2W2P
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![BU of 2w2p by Molmil](/molmil-images/mine/2w2p) | PCSK9-deltaC D374A mutant bound to WT EGF-A of LDLR | 分子名称: | CALCIUM ION, LOW-DENSITY LIPOPROTEIN RECEPTOR, PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9 | 著者 | Bottomley, M.J, Cirillo, A, Orsatti, L, Ruggeri, L, Fisher, T.S, Santoro, J.C, Cummings, R.T, Cubbon, R.M, Lo Surdo, P, Calzetta, A, Noto, A, Baysarowich, J, Mattu, M, Talamo, F, De Francesco, R, Sparrow, C.P, Sitlani, A, Carfi, A. | 登録日 | 2008-11-03 | 公開日 | 2008-11-18 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.62 Å) | 主引用文献 | Structural and Biochemical Characterization of the Wild Type Pcsk9/Egf-Ab Complex and Natural Fh Mutants. J.Biol.Chem., 284, 2009
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1DU1
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1XWH
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![BU of 1xwh by Molmil](/molmil-images/mine/1xwh) | NMR structure of the first phd finger of autoimmune regulator protein (AIRE1): insights into apeced | 分子名称: | Autoimmune regulator, ZINC ION | 著者 | Bottomley, M.J, Stier, G, Krasotkina, J, Legube, G, Simon, B, Akhtar, A, Sattler, M, Musco, G. | 登録日 | 2004-11-01 | 公開日 | 2005-01-25 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR structure of the first PHD finger of autoimmune regulator protein (AIRE1). Insights into autoimmune polyendocrinopathy-candidiasis-ectodermal dystrophy (APECED) disease J.Biol.Chem., 280, 2005
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1H5P
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![BU of 1h5p by Molmil](/molmil-images/mine/1h5p) | Solution structure of the human Sp100b SAND domain by heteronuclear NMR. | 分子名称: | NUCLEAR AUTOANTIGEN SP100-B | 著者 | Bottomley, M.J, Liu, Z, Collard, M.W, Huggenvik, J.I, Gibson, T.J, Sattler, M. | 登録日 | 2001-05-24 | 公開日 | 2001-07-06 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | The SAND domain structure defines a novel DNA-binding fold in transcriptional regulation. Nat. Struct. Biol., 8, 2001
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6S7X
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4BY2
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![BU of 4by2 by Molmil](/molmil-images/mine/4by2) | SAS-4 (dCPAP) TCP domain in complex with a Proline Rich Motif of Ana2 (dSTIL) of Drosophila Melanogaster | 分子名称: | 1,2-ETHANEDIOL, ANASTRAL SPINDLE 2, SAS 4 | 著者 | Cottee, M.A, Muschalik, N, Wong, Y.L, Johnson, C.M, Johnson, S, Andreeva, A, Oegema, K, Lea, S.M, Raff, J.W, van Breugel, M. | 登録日 | 2013-07-17 | 公開日 | 2013-09-18 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.57 Å) | 主引用文献 | Crystal structures of the CPAP/STIL complex reveal its role in centriole assembly and human microcephaly. Elife, 2, 2013
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6S7Y
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3IF9
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![BU of 3if9 by Molmil](/molmil-images/mine/3if9) | Crystal structure of Glycine Oxidase G51S/A54R/H244A mutant in complex with inhibitor glycolate | 分子名称: | FLAVIN-ADENINE DINUCLEOTIDE, GLYCOLIC ACID, Glycine oxidase | 著者 | Pedotti, M, Rosini, E, Molla, G, Moschetti, T, Vallone, B, Savino, C, Pollegioni, L. | 登録日 | 2009-07-24 | 公開日 | 2009-10-27 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Glyphosate resistance by engineering the flavoenzyme glycine oxidase. J.Biol.Chem., 284, 2009
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5AL6
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5AL7
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1S8J
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![BU of 1s8j by Molmil](/molmil-images/mine/1s8j) | Nitrate-bound D85S mutant of bacteriorhodopsin | 分子名称: | 1-[2,6,10.14-TETRAMETHYL-HEXADECAN-16-YL]-2-[2,10,14-TRIMETHYLHEXADECAN-16-YL]GLYCEROL, Bacteriorhodopsin precursor, NITRATE ION, ... | 著者 | Facciotti, M.T, Cheung, V.S, Lunde, C.S, Rouhani, S, Baliga, N.S, Glaeser, R.M. | 登録日 | 2004-02-02 | 公開日 | 2004-06-08 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Specificity of anion binding in the substrate pocket of bacteriorhodopsin. Biochemistry, 43, 2004
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1S8L
