1IUS
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![BU of 1ius by Molmil](/molmil-images/mine/1ius) | P-HYDROXYBENZOATE HYDROXYLASE COMPLEXED WITH 4-AMINOBENZOATE AT PH 5.0 | 分子名称: | 4-AMINOBENZOIC ACID, FLAVIN-ADENINE DINUCLEOTIDE, P-HYDROXYBENZOATE HYDROXYLASE | 著者 | Gatti, D.L, Entsch, B, Ballou, D.P, Ludwig, M.L. | 登録日 | 1995-11-22 | 公開日 | 1996-04-03 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | pH-dependent structural changes in the active site of p-hydroxybenzoate hydroxylase point to the importance of proton and water movements during catalysis. Biochemistry, 35, 1996
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8BOS
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6INE
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![BU of 6ine by Molmil](/molmil-images/mine/6ine) | Crystal Structure of human ASH1L-MRG15 complex | 分子名称: | GLYCEROL, Histone-lysine N-methyltransferase ASH1L, Mortality factor 4-like protein 1, ... | 著者 | Hou, P, Huang, C, Liu, C.P, Yu, T, Yin, Y, Zhu, B, Xu, R.M. | 登録日 | 2018-10-25 | 公開日 | 2019-03-20 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural Insights into Stimulation of Ash1L's H3K36 Methyltransferase Activity through Mrg15 Binding. Structure, 27, 2019
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5DS6
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![BU of 5ds6 by Molmil](/molmil-images/mine/5ds6) | Crystal structure the Escherichia coli Cas1-Cas2 complex bound to protospacer DNA with splayed ends | 分子名称: | CRISPR-associated endonuclease Cas1, CRISPR-associated endoribonuclease Cas2, DNA (28-MER), ... | 著者 | Nunez, J.K, Harrington, L.B, Kranzusch, P.J, Engelman, A.N, Doudna, J.A. | 登録日 | 2015-09-16 | 公開日 | 2015-10-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.352 Å) | 主引用文献 | Foreign DNA capture during CRISPR-Cas adaptive immunity. Nature, 527, 2015
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6L50
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![BU of 6l50 by Molmil](/molmil-images/mine/6l50) | Crystal structure of Zika NS2B-NS3 protease with compound 16 | 分子名称: | 2-sulfanylidene-1,3-thiazolidin-4-one, NS3 protease, Serine protease subunit NS2B | 著者 | Quek, J.P. | 登録日 | 2019-10-21 | 公開日 | 2020-07-15 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Identification and structural characterization of small molecule fragments targeting Zika virus NS2B-NS3 protease. Antiviral Res., 175, 2020
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8OKU
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![BU of 8oku by Molmil](/molmil-images/mine/8oku) | Salt-Inducible Kinase 3 in complex with an inhibitor | 分子名称: | Serine/threonine-protein kinase SIK3, ~{N}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamide | 著者 | Flower, T.G, Leonard, P.M, Lamers, M.B.A.C, Mollat, P. | 登録日 | 2023-03-29 | 公開日 | 2024-01-10 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Optimization of Selectivity and Pharmacokinetic Properties of Salt-Inducible Kinase Inhibitors that Led to the Discovery of Pan-SIK Inhibitor GLPG3312. J.Med.Chem., 67, 2024
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4K9B
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![BU of 4k9b by Molmil](/molmil-images/mine/4k9b) | Structure of Ternary Complex of cGAS with dsDNA and Bound c[G(2 ,5 )pA(3 ,5 )p] | 分子名称: | ADENOSINE MONOPHOSPHATE, Cyclic GMP-AMP synthase, DNA-F, ... | 著者 | Gao, P, Wu, Y, Patel, D.J. | 登録日 | 2013-04-19 | 公開日 | 2013-05-15 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.26 Å) | 主引用文献 | Cyclic [G(2',5')pA(3',5')p] is the metazoan second messenger produced by DNA-activated cyclic GMP-AMP synthase. Cell(Cambridge,Mass.), 153, 2013
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6WKL
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6WKM
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8BTL
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![BU of 8btl by Molmil](/molmil-images/mine/8btl) | Crystal structure of a complex between the E2 conjugating enzyme UBE2A and the E3 ligase module from UBR4 | 分子名称: | Ubiquitin conjugating enzyme E2 A, ZINC ION, cDNA FLJ12511 fis, ... | 著者 | Virdee, S, Mabbitt, P.D, Barnsby-Greer, L. | 登録日 | 2022-11-29 | 公開日 | 2023-12-13 | 最終更新日 | 2024-04-17 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | UBE2A and UBE2B are recruited by an atypical E3 ligase module in UBR4. Nat.Struct.Mol.Biol., 31, 2024
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8BSY
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5DVP
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![BU of 5dvp by Molmil](/molmil-images/mine/5dvp) | Crystal structure of Mycobacterium tuberculosis L,D-transpeptidase 2 with Doripenem adduct | 分子名称: | (2S,3R,4S)-2-[(2S,3R)-3-hydroxy-1-oxobutan-2-yl]-3-methyl-4-({(3S,5S)-5-[(sulfamoylamino)methyl]pyrrolidin-3-yl}sulfanyl)-3,4-dihydro-2H-pyrrole-5-carboxylic acid, L,D-transpeptidase 2, PHOSPHONOACETALDEHYDE, ... | 著者 | Kumar, P, Lamichhane, G. | 登録日 | 2015-09-21 | 公開日 | 2016-09-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | Non-classical transpeptidases yield insight into new antibacterials. Nat. Chem. Biol., 13, 2017
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6WJL
