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PDB: 306 件

4PNR
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BU of 4pnr by Molmil
Crystal Structure of human Tankyrase 2 in complex with TIQ-A.
分子名称: 4H-thieno[2,3-c]isoquinolin-5-one, ETHANOL, GLYCEROL, ...
著者Qiu, W, Lam, R, Romanov, V, Gordon, R, Gebremeskel, S, Vodsedalek, J, Thompson, C, Beletskaya, I, Battaile, K.P, Pai, E.F, Chirgadze, N.Y.
登録日2014-05-24
公開日2014-10-15
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.71 Å)
主引用文献Insights into the binding of PARP inhibitors to the catalytic domain of human tankyrase-2.
Acta Crystallogr.,Sect.D, 70, 2014
4PTU
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BU of 4ptu by Molmil
Crystal Structure of anti-23F strep Fab C05 with rhamnose
分子名称: ACETATE ION, Antibody pn132p2C05, heavy chain, ...
著者Bryson, S, Risnes, L, Damgupta, S, Thomson, C.A, Smith, K, Schrader, J.W, Pai, E.F.
登録日2014-03-11
公開日2015-03-04
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.511 Å)
主引用文献Structures of Preferred Human IgV Genes-Based Protective Antibodies Identify How Conserved Residues Contact Diverse Antigens and Assign Source of Specificity to CDR3 Loop Variation.
J. Immunol., 196, 2016
4PNT
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BU of 4pnt by Molmil
Crystal Structure of human Tankyrase 2 in complex with 1,5-IQD.
分子名称: 5-hydroxyisoquinolin-1(4H)-one, Tankyrase-2, ZINC ION
著者Qiu, W, Lam, R, Romanov, V, Gordon, R, Gebremeskel, S, Vodsedalek, J, Thompson, C, Beletskaya, I, Battaile, K.P, Pai, E.F, Chirgadze, N.Y.
登録日2014-05-25
公開日2014-10-15
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Insights into the binding of PARP inhibitors to the catalytic domain of human tankyrase-2.
Acta Crystallogr.,Sect.D, 70, 2014
1E2A
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BU of 1e2a by Molmil
ENZYME IIA FROM THE LACTOSE SPECIFIC PTS FROM LACTOCOCCUS LACTIS
分子名称: ENZYME IIA, MAGNESIUM ION
著者Sliz, P, Engelmann, R, Hengstenberg, W, Pai, E.F.
登録日1997-04-25
公開日1998-04-29
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The structure of enzyme IIAlactose from Lactococcus lactis reveals a new fold and points to possible interactions of a multicomponent system.
Structure, 5, 1997
1EKJ
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BU of 1ekj by Molmil
THE X-RAY CRYSTALLOGRAPHIC STRUCTURE OF BETA CARBONIC ANHYDRASE FROM THE C3 DICOT PISUM SATIVUM
分子名称: 1,2-ETHANEDIOL, ACETATE ION, AZIDE ION, ...
著者Kimber, M.S, Pai, E.F.
登録日2000-03-08
公開日2000-06-07
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献The active site architecture of Pisum sativum beta-carbonic anhydrase is a mirror image of that of alpha-carbonic anhydrases.
EMBO J., 19, 2000
1GNQ
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BU of 1gnq by Molmil
X-RAY CRYSTAL STRUCTURE ANALYSIS OF THE CATALYTIC DOMAIN OF THE ONCOGENE PRODUCT P21H-RAS COMPLEXED WITH CAGED GTP AND MANT DGPPNHP
分子名称: C-H-RAS P21 PROTEIN, GUANOSINE 5'-TRIPHOSPHATE P3-[1-(2-NITROPHENYL)ETHYL ESTER], MAGNESIUM ION
著者Scheidig, A, Franken, S.M, Corrie, J.E.T, Reid, G.P, Wittinghofer, A, Pai, E.F, Goody, R.S.