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![BU of 1s8l by Molmil](/molmil-images/mine/1s8l) | Anion-free form of the D85S mutant of bacteriorhodopsin from crystals grown in the presence of halide | 分子名称: | 1-[2,6,10.14-TETRAMETHYL-HEXADECAN-16-YL]-2-[2,10,14-TRIMETHYLHEXADECAN-16-YL]GLYCEROL, Bacteriorhodopsin precursor, RETINAL | 著者 | Facciotti, M.T, Cheung, V.S, Lunde, C.S, Rouhani, S, Baliga, N.S, Glaeser, R.M. | 登録日 | 2004-02-02 | 公開日 | 2004-06-08 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Specificity of anion binding in the substrate pocket of bacteriorhodopsin. Biochemistry, 43, 2004
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2VQQ
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![BU of 2vqq by Molmil](/molmil-images/mine/2vqq) | Structure of HDAC4 catalytic domain (a double cysteine-to-alanine mutant) bound to a trifluoromethylketone inhbitor | 分子名称: | 2,2,2-TRIFLUORO-1-{5-[(3-PHENYL-5,6-DIHYDROIMIDAZO[1,2-A]PYRAZIN-7(8H)-YL)CARBONYL]THIOPHEN-2-YL}ETHANE-1,1-DIOL, HISTONE DEACETYLASE 4, POTASSIUM ION, ... | 著者 | Bottomley, M.J, Lo Surdo, P, Di Giovine, P, Cirillo, A, Scarpelli, R, Ferrigno, F, Jones, P, Neddermann, P, De Francesco, R, Steinkuhler, C, Gallinari, P, Carfi, A. | 登録日 | 2008-03-18 | 公開日 | 2008-07-08 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural and Functional Analysis of the Human Hdac4 Catalytic Domain Reveals a Regulatory Zinc-Binding Domain. J.Biol.Chem., 283, 2008
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2VQO
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![BU of 2vqo by Molmil](/molmil-images/mine/2vqo) | Structure of HDAC4 catalytic domain with a gain-of-function muation bound to a trifluoromethylketone inhbitor | 分子名称: | 2,2,2-TRIFLUORO-1-{5-[(3-PHENYL-5,6-DIHYDROIMIDAZO[1,2-A]PYRAZIN-7(8H)-YL)CARBONYL]THIOPHEN-2-YL}ETHANE-1,1-DIOL, HISTONE DEACETYLASE 4, POTASSIUM ION, ... | 著者 | Bottomley, M.J, Lo Surdo, P, Di Giovine, P, Cirillo, A, Scarpelli, R, Ferrigno, F, Jones, P, Neddermann, P, De Francesco, R, Steinkuhler, C, Gallinari, P, Carfi, A. | 登録日 | 2008-03-18 | 公開日 | 2008-07-08 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Structural and Functional Analysis of the Human Hdac4 Catalytic Domain Reveals a Regulatory Zinc-Binding Domain. J.Biol.Chem., 283, 2008
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2VQV
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![BU of 2vqv by Molmil](/molmil-images/mine/2vqv) | Structure of HDAC4 catalytic domain with a gain-of-function mutation bound to a hydroxamic acid inhibitor | 分子名称: | HISTONE DEACETYLASE 4, N-hydroxy-5-[(3-phenyl-5,6-dihydroimidazo[1,2-a]pyrazin-7(8H)-yl)carbonyl]thiophene-2-carboxamide, POTASSIUM ION, ... | 著者 | Bottomley, M.J, Lo Surdo, P, Di Giovine, P, Cirillo, A, Scarpelli, R, Ferrigno, F, Jones, P, Neddermann, P, De Francesco, R, Steinkuhler, C, Gallinari, P, Carfi, A. | 登録日 | 2008-03-19 | 公開日 | 2008-07-22 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3.3 Å) | 主引用文献 | Structural and Functional Analysis of the Human Hdac4 Catalytic Domain Reveals a Regulatory Structural Zinc-Binding Domain. J.Biol.Chem., 283, 2008
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3U3F
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![BU of 3u3f by Molmil](/molmil-images/mine/3u3f) | Structural basis for the interaction of Pyk2 PAT domain with paxillin LD motifs | 分子名称: | Paxillin LD2 peptide, Protein-tyrosine kinase 2-beta | 著者 | Vanarotti, M, Miller, D.J, Guibao, C.C, Zheng, J.J. | 登録日 | 2011-10-05 | 公開日 | 2012-10-24 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.101 Å) | 主引用文献 | Structural and Mechanistic Insights into the Interaction between Pyk2 and Paxillin LD Motifs. J.Mol.Biol., 426, 2014
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1ALG
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![BU of 1alg by Molmil](/molmil-images/mine/1alg) | SOLUTION STRUCTURE OF AN HGR INHIBITOR, NMR, 10 STRUCTURES | 分子名称: | P11 | 著者 | Schott, M.K, Nordhoff, A, Becker, K, Kalbitzer, H.R, Schirmer, R.H. | 登録日 | 1997-06-03 | 公開日 | 1997-10-15 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Denaturation and reactivation of dimeric human glutathione reductase--an assay for folding inhibitors. Eur.J.Biochem., 245, 1997