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![BU of 6wjl by Molmil](/molmil-images/mine/6wjl) | Crystal structure of Glypican-2 core protein in complex with D3 Fab | 分子名称: | D3 Fab Heavy chain, D3 Fab Light Chain, Glypican-2, ... | 著者 | Raman, S, Maris, J.M, Bosse, K.R, Julien, J.P. | 登録日 | 2020-04-14 | 公開日 | 2021-04-21 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (3.3 Å) | 主引用文献 | A GPC2 antibody-drug conjugate is efficacious against neuroblastoma and small-cell lung cancer via binding a conformational epitope. Cell Rep Med, 2, 2021
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8BSX
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8BSW
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7RU0
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![BU of 7ru0 by Molmil](/molmil-images/mine/7ru0) | SthK R120A Open State 1 | 分子名称: | ADENOSINE-3',5'-CYCLIC-MONOPHOSPHATE, SthK | 著者 | Gao, X, Nimigean, C, Schmidpeter, P. | 登録日 | 2021-08-16 | 公開日 | 2022-11-23 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (4.3 Å) | 主引用文献 | Gating intermediates reveal inhibitory role of the voltage sensor in a cyclic nucleotide-modulated ion channel. Nat Commun, 13, 2022
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6I60
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4PEF
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![BU of 4pef by Molmil](/molmil-images/mine/4pef) | Dbr1 in complex with sulfate | 分子名称: | GLYCEROL, MANGANESE (II) ION, RNA lariat debranching enzyme, ... | 著者 | Montemayor, E.J, Katolik, A, Clark, N.E, Taylor, A.B, Schuermann, J.P, Combs, D.J, Johnsson, R, Holloway, S.P, Stevens, S.W, Damha, M.J, Hart, P.J. | 登録日 | 2014-04-23 | 公開日 | 2014-08-27 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | Structural basis of lariat RNA recognition by the intron debranching enzyme Dbr1. Nucleic Acids Res., 42, 2014
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8BSV
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1E70
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![BU of 1e70 by Molmil](/molmil-images/mine/1e70) | 2-F-glucosylated MYROSINASE FROM SINAPIS ALBA | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-deoxy-2-fluoro-alpha-D-glucopyranose, ... | 著者 | Burmeister, W.P. | 登録日 | 2000-08-23 | 公開日 | 2001-01-05 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | High Resolution X-Ray Crystallography Shows that Ascorbate is a Cofactor for Myrosinase and Substitutes for the Function of the Catalytic Base J.Biol.Chem., 275, 2000
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4PG9
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![BU of 4pg9 by Molmil](/molmil-images/mine/4pg9) | MHC Class I in complex with Sendai virus nucleoprotein peptide FAPGNYPAL | 分子名称: | Beta-2-microglobulin, GLYCEROL, H-2 class I histocompatibility antigen, ... | 著者 | Celie, P, Joosten, R.P, Perrakis, A, Neefjes, J. | 登録日 | 2014-05-01 | 公開日 | 2015-01-07 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | The first step of peptide selection in antigen presentation by MHC class I molecules. Proc.Natl.Acad.Sci.USA, 112, 2015
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5E38
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![BU of 5e38 by Molmil](/molmil-images/mine/5e38) | Structural basis of mapping the spontaneous mutations with 5-flourouracil in uracil phosphoribosyltransferase from Mycobacterium tuberculosis | 分子名称: | Uracil phosphoribosyltransferase | 著者 | Ghode, P, Jobichen, C, Ramachandran, S, Bifani, P, Sivaraman, J. | 登録日 | 2015-10-02 | 公開日 | 2015-10-21 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural basis of mapping the spontaneous mutations with 5-flurouracil in uracil phosphoribosyltransferase from Mycobacterium tuberculosis Biochem.Biophys.Res.Commun., 467, 2015
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6LD7
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6E0E
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![BU of 6e0e by Molmil](/molmil-images/mine/6e0e) | Crystal structure of Glucokinase in complex with compound 6 | 分子名称: | 2-({2-[(4-methyl-1,3-thiazol-2-yl)amino]pyridin-3-yl}oxy)benzonitrile, Glucokinase, alpha-D-glucopyranose | 著者 | Hinklin, R.J, Baer, B.R, Boyd, S.A, Chicarelli, M.D, Condroski, K.R, DeWolf, W.E, Fischer, J, Frank, M, Hingorani, G.P, Lee, P.A, Neitzel, N.A, Pratt, S.A, Singh, A, Sullivan, F.X, Turner, T, Voegtli, W.C, Wallace, E.M, Williams, L, Aicher, T.D. | 登録日 | 2018-07-06 | 公開日 | 2019-07-10 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Discovery and preclinical development of AR453588 as an anti-diabetic glucokinase activator. Bioorg.Med.Chem., 28, 2020
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8BV8
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![BU of 8bv8 by Molmil](/molmil-images/mine/8bv8) | Crystal structure of the phage Mu protein Mom inactive mutant S124A | 分子名称: | Methylcarbamoylase mom | 著者 | Silva, R.M.B, Slyvka, A, Lee, Y.J, Guan, C, Lund, S.R, Raleigh, E.A, Skowronek, K, Bochtler, M, Weigele, P.R. | 登録日 | 2022-12-08 | 公開日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Crystal structure of the phage Mu protein Mom catalytic mutant S124A To Be Published
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