4MC1
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![BU of 4mc1 by Molmil](/molmil-images/mine/4mc1) | HIV protease in complex with SA526P | 分子名称: | (3S)-tetrahydrofuran-3-yl {(2S,3R)-4-[(4S)-4-tert-butyl-7-fluoro-1,1-dioxido-4,5-dihydro-1,2-benzothiazepin-2(3H)-yl]-3-hydroxy-1-phenylbutan-2-yl}carbamate, CHLORIDE ION, Protease | 著者 | Ganguly, A.K, Alluri, S.S, Wang, C, Antropow, A, White, A, Caroccia, D, Biswas, D, Kang, E, Zhang, L, Carroll, S.S, Burlein, C, Munshi, V, Orth, P, Strickland, C. | 登録日 | 2013-08-21 | 公開日 | 2014-04-02 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.39 Å) | 主引用文献 | Structural Optimization of Cyclic Sulfonamide based Novel HIV-1 Protease Inhibitors to Pico Molar Affinities guided by X-ray Crystallographic Analysis Tetrahedron, 2014
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3EDZ
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![BU of 3edz by Molmil](/molmil-images/mine/3edz) | Crystal structure of catalytic domain of TACE with hydroxamate inhibitor | 分子名称: | ADAM 17, CITRIC ACID, N-{(2R)-2-[2-(hydroxyamino)-2-oxoethyl]-4-methylpentanoyl}-3-methyl-L-valyl-N-(2-aminoethyl)-L-alaninamide, ... | 著者 | Mazzola, R.D, Zhu, Z, Sinning, L, McKittrick, B, Lavey, B, Spitler, J, Kozlowski, J, Neng-Yang, S, Zhou, G, Guo, Z, Orth, P, Madison, V, Sun, J, Lundell, D, Niu, X. | 登録日 | 2008-09-03 | 公開日 | 2008-09-23 | 最終更新日 | 2021-10-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Discovery of novel hydroxamates as highly potent tumor necrosis factor-alpha converting enzyme inhibitors. Part II: optimization of the S3' pocket. Bioorg.Med.Chem.Lett., 18, 2008
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3JZI
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![BU of 3jzi by Molmil](/molmil-images/mine/3jzi) | Crystal structure of biotin carboxylase from E. Coli in complex with benzimidazole series | 分子名称: | 7-amino-2-[(2-chlorobenzyl)amino]-1-{[(1S,2S)-2-hydroxycycloheptyl]methyl}-1H-benzimidazole-5-carboxamide, Biotin carboxylase | 著者 | Cheng, C, Shipps, G.W, Yang, Z, Sun, B, Kawahata, N, Soucy, K, Soriano, A, Orth, P, Xiao, L, Mann, P, Black, T. | 登録日 | 2009-09-23 | 公開日 | 2009-11-03 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Discovery and optimization of antibacterial AccC inhibitors. Bioorg.Med.Chem.Lett., 19, 2009
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1CH0
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![BU of 1ch0 by Molmil](/molmil-images/mine/1ch0) | RNASE T1 VARIANT WITH ALTERED GUANINE BINDING SEGMENT | 分子名称: | CALCIUM ION, CHLORIDE ION, GUANOSINE-2'-MONOPHOSPHATE, ... | 著者 | Hoeschler, K, Hoier, H, Orth, P, Hubner, B, Saenger, W, Hahn, U. | 登録日 | 1999-03-30 | 公開日 | 1999-12-22 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural analysis of an RNase T1 variant with an altered guanine binding segment. J.Mol.Biol., 294, 1999
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1A9E
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![BU of 1a9e by Molmil](/molmil-images/mine/1a9e) | DECAMER-LIKE CONFORMATION OF A NANO-PEPTIDE BOUND TO HLA-B3501 DUE TO NONSTANDARD POSITIONING OF THE C-TERMINUS | 分子名称: | BETA-2-MICROGLOBULIN, HLA CLASS I HISTOCOMPATIBILITY ANTIGEN, B-35 B*3501 (ALPHA CHAIN), ... | 著者 | Menssen, R, Orth, P, Ziegler, A, Saenger, W. | 登録日 | 1998-04-05 | 公開日 | 1998-10-21 | 最終更新日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Decamer-like conformation of a nona-peptide bound to HLA-B*3501 due to non-standard positioning of the C terminus. J.Mol.Biol., 285, 1999
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1A9B
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![BU of 1a9b by Molmil](/molmil-images/mine/1a9b) | DECAMER-LIKE CONFORMATION OF A NANO-PEPTIDE BOUND TO HLA-B3501 DUE TO NONSTANDARD POSITIONING OF THE C-TERMINUS | 分子名称: | BETA-2-MICROGLOBULIN, HLA CLASS I HISTOCOMPATIBILITY ANTIGEN, B-35 B*3501 (ALPHA CHAIN), ... | 著者 | Menssen, R, Orth, P, Ziegler, A, Saenger, W. | 登録日 | 1998-04-03 | 公開日 | 1998-10-21 | 最終更新日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Decamer-like conformation of a nona-peptide bound to HLA-B*3501 due to non-standard positioning of the C terminus. J.Mol.Biol., 285, 1999