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2LK4
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2UV0
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![BU of 2uv0 by Molmil](/molmil-images/mine/2uv0) | Structure of the P. aeruginosa LasR ligand-binding domain bound to its autoinducer | 分子名称: | N-3-OXO-DODECANOYL-L-HOMOSERINE LACTONE, TRANSCRIPTIONAL ACTIVATOR PROTEIN LASR | 著者 | Bottomley, M.J, Muraglia, E, Bazzo, R, Carfi, A. | 登録日 | 2007-03-08 | 公開日 | 2007-03-27 | 最終更新日 | 2019-07-24 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Molecular Insights Into Quorum Sensing in the Human Pathogen Pseudomonas Aeruginosa from the Structure of the Virulence Regulator Lasr Bound to its Autoinducer. J.Biol.Chem., 282, 2007
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2VQW
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![BU of 2vqw by Molmil](/molmil-images/mine/2vqw) | Structure of inhibitor-free HDAC4 catalytic domain (with gain-of- function mutation His332Tyr) | 分子名称: | HISTONE DEACETYLASE 4, POTASSIUM ION, ZINC ION | 著者 | Bottomley, M.J, Lo Surdo, P, Di Giovine, P, Cirillo, A, Scarpelli, R, Ferrigno, F, Jones, P, Neddermann, P, De Francesco, R, Steinkuhler, C, Gallinari, P, Carfi, A. | 登録日 | 2008-03-19 | 公開日 | 2008-08-05 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural and Functional Analysis of the Human Hdac4 Catalytic Domain Reveals a Regulatory Structural Zinc-Binding Domain. J.Biol.Chem., 283, 2008
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2VQM
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![BU of 2vqm by Molmil](/molmil-images/mine/2vqm) | Structure of HDAC4 catalytic domain bound to a hydroxamic acid inhbitor | 分子名称: | HISTONE DEACETYLASE 4, N-hydroxy-5-[(3-phenyl-5,6-dihydroimidazo[1,2-a]pyrazin-7(8H)-yl)carbonyl]thiophene-2-carboxamide, POTASSIUM ION, ... | 著者 | Bottomley, M.J, Lo Surdo, P, Di Giovine, P, Cirillo, A, Scarpelli, R, Ferrigno, F, Jones, P, Neddermann, P, De Francesco, R, Steinkuhler, C, Gallinari, P, Carfi, A. | 登録日 | 2008-03-17 | 公開日 | 2008-07-08 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural and Functional Analysis of the Human Hdac4 Catalytic Domain Reveals a Regulatory Zinc-Binding Domain. J.Biol.Chem., 283, 2008
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2VQJ
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![BU of 2vqj by Molmil](/molmil-images/mine/2vqj) | Structure of HDAC4 catalytic domain bound to a trifluoromethylketone inhbitor | 分子名称: | 1,4-DIETHYLENE DIOXIDE, 2,2,2-TRIFLUORO-1-{5-[(3-PHENYL-5,6-DIHYDROIMIDAZO[1,2-A]PYRAZIN-7(8H)-YL)CARBONYL]THIOPHEN-2-YL}ETHANE-1,1-DIOL, HISTONE DEACETYLASE 4, ... | 著者 | Bottomley, M.J, Lo Surdo, P, Di Giovine, P, Cirillo, A, Scarpelli, R, Ferrigno, F, Jones, P, Neddermann, P, De Francesco, R, Steinkuhler, C, Gallinari, P, Carfi, A. | 登録日 | 2008-03-17 | 公開日 | 2008-07-08 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural and Functional Analysis of the Human Hdac4 Catalytic Domain Reveals a Regulatory Zinc-Binding Domain. J.Biol.Chem., 283, 2008
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1OCA
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![BU of 1oca by Molmil](/molmil-images/mine/1oca) | HUMAN CYCLOPHILIN A, UNLIGATED, NMR, 20 STRUCTURES | 分子名称: | CYCLOPHILIN A | 著者 | Ottiger, M, Zerbe, O, Guntert, P, Wuthrich, K. | 登録日 | 1997-07-07 | 公開日 | 1997-11-19 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | The NMR solution conformation of unligated human cyclophilin A. J.Mol.Biol., 272, 1997
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7NLH
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1ERD
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![BU of 1erd by Molmil](/molmil-images/mine/1erd) | THE NMR SOLUTION STRUCTURE OF THE PHEROMONE ER-2 FROM THE CILIATED PROTOZOAN EUPLOTES RAIKOVI | 分子名称: | PHEROMONE ER-2 | 著者 | Ottiger, M, Szyperski, T, Luginbuhl, P, Ortenzi, C, Luporini, P, Bradshaw, R.A, Wuthrich, K. | 登録日 | 1994-02-14 | 公開日 | 1994-10-15 | 最終更新日 | 2022-02-16 | 実験手法 | SOLUTION NMR | 主引用文献 | The NMR solution structure of the pheromone Er-2 from the ciliated protozoan Euplotes raikovi. Protein Sci., 3, 1994
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