5WLV
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![BU of 5wlv by Molmil](/molmil-images/mine/5wlv) | Carbonic Anhydrase II in complex with aryloxy-2-hydroxypropylammine sulfonamide | 分子名称: | 4-{(2R)-2-hydroxy-3-[(propan-2-yl)amino]propoxy}-N-[2-(4-sulfamoylphenyl)ethyl]benzamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ... | 著者 | Lomelino, C.L, Andring, J.T, McKenna, R. | 登録日 | 2017-07-27 | 公開日 | 2018-08-01 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Discovery of beta-Adrenergic Receptors Blocker-Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy. J. Med. Chem., 61, 2018
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5SZ5
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![BU of 5sz5 by Molmil](/molmil-images/mine/5sz5) | Carbonic anhydrase IX-mimic in complex with 4-(2-methylphenyl)-benzenesulfonamide | 分子名称: | 4-(2-methylphenyl)-benzenesulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ... | 著者 | Bhatt, A, Mahon, B.P, Cornelio, B, McKenna, R. | 登録日 | 2016-08-12 | 公開日 | 2016-12-28 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.274 Å) | 主引用文献 | Structure-Activity Relationships of Benzenesulfonamide-Based Inhibitors towards Carbonic Anhydrase Isoform Specificity. Chembiochem, 18, 2017
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5SZ1
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![BU of 5sz1 by Molmil](/molmil-images/mine/5sz1) | Carbonic anhydrase II in complex with 4-(2-methylphenyl)-benzenesulfonamide | 分子名称: | 4-(2-methylphenyl)-benzenesulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ... | 著者 | Bhatt, A, Mahon, B.P, Cornelio, B, McKenna, R. | 登録日 | 2016-08-12 | 公開日 | 2016-12-21 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structure-Activity Relationships of Benzenesulfonamide-Based Inhibitors towards Carbonic Anhydrase Isoform Specificity. Chembiochem, 18, 2017
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5WLR
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![BU of 5wlr by Molmil](/molmil-images/mine/5wlr) | |
5SZ3
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![BU of 5sz3 by Molmil](/molmil-images/mine/5sz3) | Carbonic anhydrase II in complex with 4-(3-quinolinyl)-benzenesulfonamide | 分子名称: | 4-(3-quinolinyl)-benzenesulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ... | 著者 | Bhatt, A, Mahon, B.P, Cornelio, B, McKenna, R. | 登録日 | 2016-08-12 | 公開日 | 2016-12-21 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.689 Å) | 主引用文献 | Structure-Activity Relationships of Benzenesulfonamide-Based Inhibitors towards Carbonic Anhydrase Isoform Specificity. Chembiochem, 18, 2017
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5SZ6
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![BU of 5sz6 by Molmil](/molmil-images/mine/5sz6) | Carbonic anhydrase IX-mimic in complex with 4-(3-formylphenyl)-benzenesulfonamide | 分子名称: | 4-(3-formylphenyl)-benzenesulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ... | 著者 | Bhatt, A, Mahon, B.P, Cornelio, B, McKenna, R. | 登録日 | 2016-08-12 | 公開日 | 2016-12-28 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | Structure-Activity Relationships of Benzenesulfonamide-Based Inhibitors towards Carbonic Anhydrase Isoform Specificity. Chembiochem, 18, 2017
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5WLT
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![BU of 5wlt by Molmil](/molmil-images/mine/5wlt) | Carbonic Anhydrase IX-mimic in complex with aryloxy-2-hydroxypropylammine sulfonamide | 分子名称: | 4-{(2S)-2-hydroxy-3-[(propan-2-yl)amino]propoxy}benzene-1-sulfonamide, Carbonic anhydrase 2, GLYCEROL, ... | 著者 | Lomelino, C.L, Andring, J.T, McKenna, R. | 登録日 | 2017-07-27 | 公開日 | 2018-08-01 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Discovery of beta-Adrenergic Receptors Blocker-Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy. J. Med. Chem., 61, 2018
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5T84
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![BU of 5t84 by Molmil](/molmil-images/mine/5t84) | HIV-1 protease, unbound subtype B L63P construct | 分子名称: | Protease | 著者 | Liu, Z, Norell, J, Mahon, B, Poole, K, McKenna, R, Fanucci, G. | 登録日 | 2016-09-06 | 公開日 | 2017-09-20 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Single mutation, L63P, capable of shutting down the flaps of HIV-1 protease To Be Published
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1EM0