登録日1995-05-11
公開日1995-07-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献X-ray crystal structure analysis of the catalytic domain of the oncogene product p21H-ras complexed with caged GTP and mant dGppNHp.
J.Mol.Biol., 253, 1995
1GNR
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BU of 1gnr by Molmil
X-RAY CRYSTAL STRUCTURE ANALYSIS OF THE CATALYTIC DOMAIN OF THE ONCOGENE PRODUCT P21H-RAS COMPLEXED WITH CAGED GTP AND MANT DGPPNHP
分子名称: C-H-RAS P21 PROTEIN, GUANOSINE 5'-TRIPHOSPHATE P3-[1-(2-NITROPHENYL)ETHYL ESTER], MAGNESIUM ION
著者Scheidig, A, Franken, S.M, Corrie, J.E.T, Reid, G.P, Wittinghofer, A, Pai, E.F, Goody, R.S.
登録日1995-05-11
公開日1995-07-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献X-ray crystal structure analysis of the catalytic domain of the oncogene product p21H-ras complexed with caged GTP and mant dGppNHp.
J.Mol.Biol., 253, 1995
4HHA
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BU of 4hha by Molmil
Anti-Human Cytomegalovirus (HCMV) Fab KE5 with epitope peptide AD-2S1
分子名称: Antibody KE5, CHLORIDE ION, Fab KE5, ...
著者Bryson, S, Risnes, L, Damgupta, S, Thomson, C.A, Pfoh, R, Schrader, J.W, Pai, E.F.
登録日2012-10-09
公開日2013-10-23
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structures of Preferred Human IgV Genes-Based Protective Antibodies Identify How Conserved Residues Contact Diverse Antigens and Assign Source of Specificity to CDR3 Loop Variation.
J. Immunol., 196, 2016
4HH9
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BU of 4hh9 by Molmil
Anti-Human Cytomegalovirus (HCMV) Fab KE5
分子名称: Fab KE5, heavy chain, light chain
著者Bryson, S, Risnes, L, Damgupta, S, Thomson, C.A, Pfoh, R, Schrader, J.W, Pai, E.F.
登録日2012-10-09
公開日2013-10-23
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structures of Preferred Human IgV Genes-Based Protective Antibodies Identify How Conserved Residues Contact Diverse Antigens and Assign Source of Specificity to CDR3 Loop Variation.
J. Immunol., 196, 2016
4HIJ
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BU of 4hij by Molmil
Anti-Streptococcus pneumoniae 23F Fab 023.102 with bound L-rhamnose-(1-2)-alpha-D-galactose-(3-O)-phosphate-2-glycerol
分子名称: Fab 023.102 heavy chain, Fab 023.102 light chain, GLYCEROL, ...
著者Bryson, S, Risnes, L, Damgupta, S, Thomson, C.A, Schrader, J.W, Pai, E.F.
登録日2012-10-11
公開日2013-08-28
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structures of Preferred Human IgV Genes-Based Protective Antibodies Identify How Conserved Residues Contact Diverse Antigens and Assign Source of Specificity to CDR3 Loop Variation.
J. Immunol., 196, 2016
4HIE
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BU of 4hie by Molmil
Anti-Streptococcus pneumoniae 23F Fab 023.102
分子名称: Antibody 023.102, Fab 023.102
著者Bryson, S, Risnes, L, Damgupta, S, Thomson, C.A, Schrader, J.W, Pai, E.F.
登録日2012-10-11
公開日2013-08-28
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structures of Preferred Human IgV Genes-Based Protective Antibodies Identify How Conserved Residues Contact Diverse Antigens and Assign Source of Specificity to CDR3 Loop Variation.
J. Immunol., 196, 2016
4HII
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BU of 4hii by Molmil
Anti-Streptococcus pneumoniae 23F Fab 023.102 with bound rhamnose-galactose
分子名称: Fab 023.102 heavy chain, Fab 023.102 light chain, alpha-L-rhamnopyranose-(1-2)-beta-D-galactopyranose
著者Bryson, S, Risnes, L, Damgupta, S, Thomson, C.A, Schrader, J.W, Pai, E.F.
