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PDB: 3 results

7OVD
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BU of 7ovd by Molmil
Human soluble adenylyl cyclase in complex with the inhibitor TDI10229
Descriptor: 1,2-ETHANEDIOL, 4-chloranyl-6-[1,5-dimethyl-4-(phenylmethyl)pyrazol-3-yl]pyrimidin-2-amine, ACETATE ION, ...
Authors:Steegborn, C, Quast, J.
Deposit date:2021-06-14
Release date:2021-10-06
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Discovery of TDI-10229: A Potent and Orally Bioavailable Inhibitor of Soluble Adenylyl Cyclase (sAC, ADCY10).
Acs Med.Chem.Lett., 12, 2021
4D5C
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BU of 4d5c by Molmil
tetracycline repressor class J, apo form
Descriptor: SULFATE ION, TETRACYCLINE REPRESSOR PROTEIN TETR
Authors:Palm, G.J, Quast, J, Hinrichs, W.
Deposit date:2014-11-03
Release date:2016-01-20
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Domain Movement in Tetracycline Repressor Classes
To be Published
4D5F
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BU of 4d5f by Molmil
tetracycline repressor class H, apo form
Descriptor: CHLORIDE ION, GLYCEROL, SULFATE ION, ...
Authors:Palm, G.J, Quast, J, Hinrichs, W.
Deposit date:2014-11-04
Release date:2016-01-20
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Domain Movement in Tetracycline Repressor Classes
To be Published

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