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1CG9
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![BU of 1cg9 by Molmil](/molmil-images/mine/1cg9) | COMPLEX RECOGNITION OF THE SUPERTYPIC BW6-DETERMINANT ON HLA-B AND-C MOLECULES BY THE MONOCLONAL ANTIBODY SFR8-B6 | 分子名称: | PROTEIN (BETA-2-MICROGLOBULIN), PROTEIN (EBNA-6 NUCLEAR PROTEIN (EBNA-3C) (EBNA-4B)), PROTEIN (HLA CLASS I HISTOCOMPATIBILITY ANTIGEN, ... | 著者 | Menssen, R, Orth, P, Ziegler, A, Saenger, W. | 登録日 | 1999-03-25 | 公開日 | 2003-11-18 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Complex Recognition of the Supertypic Bw6-Determinant on HLA-B and-C Molecules
by the Monoclonal Antibody SFR8-B6 To be Published
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3MKB
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![BU of 3mkb by Molmil](/molmil-images/mine/3mkb) | Crystal structure determination of Shortfin Mako (Isurus oxyrinchus) hemoglobin at 1.9 Angstrom resolution | 分子名称: | Hemoglobin subunit alpha, Hemoglobin subunit beta, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Ramesh, P, Sundaresan, S.S, Sathya Moorthy, P, Balasubramanian, M, Ponnuswamy, M.N. | 登録日 | 2010-04-14 | 公開日 | 2011-01-26 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural studies of haemoglobin from pisces species shortfin mako shark (Isurus oxyrinchus) at 1.9 angstrom resolution J.SYNCHROTRON RADIAT., 20, 2013
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2RI4
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![BU of 2ri4 by Molmil](/molmil-images/mine/2ri4) | |
4BEV
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![BU of 4bev by Molmil](/molmil-images/mine/4bev) | ATPase crystal structure with bound phosphate analogue | 分子名称: | COPPER EFFLUX ATPASE, MAGNESIUM ION, TRIFLUOROMAGNESATE | 著者 | Mattle, D, Drachmann, N.D, Liu, X.Y, Gourdon, P, Pedersen, B.P, Morth, P, Wang, J, Nissen, P. | 登録日 | 2013-03-12 | 公開日 | 2014-04-02 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (3.583 Å) | 主引用文献 | ATPase Crystal Structure with Bound Phosphate Analogue To be Published
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2YKH
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![BU of 2ykh by Molmil](/molmil-images/mine/2ykh) | Sensor region of a sensor histidine kinase | 分子名称: | PROBABLE SENSOR HISTIDINE KINASE PDTAS | 著者 | Preu, J, Panjikar, S, Morth, P, Jaiswal, R, Karunakar, P, Tucker, P.A. | 登録日 | 2011-05-27 | 公開日 | 2012-06-06 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.78 Å) | 主引用文献 | The Sensor Region of the Ubiquitous Cytosolic Sensor Kinase, Pdtas, Contains Pas and Gaf Domain Sensing Modules. J.Struct.Biol., 177, 2012
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2YKF
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![BU of 2ykf by Molmil](/molmil-images/mine/2ykf) | Sensor region of a sensor histidine kinase | 分子名称: | BROMIDE ION, PROBABLE SENSOR HISTIDINE KINASE PDTAS, SULFATE ION | 著者 | Preu, J, Panjikar, S, Morth, P, Jaiswal, R, Karunakar, P, Tucker, P.A. | 登録日 | 2011-05-26 | 公開日 | 2012-06-06 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The Sensor Region of the Ubiquitous Cytosolic Sensor Kinase, Pdtas, Contains Pas and Gaf Domain Sensing Modules. J.Struct.Biol., 177, 2012
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3CY5
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![BU of 3cy5 by Molmil](/molmil-images/mine/3cy5) | |
3D4X
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![BU of 3d4x by Molmil](/molmil-images/mine/3d4x) | |
1H15
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![BU of 1h15 by Molmil](/molmil-images/mine/1h15) | X-ray crystal structure of HLA-DRA1*0101/DRB5*0101 complexed with a peptide from Epstein Barr Virus DNA polymerase | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, DNA POLYMERASE, ... | 著者 | Lang, H, Jacobsen, H, Ikemizu, S, Andersson, C, Harlos, K, Madsen, L, Hjorth, P, Sondergaard, L, Svejgaard, A, Wucherpfennig, K, Stuart, D.I, Bell, J.I, Jones, E.Y, Fugger, L. | 登録日 | 2002-07-02 | 公開日 | 2002-10-03 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | A Functional and Structural Basis for Tcr Cross-Reactivity in Multiple Sclerosis Nat.Immunol., 3, 2002
