3NR5
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![BU of 3nr5 by Molmil](/molmil-images/mine/3nr5) | Crystal structure of human Maf1 | 分子名称: | Repressor of RNA polymerase III transcription MAF1 homolog | 著者 | Ringel, R, Vannini, A, Kusser, A.G, Berninghausen, O, Kassavetis, G.A, Cramer, P. | 登録日 | 2010-06-30 | 公開日 | 2010-10-13 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Molecular Basis of RNA Polymerase III Transcription Repression by Maf1 Cell(Cambridge,Mass.), 143, 2010
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3ON1
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![BU of 3on1 by Molmil](/molmil-images/mine/3on1) | The structure of a protein with unknown function from Bacillus halodurans C | 分子名称: | BH2414 protein | 著者 | Fan, Y, Kagan, O, Savchenko, A, Joachimiak, A, Edwards, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2010-08-27 | 公開日 | 2010-09-22 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | The structure of a protein with unknown function from Bacillus halodurans C To be Published
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3OHS
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3ON2
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![BU of 3on2 by Molmil](/molmil-images/mine/3on2) | Structure of a protein with unknown function from Rhodococcus sp. RHA1 | 分子名称: | 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, Probable transcriptional regulator, SULFATE ION | 著者 | Fan, Y, Evdokimova, E, Egorova, O, Savchenko, A, Joachimiak, A, Edwards, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2010-08-27 | 公開日 | 2010-09-22 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | Structure of a protein with unknown function from Rhodococcus sp. RHA1 To be Published
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3OYT
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![BU of 3oyt by Molmil](/molmil-images/mine/3oyt) | 1.84 Angstrom resolution crystal structure of 3-oxoacyl-(acyl carrier protein) synthase I (fabB) from Yersinia pestis CO92 | 分子名称: | 1,2-ETHANEDIOL, 3-oxoacyl-[acyl-carrier-protein] synthase I, DI(HYDROXYETHYL)ETHER, ... | 著者 | Halavaty, A.S, Wawrzak, Z, Onopriyenko, O, Peterson, S, Savchenko, A, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2010-09-23 | 公開日 | 2011-01-12 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | 1.84 Angstrom resolution crystal structure of 3-oxoacyl-(acyl carrier protein) synthase I (fabB) from Yersinia pestis CO92 To be Published
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5MMV
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![BU of 5mmv by Molmil](/molmil-images/mine/5mmv) | Crystal structure of human Caspase-1 with 2-((2-naphthoyl)-L-valyl)-4-hydroxy-N-((3S)-2-hydroxy-5-oxotetrahydrofuran-3-yl)-2-azabicyclo[2.2.2]octane-3-carboxamide (Compound 1) | 分子名称: | (3~{S})-3-[[(3~{S})-2-[(2~{S})-3-methyl-2-(naphthalen-2-ylcarbonylamino)butanoyl]-4-oxidanyl-2-azabicyclo[2.2.2]octan-3-yl]carbonylamino]-4-oxidanyl-butanoic acid, Caspase-1 | 著者 | Brethon, A, Chantalat, L, Christin, O, Clary, L, Fournier, J.F, Gastreich, M, Harris, C, Pascau, J, Isabet, T, Rodeschin, V, Thoreau, E, Roche, D. | 登録日 | 2016-12-12 | 公開日 | 2017-12-20 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Crystal structure of human Caspase-1 with 2-((2-naphthoyl)-L-valyl)-4-hydroxy-N-((3S)-2-hydroxy-5-oxotetrahydrofuran-3-yl)-2-azabicyclo[2.2.2]octane-3-carboxamide (Compound 1) To Be Published
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5MYG
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![BU of 5myg by Molmil](/molmil-images/mine/5myg) | Crystal structure of the bromodomain of human BRPF1 in complex with NI-57 chemical probe | 分子名称: | 4-cyano-~{N}-(1,3-dimethyl-2-oxidanylidene-quinolin-6-yl)-2-methoxy-benzenesulfonamide, Peregrin | 著者 | Tallant, C, Igoe, N, Bayle, E.D, Krojer, T, Nunez-Alonso, G, Kopec, J, Fitzpatrick, F, Savitsky, P, Fedorov, O, Brennan, P.E, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Muller, S, Fish, P, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2017-01-26 | 公開日 | 2017-08-09 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Design of a Chemical Probe for the Bromodomain and Plant Homeodomain Finger-Containing (BRPF) Family of Proteins. J. Med. Chem., 60, 2017
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5MTJ
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![BU of 5mtj by Molmil](/molmil-images/mine/5mtj) | Yes1-SH2 in complex with monobody Mb(Yes_1) | 分子名称: | 3-CYCLOHEXYL-1-PROPYLSULFONIC ACID, Monobody Mb(Yes_1), SULFATE ION, ... | 著者 | Sha, F, Kukenshoner, T, Koide, S, Hantschel, O. | 登録日 | 2017-01-09 | 公開日 | 2017-04-05 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.949 Å) | 主引用文献 | Selective Targeting of SH2 Domain-Phosphotyrosine Interactions of Src Family Tyrosine Kinases with Monobodies. J. Mol. Biol., 429, 2017