登録日2012-10-11
公開日2013-08-28
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structures of Preferred Human IgV Genes-Based Protective Antibodies Identify How Conserved Residues Contact Diverse Antigens and Assign Source of Specificity to CDR3 Loop Variation.
J. Immunol., 196, 2016
4HKP
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BU of 4hkp by Molmil
Crystal structure of human orotidine 5'-monophosphate decarboxylase complexed with CMP-N3-oxide
分子名称: 5-hydroxycytidine 5'-(dihydrogen phosphate), GLYCEROL, N-hydroxycytidine 5'-(dihydrogen phosphate), ...
著者To, T.K, Kotra, L.P, Pai, E.F.
登録日2012-10-15
公開日2012-11-14
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Novel cytidine-based orotidine-5'-monophosphate decarboxylase inhibitors with an unusual twist.
J.Med.Chem., 55, 2012
4HMM
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BU of 4hmm by Molmil
Crystal structure of mutant rabbit PRP 121-230 (S174N)
分子名称: CHLORIDE ION, GLYCEROL, Major prion protein, ...
著者Sweeting, B, Chakrabartty, A, Pai, E.F.
登録日2012-10-18
公開日2013-05-15
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献N-Terminal Helix-Cap in alpha-Helix 2 Modulates beta-State Misfolding in Rabbit and Hamster Prion Proteins.
Plos One, 8, 2013
4HLS
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BU of 4hls by Molmil
Crystal structure of mutant rabbit PRP 121-230 (S170N)
分子名称: CHLORIDE ION, GLYCEROL, Major prion protein, ...
著者Sweeting, B, Chakrabartty, A, Pai, E.F.
登録日2012-10-17
公開日2013-05-15
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献N-Terminal Helix-Cap in alpha-Helix 2 Modulates beta-State Misfolding in Rabbit and Hamster Prion Proteins.
Plos One, 8, 2013
4HIB
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BU of 4hib by Molmil
Crystal structure of human orotidine 5'-monophosphate decarboxylase complexed with CMP-N4-OH
分子名称: CHLORIDE ION, GLYCEROL, N-hydroxycytidine 5'-(dihydrogen phosphate), ...
著者To, T.K, Kotra, L.P, Pai, E.F.
登録日2012-10-11
公開日2012-11-14
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Novel cytidine-based orotidine-5'-monophosphate decarboxylase inhibitors with an unusual twist.
J.Med.Chem., 55, 2012
4HMR
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BU of 4hmr by Molmil
Crystal structure of mutant rabbit PRP 121-230 (S170N/S174N)
分子名称: CHLORIDE ION, GLYCEROL, Major prion protein, ...
著者Sweeting, B, Chakrabartty, A, Pai, E.F.
登録日2012-10-18
公開日2013-05-15
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献N-Terminal Helix-Cap in alpha-Helix 2 Modulates beta-State Misfolding in Rabbit and Hamster Prion Proteins.
Plos One, 8, 2013
4HIH
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BU of 4hih by Molmil
Anti-Streptococcus pneumoniae 23F Fab 023.102 with bound rhamnose.
分子名称: Antibody 023.102, Fab 023.102, alpha-L-rhamnopyranose
著者Bryson, S, Risnes, L, Damgupta, S, Thomson, C.A, Schrader, J.W, Pai, E.F.
登録日2012-10-11
公開日2013-08-28
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structures of Preferred Human IgV Genes-Based Protective Antibodies Identify How Conserved Residues Contact Diverse Antigens and Assign Source of Specificity to CDR3 Loop Variation.
J. Immunol., 196, 2016
4J4Q
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BU of 4j4q by Molmil
Crystal structure of active conformation of GPCR opsin stabilized by octylglucoside
分子名称: ACETATE ION, Guanine nucleotide-binding protein G(t) subunit alpha-1, PALMITIC ACID, ...