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![BU of 1em0 by Molmil](/molmil-images/mine/1em0) | COMPLEX OF D(CCTAGG) WITH TETRA-[N-METHYL-PYRIDYL] PORPHYRIN | 分子名称: | DNA (5'-D(*(CBR)P*CP*TP*AP*GP*G)-3'), MAGNESIUM ION, TETRA[N-METHYL-PYRIDYL] PORPHYRIN-NICKEL | 著者 | Neidle, S, Sanderson, M, Bennett, M, Krah, A, Wien, F, Garman, E, McKenna, R. | 登録日 | 2000-03-14 | 公開日 | 2000-08-21 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (0.9 Å) | 主引用文献 | A DNA-porphyrin minor-groove complex at atomic resolution: the structural consequences of porphyrin ruffling. Proc.Natl.Acad.Sci.USA, 97, 2000
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1XV8
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![BU of 1xv8 by Molmil](/molmil-images/mine/1xv8) | Crystal Structure of Human Salivary Alpha-Amylase Dimer | 分子名称: | Alpha-amylase, CALCIUM ION, CHLORIDE ION | 著者 | Fisher, S.Z, Govindasamy, L, Tu, C.K, Silverman, D.N, Rajaniemi, H, McKenna, R. | 登録日 | 2004-10-27 | 公開日 | 2005-10-11 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Crystal Structure of Human Salivary Alpha-Amylase Dimer To be Published
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3RAA
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![BU of 3raa by Molmil](/molmil-images/mine/3raa) | Structural studies of AAV8 capsid transitions associated with endosomal trafficking | 分子名称: | ADENOSINE MONOPHOSPHATE, Capsid protein | 著者 | Nam, H.-J, Gurda, B, McKenna, R, Porter, M, Byrne, B, Salganik, M, Muzyczka, N, Agbandje-McKenna, M. | 登録日 | 2011-03-27 | 公開日 | 2011-09-21 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Structural studies of adeno-associated virus serotype 8 capsid transitions associated with endosomal trafficking. J.Virol., 85, 2011
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1YO1
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![BU of 1yo1 by Molmil](/molmil-images/mine/1yo1) | Proton Transfer from His200 in Human Carbonic Anhydrase II | 分子名称: | Carbonic anhydrase II, SULFATE ION, ZINC ION | 著者 | Bhatt, D, Tu, C, Fisher, S.Z, Hernandez Prada, J.A, McKenna, R, Silverman, D.N. | 登録日 | 2005-01-26 | 公開日 | 2005-09-20 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Proton transfer in a Thr200His mutant of human carbonic anhydrase II Proteins, 61, 2005
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1YO0
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![BU of 1yo0 by Molmil](/molmil-images/mine/1yo0) | Proton Transfer from His200 in Human Carbonic Anhydrase II | 分子名称: | CHLORIDE ION, Carbonic anhydrase II, ZINC ION | 著者 | Bhatt, D, Tu, C, Fisher, S.Z, Hernandez Prada, J.A, McKenna, R, Silverman, D.N. | 登録日 | 2005-01-26 | 公開日 | 2005-09-20 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Proton transfer in a Thr200His mutant of human carbonic anhydrase II Proteins, 61, 2005
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1YO2
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![BU of 1yo2 by Molmil](/molmil-images/mine/1yo2) | Proton Transfer from His200 in Human Carbonic Anhydrase II | 分子名称: | Carbonic anhydrase II, ZINC ION | 著者 | Bhatt, D, Tu, C, Fisher, S.Z, Hernandez Prada, J.A, McKenna, R, Silverman, D.N. | 登録日 | 2005-01-26 | 公開日 | 2005-09-20 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Proton transfer in a Thr200His mutant of human carbonic anhydrase II Proteins, 61, 2005
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3RA4
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![BU of 3ra4 by Molmil](/molmil-images/mine/3ra4) | Structural studies of AAV8 capsid transitions associated with endosomal trafficking | 分子名称: | Capsid protein, DNA (5'-D(*CP*A)-3') | 著者 | Nam, H.-J, Gurda, B, McKenna, R, Porter, M, Byrne, B, Salganik, M, Muzyczka, N, Agbandje-McKenna, M. | 登録日 | 2011-03-27 | 公開日 | 2011-09-21 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural studies of adeno-associated virus serotype 8 capsid transitions associated with endosomal trafficking. J.Virol., 85, 2011
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3RA8
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![BU of 3ra8 by Molmil](/molmil-images/mine/3ra8) | Structural studies of AAV8 capsid transitions associated with endosomal trafficking | 分子名称: | ADENOSINE MONOPHOSPHATE, Capsid protein | 著者 | Nam, H.-J, Gurda, B, McKenna, R, Porter, M, Byrne, B, Salganik, M, Muzyczka, N, Agbandje-McKenna, M. | 登録日 | 2011-03-27 | 公開日 | 2011-09-21 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural studies of adeno-associated virus serotype 8 capsid transitions associated with endosomal trafficking. J.Virol., 85, 2011
