Langenegger, S.M, Stocker, A, Haener, R.
登録日2016-01-18
公開日2016-08-17
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.876 Å)
主引用文献Structural insight into DNA-assembled oligochromophores: crystallographic analysis of pyrene- and phenanthrene-modified DNA in complex with BpuJI endonuclease.
Nucleic Acids Res., 44, 2016
3IXM
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Structure of the Gly74Cys mutant of arylmalonate decarboxylase in the sulfate ion associated form
分子名称: Arylmalonate decarboxylase, SULFATE ION
著者Nakasako, M, Obata, R.
登録日2009-09-04
公開日2010-02-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Basis for Inverting the Enantioselectivity of Arylmalonate Decarboxylase Revealed by the Structural Analysis of the Gly74Cys/Cys188Ser Mutant in the Liganded Form
Biochemistry, 49, 2010
1RB8
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The phiX174 DNA binding protein J in two different capsid environments.
分子名称: 2'-DEOXYCYTIDINE-5'-MONOPHOSPHATE, Capsid protein, DNA (5'-D(P*CP*AP*AP*A)-3'), ...
著者Bernal, R.A, Hafenstein, S, Esmeralda, R, Fane, B.A, Rossmann, M.G.
登録日2003-11-03
公開日2004-04-13
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献The phiX174 Protein J Mediates DNA Packaging and Viral Attachment to Host Cells.
J.Mol.Biol., 337, 2004
6CNM
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Cryo-EM structure of the human SK4/calmodulin channel complex
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, Calmodulin-1, DODECYL-BETA-D-MALTOSIDE, ...
著者Lee, C.H, MacKinnon, R.
登録日2018-03-08
公開日2018-05-02
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Activation mechanism of a human SK-calmodulin channel complex elucidated by cryo-EM structures.
Science, 360, 2018
6COZ
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Human CLC-1 chloride ion channel, C-terminal cytosolic domain
分子名称: Chloride channel protein 1
著者Park, E, MacKinnon, R.
登録日2018-03-13
公開日2018-06-13
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (3.36 Å)
主引用文献Structure of the CLC-1 chloride channel fromHomo sapiens.
Elife, 7, 2018
6CPE
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Structure of apo, dephosphorylated Aurora A (122-403) in an active conformation
分子名称: 1-ETHOXY-2-(2-ETHOXYETHOXY)ETHANE, Aurora kinase A
著者Otten, R, Kutter, S, Buosi, V, Padua, R.A.P, Kern, D.
登録日2018-03-13
公開日2018-06-27
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Dynamics of human protein kinase Aurora A linked to drug selectivity.
Elife, 7, 2018
1A8R
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GTP CYCLOHYDROLASE I (H112S MUTANT) IN COMPLEX WITH GTP
分子名称: GTP CYCLOHYDROLASE I, GUANOSINE-5'-TRIPHOSPHATE
著者Auerbach, G, Nar, H, Bracher, A, Bacher, A, Huber, R.
登録日1998-03-27
公開日1999-05-11
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Biosynthesis of pteridines. Reaction mechanism of GTP cyclohydrolase I.
J.Mol.Biol., 326, 2003
6C9X
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THE CRYSTAL STRUCTURE OF THE alpha-Glucosidase (GH 31) FROM RUMINOCOCCUS OBEUM ATCC 29174 in complex with voglibose
分子名称: (1S,2S,3R,4S,5S)-5-[(1,3-dihydroxypropan-2-yl)amino]-1-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol, CHLORIDE ION, FORMIC ACID, ...
著者Tan, K, Tesar, C, Jedrzejczak, R, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2018-01-29
公開日2018-03-07
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.457 Å)
主引用文献THE CRYSTAL STRUCTURE OF THE alpha-Glucosidase (GH 31) FROM RUMINOCOCCUS OBEUM ATCC 29174 in complex with voglibose
To Be Published
6BP6
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Crystal structure of Commd9 COMM domain
分子名称: COMM domain-containing protein 9
著者Healy, M.D, Chandra, M, Collins, B.M, Ghai, R.
