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PDB: 3 件

4D7G
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BU of 4d7g by Molmil
Human FXIa in complex with small molecule inhibitors.
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, COAGULATION FACTOR XIA, GLYCEROL, ...
著者Sandmark, J, Oster, L, Jacso, T, Ullah, V, Redzick, A, Borjesson, U, Olsson, T, Norberg, M, Akerud, T.
登録日2014-11-24
公開日2016-01-20
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献From Mm Fragments to Nm Compounds Using Iloe-NMR to Guide Linking of Compounds in Fragment Based Drug Discovery (Fbdd).
To be Published
4D76
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BU of 4d76 by Molmil
Human FXIa in complex with small molecule inhibitors.
分子名称: COAGULATION FACTOR XI, GLYCEROL, N-[(2S)-1-({5-[(diaminomethylidene)amino]pentyl}amino)-1-oxo-3-phenylpropan-2-yl]-4-hydroxy-2-oxo-1,2-dihydroquinoline-6-carboxamide, ...
著者Sandmark, J, Oster, L, Jacso, T, Ullah, V, Redzick, A, Borjesson, U, Olsson, T, Norberg, M, Akerud, T.
登録日2014-11-20
公開日2016-01-20
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献From Mm Fragments to Nm Compounds Using Iloe-NMR to Guide Linking of Compounds in Fragment Based Drug Discovery (Fbdd).
To be Published
4D7F
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BU of 4d7f by Molmil
Human FXIa in complex with small molecule inhibitors.
分子名称: COAGULATION FACTOR XI, GLYCEROL, N-[(2S)-1-({4-[(diaminomethylidene)amino]butyl}amino)-1-oxo-3-phenylpropan-2-yl]-4-hydroxy-2-oxo-1,2-dihydroquinoline-6-carboxamide, ...
著者Sandmark, J, Oster, L, Jacso, T, Ullah, V, Redzick, A, Borjesson, U, Olsson, T, Norberg, M, Akerud, T.
登録日2014-11-24
公開日2016-01-20
実験手法X-RAY DIFFRACTION (1.62 Å)
主引用文献From Mm Fragments to Nm Compounds Using Iloe-NMR to Guide Linking of Compounds in Fragment Based Drug Discovery (Fbdd).
To be Published

219869

件を2024-05-15に公開中

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