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PDB: 492 件

6UL7
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Structure of human ketohexokinase-C in complex with fructose, NO3, and osthole
分子名称: 7-methoxy-8-(3-methylbut-2-enyl)chromen-2-one, Ketohexokinase, NITRATE ION, ...
著者Gasper, W.C, Gardner, S, Allen, K.N, Tolan, D.R.
登録日2019-10-07
公開日2021-04-07
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure of human ketohexokinase-C in complex with fructose, NO3, and osthole
To be Published
8Q6S
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A carbohydrate esterase family 15 (CE15) glucuronoyl esterase from Phocaeicola vulgatus ATCC 8482
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, DI(HYDROXYETHYL)ETHER, Putative acetyl xylan esterase, ...
著者Mazurkewich, S, Seveso, A, Banerjee, S, Lo Leggio, L, Larsbrink, J.
登録日2023-08-14
公開日2023-12-13
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Polysaccharide utilization loci from Bacteroidota encode CE15 enzymes with possible roles in cleaving pectin-lignin bonds.
Appl.Environ.Microbiol., 90, 2024
7ZJ2
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Amyloid fibril (in vitro) from full-length hnRNPA1 protein
分子名称: Isoform A1-A of Heterogeneous nuclear ribonucleoprotein A1
著者Sharma, K, Banerjee, S, Schmidt, M, Faendrich, M.
登録日2022-04-08
公開日2023-08-02
最終更新日2023-08-09
実験手法ELECTRON MICROSCOPY (3.32 Å)
主引用文献Cryo-EM Structure of the Full-length hnRNPA1 Amyloid Fibril.
J.Mol.Biol., 435, 2023
6FHE
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Highly active enzymes by automated modular backbone assembly and sequence design
分子名称: Synthetic construct
著者Lapidot, G, Khersonsky, O, Lipsh, R, Dym, O, Albeck, S, Rogotner, S, Fleishman, J.S.
登録日2018-01-14
公開日2018-07-25
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Highly active enzymes by automated combinatorial backbone assembly and sequence design.
Nat Commun, 9, 2018
6FQE
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Phosphotriesterase PTE_A53_4
分子名称: (4~{S},6~{R})-2,2,6-trimethyl-1,3-dioxan-4-ol, DI(HYDROXYETHYL)ETHER, FORMIC ACID, ...
著者Dym, O, Aggarwal, N, Albeck, S, Unger, T, Hamer Rogotner, S, Silman, I, Leader, H, Ashani, Y, Goldsmith, M, Greisen, P, Tawfik, D, Sussman, L.J.
登録日2018-02-14
公開日2019-03-13
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Phosphotriesterase PTE_A53_4
To Be Published
6FYH
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Disulfide between ubiquitin G76C and the E3 HECT ligase Huwe1
分子名称: E3 ubiquitin-protein ligase HUWE1, Polyubiquitin-B, SULFATE ION, ...
著者Jaeckl, M, Hartmann, M.D, Wiesner, S.
登録日2018-03-12
公開日2018-07-11
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.906 Å)
主引用文献beta-Sheet Augmentation Is a Conserved Mechanism of Priming HECT E3 Ligases for Ubiquitin Ligation.
J. Mol. Biol., 430, 2018
8BA5
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Crystal structure of the DNMT3A ADD domain
分子名称: 1,2-ETHANEDIOL, DNA (cytosine-5)-methyltransferase 3A, MAGNESIUM ION, ...
著者Linhard, V, Kunert, S, Wollenhaupt, J, Broehm, A, Schwalbe, H, Jeltsch, A.
登録日2022-10-11
公開日2022-11-23
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献The MECP2-TRD domain interacts with the DNMT3A-ADD domain at the H3-tail binding site.
Protein Sci., 32, 2023
6FX4
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Disulfide between E3 HECT ligase Smurf2 and Ubiquitin G76C
分子名称: E3 ubiquitin-protein ligase SMURF2, GLYCEROL, Polyubiquitin-B
著者Jaeckl, M, Holdermann, I, Wiesner, S.
登録日2018-03-08
公開日2018-07-11
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献beta-Sheet Augmentation Is a Conserved Mechanism of Priming HECT E3 Ligases for Ubiquitin Ligation.
J. Mol. Biol., 430, 2018
6FU6
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BU of 6fu6 by Molmil
Phosphotriesterase PTE_C23_2
分子名称: FORMIC ACID, POLYACRYLIC ACID, Parathion hydrolase, ...
著者Dym, O, Aggarwal, N, Albeck, S, Unger, T, Hamer Rogotner, S, Silman, I, Leader, H, Ashani, Y, Goldsmith, M, Greisen, P, Tawfik, D, Sussman, L.J.
登録日2018-02-26
公開日2019-03-20
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Phosphotriesterase PTE_A53_4
To Be Published
6WMV
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BU of 6wmv by Molmil
Structure of a phosphatidylinositol-phosphate synthase (PIPS) from Mycobacterium kansasii with evidence of substrate binding
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 3,3',3''-phosphanetriyltripropanoic acid, AfCTD-Phosphatidylinositol-phosphate synthase (PIPS) fusion, ...