登録日2017-11-22
公開日2018-08-15
最終更新日2020-01-01
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Structural insights into the architecture and membrane interactions of the conserved COMMD proteins.
Elife, 7, 2018
6CA3
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THE CRYSTAL STRUCTURE OF THE W169Y MUTANT OF ALPHA-GLUCOSIDASE (GH 31) FROM RUMINOCOCCUS OBEUM ATCC 29174 in complex with miglitol
分子名称: (2R,3R,4R,5S)-1-(2-hydroxyethyl)-2-(hydroxymethyl)piperidine-3,4,5-triol, GLYCEROL, Glycosyl hydrolase, ...
著者Tan, K, Tesar, C, Jedrzejczak, R, Joachimiak, A, Midwest Center for Macromolecular Research (MCMR)
登録日2018-01-29
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.743 Å)
主引用文献THE CRYSTAL STRUCTURE OF THE W169Y MUTANT OF ALPHA-GLUCOSIDASE (GH 31) FROM RUMINOCOCCUS OBEUM ATCC 29174 in complex with miglitol
To Be Published
6BYA
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Crystal structure of LdBPK_091320 with inhibitor bound
分子名称: 2-[2-(3-chloro-4-methoxyphenyl)ethyl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[(2S)-2-(morpholin-4-yl)propyl]-1H-benzimidazole, UNKNOWN ATOM OR ION, Uncharacterized protein
著者Dong, A, Lin, Y.H, Loppnau, P, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Hui, R, Structural Genomics Consortium (SGC)
登録日2017-12-20
公開日2018-01-17
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献Crystal structure of LdBPK_091320.1 with with inhibitor bound
to be published
1A0D
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XYLOSE ISOMERASE FROM BACILLUS STEAROTHERMOPHILUS
分子名称: MANGANESE (II) ION, XYLOSE ISOMERASE
著者Gallay, O, Chopra, R, Conti, E, Brick, P, Blow, D.
登録日1997-11-28
公開日1998-06-03
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal Structures of Class II Xylose Isomerases from Two Thermophiles and a Hyperthermophile
To be Published
6C95
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The Human NatA (Naa10/Naa15) amino-terminal acetyltransferase complex bound to HYPK
分子名称: Huntingtin-interacting protein K, INOSITOL HEXAKISPHOSPHATE, N-alpha-acetyltransferase 10, ...
著者Gottlieb, L, Marmorstein, R.
登録日2018-01-25
公開日2018-06-06
最終更新日2021-07-21
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献Structure of Human NatA and Its Regulation by the Huntingtin Interacting Protein HYPK.
Structure, 26, 2018
6C9M
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The Human NatA (Naa10/Naa15) amino-terminal acetyltransferase complex
分子名称: INOSITOL HEXAKISPHOSPHATE, N-alpha-acetyltransferase 10, N-alpha-acetyltransferase 15, ...
著者Gottlieb, L, Marmorstein, R.
登録日2018-01-26
公開日2018-06-06
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of Human NatA and Its Regulation by the Huntingtin Interacting Protein HYPK.
Structure, 26, 2018
5HLT
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BU of 5hlt by Molmil
Crystal structure of pyrene- and phenanthrene-modified DNA in complex with the BpuJ1 endonuclease binding domain
分子名称: DNA (5'-D(*GP*YPY*TP*AP*CP*CP*CP*GP*TP*GP*GP*A)-3'), DNA (5'-D(*TP*CP*CP*AP*CP*GP*GP*GP*TP*AP*YPY*C)-3'), Restriction endonuclease R.BpuJI
著者Probst, M, Aeschimann, W, Chau, T.-T.-H, Langenegger, S.M, Stocker, A, Haener, R.
登録日2016-01-15
公開日2016-08-17
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.672 Å)
主引用文献Structural insight into DNA-assembled oligochromophores: crystallographic analysis of pyrene- and phenanthrene-modified DNA in complex with BpuJI endonuclease.
Nucleic Acids Res., 44, 2016
6BH9
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Caspase-3 Mutant - T152A
分子名称: Ac-Asp-Glu-Val-Asp-CMK, CHLORIDE ION, Caspase-3, ...