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1HYO
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![BU of 1hyo by Molmil](/molmil-images/mine/1hyo) | CRYSTAL STRUCTURE OF FUMARYLACETOACETATE HYDROLASE COMPLEXED WITH 4-(HYDROXYMETHYLPHOSPHINOYL)-3-OXO-BUTANOIC ACID | 分子名称: | 4-[HYDROXY-[METHYL-PHOSPHINOYL]]-3-OXO-BUTANOIC ACID, ACETATE ION, CALCIUM ION, ... | 著者 | Bateman, R.L, Bhanumoorthy, P, Witte, J.F, McClard, R.W, Grompe, M, Timm, D.E. | 登録日 | 2001-01-21 | 公開日 | 2001-02-14 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Mechanistic inferences from the crystal structure of fumarylacetoacetate hydrolase with a bound phosphorus-based inhibitor. J.Biol.Chem., 276, 2001
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3D1A
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![BU of 3d1a by Molmil](/molmil-images/mine/3d1a) | |
1QCN
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![BU of 1qcn by Molmil](/molmil-images/mine/1qcn) | CRYSTAL STRUCTURE OF FUMARYLACETOACETATE HYDROLASE | 分子名称: | ACETATE ION, CALCIUM ION, FUMARYLACETOACETATE HYDROLASE, ... | 著者 | Timm, D.E, Mueller, H.A, Bhanumoorthy, P, Harp, J.M, Bunick, G.J. | 登録日 | 1999-05-14 | 公開日 | 2000-06-07 | 最終更新日 | 2022-12-21 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure and mechanism of a carbon-carbon bond hydrolase. Structure Fold.Des., 7, 1999
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1QQJ
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![BU of 1qqj by Molmil](/molmil-images/mine/1qqj) | CRYSTAL STRUCTURE OF MOUSE FUMARYLACETOACETATE HYDROLASE REFINED AT 1.55 ANGSTROM RESOLUTION | 分子名称: | ACETATE ION, CACODYLATE ION, CALCIUM ION, ... | 著者 | Timm, D.E, Mueller, H.A, Bhanumoorthy, P, Harp, J.M, Bunick, G.J. | 登録日 | 1999-06-07 | 公開日 | 2000-06-07 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Crystal structure and mechanism of a carbon-carbon bond hydrolase. Structure Fold.Des., 7, 1999
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1QCO
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![BU of 1qco by Molmil](/molmil-images/mine/1qco) | CRYSTAL STRUCTURE OF FUMARYLACETOACETATE HYDROLASE COMPLEXED WITH FUMARATE AND ACETOACETATE | 分子名称: | ACETOACETIC ACID, CALCIUM ION, FUMARIC ACID, ... | 著者 | Timm, D.E, Mueller, H.A, Bhanumoorthy, P, Harp, J.M, Bunick, G.J. | 登録日 | 1999-05-17 | 公開日 | 2000-06-07 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure and mechanism of a carbon-carbon bond hydrolase. Structure Fold.Des., 7, 1999
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1TUX
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![BU of 1tux by Molmil](/molmil-images/mine/1tux) | HIGH RESOLUTION CRYSTAL STRUCTURE OF A THERMOSTABLE XYLANASE FROM THERMOASCUS AURANTIACUS | 分子名称: | XYLANASE | 著者 | Natesh, R, Bhanumoorthy, P, Vithayathil, P.J, Sekar, K, Ramakumar, S, Viswamitra, M.A. | 登録日 | 1998-10-29 | 公開日 | 1999-07-22 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure at 1.8 A resolution and proposed amino acid sequence of a thermostable xylanase from Thermoascus aurantiacus. J.Mol.Biol., 288, 1999
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3GQP
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![BU of 3gqp by Molmil](/molmil-images/mine/3gqp) | |
3GYS
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![BU of 3gys by Molmil](/molmil-images/mine/3gys) | |
3GQR
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![BU of 3gqr by Molmil](/molmil-images/mine/3gqr) | |
2XSE
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![BU of 2xse by Molmil](/molmil-images/mine/2xse) | The structural basis for recognition of J-base containing DNA by a novel DNA-binding domain in JBP1 | 分子名称: | GLYCEROL, NITRATE ION, THYMINE DIOXYGENASE JBP1 | 著者 | Heidebrecht, T, Christodoulou, E, Chalmers, M.J, Jan, S, ter Riete, B, Grover, R.K, Joosten, R.P, Littler, D, vanLuenen, H, Griffin, P.R, Wentworth, P, Borst, P, Perrakis, A. | 登録日 | 2010-09-28 | 公開日 | 2011-03-30 | 最終更新日 | 2011-08-03 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | The Structural Basis for Recognition of Base J Containing DNA by a Novel DNA Binding Domain in Jbp1. Nucleic Acids Res., 39, 2011
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