著者Belcher Dufrisne, M, Jorge, C.D, Timoteo, C.G, Petrou, V.I, Ashraf, K.U, Banerjee, S, Clarke, O.B, Santos, H, Mancia, F.
登録日2020-04-21
公開日2020-05-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.142 Å)
主引用文献Structural and Functional Characterization of Phosphatidylinositol-Phosphate Biosynthesis in Mycobacteria.
J.Mol.Biol., 432, 2020
6WM5
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Structure of a phosphatidylinositol-phosphate synthase (PIPS) from Mycobacterium kansasii
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHATE, 3,3',3''-phosphanetriyltripropanoic acid, ...
著者Belcher Dufrisne, M, Jorge, C.D, Timoteo, C.G, Petrou, V.I, Ashraf, K.U, Banerjee, S, Clarke, O.B, Santos, H, Mancia, F, New York Consortium on Membrane Protein Structure (NYCOMPS)
登録日2020-04-20
公開日2020-05-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.961 Å)
主引用文献Structural and Functional Characterization of Phosphatidylinositol-Phosphate Biosynthesis in Mycobacteria.
J.Mol.Biol., 432, 2020
6UAN
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BU of 6uan by Molmil
B-Raf:14-3-3 complex
分子名称: 14-3-3 zeta, Serine/threonine-protein kinase B-raf
著者Kondo, Y, Ognjenovic, J, Banerjee, S, Karandur, D, Merk, A, Kulhanek, K, Wong, K, Roose, J.P, Subramaniam, S, Kuriyan, J.
登録日2019-09-11
公開日2019-09-25
最終更新日2019-12-18
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Cryo-EM structure of a dimeric B-Raf:14-3-3 complex reveals asymmetry in the active sites of B-Raf kinases.
Science, 366, 2019
6FHO
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Crystal structure of pqsL, a probable FAD-dependent monooxygenase from Pseudomonas aeruginosa - new refinement
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, Probable FAD-dependent monooxygenase
著者Belviso, B.D, Drees, S.L, Ernst, S, Jagmann, N, Hennecke, U, Fetzner, S.
登録日2018-01-15
公開日2018-04-25
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献PqsL uses reduced flavin to produce 2-hydroxylaminobenzoylacetate, a preferred PqsBC substrate in alkyl quinolone biosynthesis inPseudomonas aeruginosa.
J. Biol. Chem., 293, 2018
6N47
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BU of 6n47 by Molmil
The structure of SB-2-204-tubulin complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-(2-chloropyrido[3,2-d]pyrimidin-4-yl)-7-methoxy-3,4-dihydroquinoxalin-2(1H)-one, CALCIUM ION, ...
著者Arnst, K, Banerjee, S, Wang, Y, Li, W, Miller, D, Li, W.
登録日2018-11-17
公開日2019-11-13
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献X-ray Crystal Structure Guided Discovery and Antitumor Efficacy of Dihydroquinoxalinone as Potent Tubulin Polymerization Inhibitors.
Acs Chem.Biol., 14, 2019
6FFW
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BU of 6ffw by Molmil
Phosphotriesterase PTE_A53_5
分子名称: (4~{S},6~{R})-2,2,6-trimethyl-1,3-dioxan-4-ol, 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ...
著者Dym, O, Aggarwal, N, Albeck, S, Unger, T, Hamer Rogotner, S, Silman, I, Leader, H, Ashani, Y, Goldsmith, M, Greisen, P, Tawfik, D, Sussman, L.J.
登録日2018-01-09
公開日2019-03-13
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.495 Å)
主引用文献Phosphotriesterase PTE_A53_5
To Be Published
6FHF
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BU of 6fhf by Molmil
Highly active enzymes by automated modular backbone assembly and sequence design
分子名称: Design, SODIUM ION
著者Lapidot, G, Khersonsky, O, Lipsh, R, Dym, O, Albeck, S, Rogotner, S, Fleishman, J.S.
登録日2018-01-14
公開日2018-07-25
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Highly active enzymes by automated combinatorial backbone assembly and sequence design.
Nat Commun, 9, 2018
6G1J
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BU of 6g1j by Molmil
Phosphotriesterase PTE_C23M_1
分子名称: 1-ethyl-1-methyl-cyclohexane, FORMIC ACID, GLYCEROL, ...
著者Dym, O, Aggarwal, N, Albeck, S, Unger, T, Hamer Rogotner, S, Silman, I, Leader, H, Ashani, Y, Goldsmith, M, Greisen, P, Tawfik, D, Sussman, L.J.
登録日2018-03-21
公開日2019-04-10
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Phosphotriesterase PTE_C23M_1
To Be Published
6FWE
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BU of 6fwe by Molmil
Phosphotriesterase PTE_C23_6
分子名称: 1-[methoxy(methyl)phosphoryl]oxyethane, 1-ethyl-1-methyl-cyclohexane, FORMIC ACID, ...