著者Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
登録日2017-10-30
公開日2018-02-21
最終更新日2018-04-25
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
6C9Z
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THE CRYSTAL STRUCTURE OF THE alpha-Glucosidase (GH 31) W169Y mutant FROM RUMINOCOCCUS OBEUM ATCC 29174 in complex with voglibose
分子名称: (1S,2S,3R,4S,5S)-5-[(1,3-dihydroxypropan-2-yl)amino]-1-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol, Glycosyl hydrolase, family 31
著者Tan, K, Tesar, C, Jedrzejczak, R, Joachimiak, A, Midwest Center for Macromolecular Research (MCMR)
登録日2018-01-29
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.101 Å)
主引用文献THE CRYSTAL STRUCTURE OF THE alpha-Glucosidase (GH 31) W169Y mutant FROM RUMINOCOCCUS OBEUM ATCC 29174 in complex with voglibose
To Be Published
6BGS
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Caspase-3 Mutant - S150Y
分子名称: Ac-Asp-Glu-Val-Asp-CMK, Caspase-3
著者Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
登録日2017-10-29
公開日2018-02-21
最終更新日2018-04-25
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
6BK8
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S. cerevisiae spliceosomal post-catalytic P complex
分子名称: GUANOSINE-5'-TRIPHOSPHATE, INOSITOL HEXAKISPHOSPHATE, Lea1, ...
著者Liu, S, Li, X, Zhou, Z.H, Zhao, R.
登録日2017-11-07
公開日2018-02-21
最終更新日2020-10-14
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Structure of the yeast spliceosomal postcatalytic P complex.
Science, 358, 2017
6AK4
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Crystal structure of human FTO in complex with small-molecule inhibitors
分子名称: (~{E})-2-cyano-~{N},~{N}-diethyl-3-[3-nitro-4,5-bis(oxidanyl)phenyl]prop-2-enamide, Alpha-ketoglutarate-dependent dioxygenase FTO,Alpha-ketoglutarate-dependent dioxygenase FTO, ZINC ION
著者Wang, Y, Cao, R, Peng, S, Zhang, W, Huang, N.
登録日2018-08-30
公開日2019-07-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Identification of entacapone as a chemical inhibitor of FTO mediating metabolic regulation through FOXO1.
Sci Transl Med, 11, 2019
6ALZ
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Crystal structure of Protein Phosphatase 1 bound to the natural inhibitor Tautomycetin
分子名称: (2Z)-2-[(1R)-3-{[(2R,3S,4R,7S,8S,11S,13R,16E)-17-ethyl-4,8-dihydroxy-3,7,11,13-tetramethyl-6,15-dioxononadeca-16,18-dien-2-yl]oxy}-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid, CHLORIDE ION, DIMETHYL SULFOXIDE, ...
著者Choy, M.S, Peti, W, Page, R.
登録日2017-08-08
公開日2017-11-29
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.208 Å)
主引用文献PP1:Tautomycetin Complex Reveals a Path toward the Development of PP1-Specific Inhibitors.
J. Am. Chem. Soc., 139, 2017
5ZVF
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Structure of [T9,K7]indolicidin, a non glycosylated analogue of indolicidin
分子名称: non glycosylated analogue of Indolicidin
著者Dwivedi, R, Aggarwal, P, Kaur, K.J, Bhavesh, N.S.
登録日2018-05-10
公開日2019-06-19
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Design of therapeutically improved analogue of the antimicrobial peptide, indolicidin, using a glycosylation strategy.
Amino Acids, 51, 2019
6APX
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Crystal structure of human dual specificity phosphatase 1 catalytic domain (C258S) as a maltose binding protein fusion in complex with the monobody YSX1
分子名称: GLYCEROL, Maltose-binding periplasmic protein,Dual specificity protein phosphatase 1, Monobody YSX1, ...
著者Gumpena, R, Lountos, G.T, Sreejith, R.K, Tropea, J.E, Cherry, S, Waugh, D.S.
登録日2017-08-18
公開日2017-11-01
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.491 Å)
主引用文献Crystal structure of the human dual specificity phosphatase 1 catalytic domain.
Protein Sci., 27, 2018

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