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5MTM
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![BU of 5mtm by Molmil](/molmil-images/mine/5mtm) | Monobody Mb(Lck_3) bound to Lck-SH2 domain | 分子名称: | Monobody Mb(Lck_3), Tyrosine-protein kinase Lck, ZINC ION | 著者 | Pojer, F, Kukenshoner, T, Koide, S, Hantschel, O. | 登録日 | 2017-01-10 | 公開日 | 2017-04-05 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.405 Å) | 主引用文献 | Selective Targeting of SH2 Domain-Phosphotyrosine Interactions of Src Family Tyrosine Kinases with Monobodies. J. Mol. Biol., 429, 2017
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5MUQ
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![BU of 5muq by Molmil](/molmil-images/mine/5muq) | Crystal structure of DC8E8 Fab at pH 7.0 containing a Zn atom | 分子名称: | IMIDAZOLE, ZINC ION, antibody Fab heavy chain, ... | 著者 | Skrabana, R, Novak, M, Cehlar, O, Kontsekova, E. | 登録日 | 2017-01-13 | 公開日 | 2018-05-02 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.62 Å) | 主引用文献 | Crystal structure of DC8E8 Fab at pH 7.0 containing a Zn atom To be published
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5M9D
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3OUT
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![BU of 3out by Molmil](/molmil-images/mine/3out) | Crystal structure of glutamate racemase from Francisella tularensis subsp. tularensis SCHU S4 in complex with D-glutamate. | 分子名称: | D-GLUTAMIC ACID, Glutamate racemase | 著者 | Filippova, E.V, Wawrzak, Z, Onopriyenko, O, Kudriska, M, Edwards, A, Savchenko, A, Anderson, F.W, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2010-09-15 | 公開日 | 2010-09-29 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Crystal structure of glutamate racemase from Francisella tularensis subsp. tularensis SCHU S4 in complex with D-glutamate. To be Published
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3P1F
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![BU of 3p1f by Molmil](/molmil-images/mine/3p1f) | Crystal structure of the bromodomain of human CREBBP in complex with a hydroquinazolin ligand | 分子名称: | 1,2-ETHANEDIOL, 3-methyl-3,4-dihydroquinazolin-2(1H)-one, CREB-binding protein, ... | 著者 | Filippakopoulos, P, Picaud, S, Fedorov, O, Muniz, J, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Weigelt, J, Bountra, C, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2010-09-30 | 公開日 | 2010-12-08 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Crystal structure of the bromodomain of human CREBBP in complex with a hydroquinazolin ligand To be Published
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3OHI
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![BU of 3ohi by Molmil](/molmil-images/mine/3ohi) | Structure of Giardia fructose-1,6-biphosphate aldolase in complex with 3-hydroxy-2-pyridone | 分子名称: | ({3-hydroxy-2-oxo-4-[2-(phosphonooxy)ethyl]pyridin-1(2H)-yl}methyl)phosphonic acid, Putative fructose-1,6-bisphosphate aldolase, ZINC ION | 著者 | Herzberg, O, Galkin, A. | 登録日 | 2010-08-17 | 公開日 | 2011-01-19 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Rational design, synthesis and evaluation of first generation inhibitors of the Giardia lamblia fructose-1,6-biphosphate aldolase. J.Inorg.Biochem., 105, 2010
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3P52
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![BU of 3p52 by Molmil](/molmil-images/mine/3p52) | NH3-dependent NAD synthetase from Campylobacter jejuni subsp. jejuni NCTC 11168 in complex with the nitrate ion | 分子名称: | NH(3)-dependent NAD(+) synthetase, NITRATE ION | 著者 | Filippova, E.V, Wawrzak, Z, Onopriyenko, O, Skarina, T, Edwards, A, Savchenko, A, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2010-10-07 | 公開日 | 2010-10-27 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2.74 Å) | 主引用文献 | NH3-dependent NAD synthetase from Campylobacter jejuni subsp. jejuni NCTC 11168 in complex with the nitrate ion To be Published
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5NJ8
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3OP3