著者Dym, O, Aggarwal, N, Albeck, S, Unger, T, Hamer Rogotner, S, Silman, I, Leader, H, Ashani, Y, Goldsmith, M, Greisen, P, Tawfik, D, Sussman, L.J.
登録日2018-03-06
公開日2019-03-27
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.774 Å)
主引用文献Phosphotriesterase PTE_C23_6
To Be Published
5EJK
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BU of 5ejk by Molmil
Crystal structure of the Rous sarcoma virus intasome
分子名称: DNA (5'-D(*AP*AP*TP*GP*TP*TP*GP*TP*CP*TP*TP*AP*TP*GP*CP*AP*AP*TP*AP*CP*TP*C)-3'), DNA (5'-D(*AP*GP*TP*GP*TP*CP*TP*T)-3'), DNA (5'-D(*CP*TP*TP*CP*TP*CP*TP*C)-3'), ...
著者Yin, Z, Shi, K, Banerjee, S, Aihara, H.
登録日2015-11-02
公開日2016-02-17
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Crystal structure of the Rous sarcoma virus intasome.
Nature, 530, 2016
5EG4
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BOVINE TRYPSIN IN COMPLEX WITH CYCLIC INHIBITOR
分子名称: (13S,16R)-N-(4-carbamimidoylbenzyl)-16-((N-cyclohexylsulfamoyl)amino)-3,9,15-trioxo-2,10,14-triaza-6(1,4)-piperazina-1, 11(1,4)-dibenzenacycloheptadecaphane-13-carboxamide, ACETATE ION, ...
著者Knoerlein, A, Wagner, S, Heine, A, Steinmetzer, T, Klebe, G.
登録日2015-10-26
公開日2016-07-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.32 Å)
主引用文献Optimization of Cyclic Plasmin Inhibitors: From Benzamidines to Benzylamines.
J.Med.Chem., 59, 2016
6FRZ
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BU of 6frz by Molmil
Phosphotriesterase PTE_A53_7
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 5-methylcyclohexane-1,1,3,3-tetrol, DI(HYDROXYETHYL)ETHER, ...
著者Dym, O, Aggarwal, N, Albeck, S, Unger, T, Hamer Rogotner, S, Silman, I, Leader, H, Ashani, Y, Goldsmith, M, Greisen, P, Tawfik, D, Sussman, L.J.
登録日2018-02-18
公開日2019-03-13
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Phosphotriesterase PTE_A53_7
To Be Published
6WQX
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BU of 6wqx by Molmil
Human PRPK-TPRKB complex
分子名称: EKC/KEOPS complex subunit TP53RK, EKC/KEOPS complex subunit TPRKB, MAGNESIUM ION, ...
著者Li, J, Ma, X.L, Banerjee, S, Dong, Z.G.
登録日2020-04-29
公開日2021-02-17
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.53 Å)
主引用文献Crystal structure of the human PRPK-TPRKB complex.
Commun Biol, 4, 2021
6G3M
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BU of 6g3m by Molmil
Phosphotriesterase PTE_C23M_4
分子名称: 1-ethyl-1-methyl-cyclohexane, CHLORIDE ION, FORMIC ACID, ...
著者Dym, O, Aggarwal, N, Albeck, S, Unger, T, Hamer Rogotner, S, Silman, I, Leader, H, Ashani, Y, Goldsmith, M, Greisen, P, Tawfik, D, Sussman, L.J.
登録日2018-03-26
公開日2019-04-10
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.665 Å)
主引用文献Phosphotriesterase PTE_C23M_4
To Be Published
5HBS
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BU of 5hbs by Molmil
Crystal structure of human cellular retinol binding protein 1 in complex with all-trans-retinol at 0.89 angstrom.
分子名称: RETINOL, Retinol-binding protein 1
著者Golczak, M, Arne, J.M, Silvaroli, J.A, Kiser, P.D, Banerjee, S.
登録日2016-01-02
公開日2016-03-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (0.89 Å)
主引用文献Ligand Binding Induces Conformational Changes in Human Cellular Retinol-binding Protein 1 (CRBP1) Revealed by Atomic Resolution Crystal Structures.
J.Biol.Chem., 291, 2016
5HA1
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Crystal structure of human cellular retinol binding protein 1 in complex with retinylamine
分子名称: (2~{E},4~{E},6~{E},8~{E})-3,7-dimethyl-9-(2,6,6-trimethylcyclohexen-1-yl)nona-2,4,6,8-tetraen-1-amine, Retinol-binding protein 1
著者Golczak, M, Arne, J.M, Silvaroli, J.A, Kiser, P.D, Banerjee, S.
登録日2015-12-29
公開日2016-03-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Ligand Binding Induces Conformational Changes in Human Cellular Retinol-binding Protein 1 (CRBP1) Revealed by Atomic Resolution Crystal Structures.
J.Biol.Chem., 291, 2016

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件を2024-07-17に公開中

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