著者Park, J.H, Morizumi, T, Li, Y, Hong, J.E, Pai, E.F, Hofmann, K.P, Choe, H.W, Ernst, O.P.
登録日2013-02-07
公開日2013-10-30
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Opsin, a structural model for olfactory receptors?
Angew.Chem.Int.Ed.Engl., 52, 2013
2ZZ7
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BU of 2zz7 by Molmil
Orotidine Monophosphate Decarboxylase K72A mutant complexed with BMP (produced from 6-Iodo-UMP)
分子名称: 6-HYDROXYURIDINE-5'-PHOSPHATE, GLYCEROL, Orotidine 5'-phosphate decarboxylase
著者Fujihashi, M, Pai, E.F.
登録日2009-02-05
公開日2009-03-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.58 Å)
主引用文献Structural characterization of the molecular events during a slow substrate-product transition in orotidine 5'-monophosphate decarboxylase
J.Mol.Biol., 387, 2009
2ZZ3
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BU of 2zz3 by Molmil
Covalent complex of orotidine monophosphate decarboxylase D70A mutant from M. thermoautotrophicus with 6-cyano-UMP
分子名称: 6-cyanouridine 5'-phosphate, GLYCEROL, Orotidine 5'-phosphate decarboxylase
著者Fujihashi, M, Pai, E.F.
登録日2009-02-05
公開日2009-03-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural characterization of the molecular events during a slow substrate-product transition in orotidine 5'-monophosphate decarboxylase
J.Mol.Biol., 387, 2009
2ZZ5
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BU of 2zz5 by Molmil
Orotidine Monophosphate Deacarboxylase D70A/K72A double mutant from M. thermoautotrophicum complexed with 6- cyano-UMP
分子名称: 6-cyanouridine 5'-phosphate, Orotidine 5'-phosphate decarboxylase
著者Fujihashi, M, Pai, E.F.
登録日2009-02-05
公開日2009-03-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Structural characterization of the molecular events during a slow substrate-product transition in orotidine 5'-monophosphate decarboxylase
J.Mol.Biol., 387, 2009
2ZZ4
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BU of 2zz4 by Molmil
Covalent complex of orotidine monophosphate decarboxylase D75N mutant from M. thermoautotrophicum with 6-cyano-UMP
分子名称: 6-cyanouridine 5'-phosphate, GLYCEROL, Orotidine 5'-phosphate decarboxylase
著者Fujihashi, M, Pai, E.F.
登録日2009-02-05
公開日2009-03-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Structural characterization of the molecular events during a slow substrate-product transition in orotidine 5'-monophosphate decarboxylase
J.Mol.Biol., 387, 2009
2ZZ1
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BU of 2zz1 by Molmil
Snapshot of the reaction from 6-CN-UMP to BMP catalyzed by Orotidine Monophosphate Deacarboxylase from M. thermoautotrophicum
分子名称: 6-HYDROXYURIDINE-5'-PHOSPHATE, 6-cyanouridine 5'-phosphate, GLYCEROL, ...
著者Fujihashi, M, Pai, E.F.
登録日2009-02-05
公開日2009-03-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.57 Å)
主引用文献Structural characterization of the molecular events during a slow substrate-product transition in orotidine 5'-monophosphate decarboxylase
J.Mol.Biol., 387, 2009
2ZZ2
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BU of 2zz2 by Molmil
Orotidine Monophosphate Decarboxylase K72A mutant from M. thermoautotrophicum complexed with 6-cyano-UMP
分子名称: 6-cyanouridine 5'-phosphate, GLYCEROL, Orotidine 5'-phosphate decarboxylase
著者Fujihashi, M, Pai, E.F.
登録日2009-02-05
公開日2009-03-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Structural characterization of the molecular events during a slow substrate-product transition in orotidine 5'-monophosphate decarboxylase
J.Mol.Biol., 387, 2009

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