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![BU of 3op3 by Molmil](/molmil-images/mine/3op3) | Crystal Structure of Cell Division Cycle 25C Protein Isoform A from Homo sapiens | 分子名称: | M-phase inducer phosphatase 3, SULFATE ION | 著者 | Kim, Y, Weger, A, Hatzos, C, Savitsky, P, Johansson, C, Ball, L, Barr, A, Vollmar, M, Muniz, J, Weigelt, J, Arrowsmith, C.H, Edwards, A, Bountra, C, Gileadi, O, von Delft, F, Knapp, S, Joachimiak, A, Structural Genomics Consortium (SGC) | 登録日 | 2010-08-31 | 公開日 | 2010-09-29 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.63 Å) | 主引用文献 | Crystal Structure of Cell Division Cycle 25C Protein Isoform A from Homo sapiens TO BE PUBLISHED
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3OQJ
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![BU of 3oqj by Molmil](/molmil-images/mine/3oqj) | Crystal structure of B. licheniformis CDPS yvmC-BLIC in complex with CAPSO | 分子名称: | (2S)-3-(cyclohexylamino)-2-hydroxypropane-1-sulfonic acid, Putative uncharacterized protein yvmC | 著者 | Bonnefond, L, Arai, T, Suzuki, T, Ishitani, R, Nureki, O. | 登録日 | 2010-09-03 | 公開日 | 2011-02-23 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.399 Å) | 主引用文献 | Structural basis for nonribosomal peptide synthesis by an aminoacyl-tRNA synthetase paralog. Proc.Natl.Acad.Sci.USA, 108, 2011
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3OT7
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![BU of 3ot7 by Molmil](/molmil-images/mine/3ot7) | Escherichia coli apo-manganese superoxide dismutase | 分子名称: | Superoxide dismutase [Mn] | 著者 | Whittaker, M.M, Lerch, T.F, Kirillova, O, Chapman, M.S, Whittaker, J.W. | 登録日 | 2010-09-10 | 公開日 | 2010-12-22 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.901 Å) | 主引用文献 | Subunit dissociation and metal binding by Escherichia coli apo-manganese superoxide dismutase. Arch.Biochem.Biophys., 505, 2011
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5N2N
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![BU of 5n2n by Molmil](/molmil-images/mine/5n2n) | Crystal structure of the receiver domain of the histidine kinase CKI1 from Arabidopsis thaliana complexed with Mg2+ and BeF3- | 分子名称: | BERYLLIUM TRIFLUORIDE ION, Histidine kinase CKI1, MAGNESIUM ION | 著者 | Otrusinova, O, Demo, G, Padrta, P, Jasenakova, Z, Pekarova, B, Gelova, Z, Szmitkowska, A, Kaderavek, P, Jansen, S, Zachrdla, M, Klumpler, T, Marek, J, Hritz, J, Janda, L, Iwai, H, Wimmerova, M, Hejatko, J, Zidek, L. | 登録日 | 2017-02-08 | 公開日 | 2017-09-13 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Conformational dynamics are a key factor in signaling mediated by the receiver domain of a sensor histidine kinase from Arabidopsis thaliana. J. Biol. Chem., 292, 2017
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3P0A
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3P77
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![BU of 3p77 by Molmil](/molmil-images/mine/3p77) | Crystal Structures of the Chicken YF1*7.1 molecule | 分子名称: | ACETATE ION, Beta-2-microglobulin, MHC Rfp-Y class I alpha chain, ... | 著者 | Hee, C.S, Gao, S, Loll, B, Miller, M.M, Uchanska-Ziegler, B, Daumke, O, Ziegler, A. | 登録日 | 2010-10-12 | 公開日 | 2010-11-24 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structure of a Classical MHC Class I Molecule That Binds "Non-Classical" Ligands. Plos Biol., 8, 2010
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5N9R
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![BU of 5n9r by Molmil](/molmil-images/mine/5n9r) | Crystal structure of USP7 in complex with a potent, selective and reversible small-molecule inhibitor | 分子名称: | 7-bromanyl-3-[[4-oxidanyl-1-[(3~{R})-3-phenylbutanoyl]piperidin-4-yl]methyl]thieno[3,2-d]pyrimidin-4-one, DIMETHYL SULFOXIDE, GLYCEROL, ... | 著者 | Harrison, T, Gavory, G, O'Dowd, C, Helm, M, Flasz, I, Arkoudis, E, Dossang, A, Hughes, C, Cassidy, E, McClelland, K, Odrzywol, E, Page, N, Barker, O, Miel, H. | 登録日 | 2017-02-27 | 公開日 | 2017-12-06 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.23 Å) | 主引用文献 | Discovery and characterization of highly potent and selective allosteric USP7 inhibitors. Nat. Chem. Biol., 14, 2018
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3OPZ
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![BU of 3opz by Molmil](/molmil-images/mine/3opz) | Crystal structure of trans-sialidase in complex with the Fab fragment of a neutralizing monoclonal IgG antibody | 分子名称: | 1,4-DIETHYLENE DIOXIDE, SODIUM ION, Trans-sialidase, ... | 著者 | Larrieux, N, Muia, R, Campetella, O, Buschiazzo, A. | 登録日 | 2010-09-02 | 公開日 | 2011-11-09 | 最終更新日 | 2021-10-06 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | Trypanosoma cruzi trans-sialidase in complex with a neutralizing antibody: structure/function studies towards the rational design of inhibitors. Plos Pathog., 8, 2012
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3P05
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