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3RA2
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![BU of 3ra2 by Molmil](/molmil-images/mine/3ra2) | Structural studies of AAV8 capsid transitions associated with endosomal trafficking | 分子名称: | Capsid protein | 著者 | Nam, H.-J, Gurda, B, McKenna, R, Porter, M, Byrne, B, Salganik, M, Muzyczka, N, Agbandje-McKenna, M. | 登録日 | 2011-03-26 | 公開日 | 2011-09-21 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural studies of adeno-associated virus serotype 8 capsid transitions associated with endosomal trafficking. J.Virol., 85, 2011
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3RA9
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![BU of 3ra9 by Molmil](/molmil-images/mine/3ra9) | Structural studies of AAV8 capsid transitions associated with endosomal trafficking | 分子名称: | Capsid protein, DNA (5'-D(P*CP*A)-3') | 著者 | Nam, H.-J, Gurda, B, McKenna, R, Porter, M, Byrne, B, Salganik, M, Muzyczka, N, Agbandje-McKenna, M. | 登録日 | 2011-03-27 | 公開日 | 2011-09-21 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural studies of adeno-associated virus serotype 8 capsid transitions associated with endosomal trafficking. J.Virol., 85, 2011
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5BQ1
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![BU of 5bq1 by Molmil](/molmil-images/mine/5bq1) | Capturing Carbon Dioxide in beta Carbonic Anhydrase | 分子名称: | CARBON DIOXIDE, Carbonic anhydrase, ZINC ION | 著者 | Aggarwal, M, Chua, T.K, Pinard, M.A, Szebenyi, D.M, McKenna, R. | 登録日 | 2015-05-28 | 公開日 | 2015-10-28 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Carbon Dioxide "Trapped" in a beta-Carbonic Anhydrase. Biochemistry, 54, 2015
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3UYN
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![BU of 3uyn by Molmil](/molmil-images/mine/3uyn) | HCA 3 | 分子名称: | Carbonic anhydrase 3, ZINC ION | 著者 | Fisher, Z, McKenna, R. | 登録日 | 2011-12-06 | 公開日 | 2012-02-01 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural and kinetic analysis of proton shuttle residues in the active site of human carbonic anhydrase III. Proteins, 68, 2007
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3UYQ
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![BU of 3uyq by Molmil](/molmil-images/mine/3uyq) | HCA 3 | 分子名称: | Carbonic anhydrase 3, ZINC ION | 著者 | Fisher, Z, McKenna, R. | 登録日 | 2011-12-06 | 公開日 | 2011-12-21 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural and kinetic analysis of proton shuttle residues in the active site of human carbonic anhydrase III. Proteins, 68, 2007
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4G0C
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![BU of 4g0c by Molmil](/molmil-images/mine/4g0c) | Neutron structure of acetazolamide-bound human carbonic anhydrase II reveal molecular details of drug binding. | 分子名称: | 5-ACETAMIDO-1,3,4-THIADIAZOLE-2-SULFONAMIDE, Carbonic anhydrase 2, ZINC ION | 著者 | Fisher, S.Z, McKenna, R, Aggarwal, M. | 登録日 | 2012-07-09 | 公開日 | 2012-09-19 | 最終更新日 | 2023-09-13 | 実験手法 | NEUTRON DIFFRACTION (2 Å) | 主引用文献 | Neutron diffraction of acetazolamide-bound human carbonic anhydrase II reveals atomic details of drug binding. J.Am.Chem.Soc., 134, 2012
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4HEY
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![BU of 4hey by Molmil](/molmil-images/mine/4hey) | |
4HEW
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![BU of 4hew by Molmil](/molmil-images/mine/4hew) | |
4HBA
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![BU of 4hba by Molmil](/molmil-images/mine/4hba) | Structural and Catalytic Characterization of a Thermal and Acid Stable Variant of Human Carbonic Anhydrase II Containing an Engineered Disulfide Bond | 分子名称: | Carbonic anhydrase 2, GLYCEROL, ZINC ION | 著者 | Boone, C.D, Habibzadegan, A, McKenna, R. | 登録日 | 2012-09-27 | 公開日 | 2013-07-31 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.762 Å) | 主引用文献 | Structural and catalytic characterization of a thermally stable and acid-stable variant of human carbonic anhydrase II containing an engineered disulfide bond. Acta Crystallogr.,Sect.D, 69, 2013
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