2Y5P
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5FWH
| N-terminal FHA domain from EssC a component of the bacterial Type VII secretion apparatus | 分子名称: | ESSC | 著者 | Zoltner, M, Ng, W.M.A.V, Money, J.J, Fyfe, P.K, Kneuper, H, Palmer, T, Hunter, W.N. | 登録日 | 2016-02-17 | 公開日 | 2016-04-06 | 最終更新日 | 2016-10-12 | 実験手法 | X-RAY DIFFRACTION (2.06 Å) | 主引用文献 | Essc: Domain Structures Inform on the Elusive Translocation Channel in the Type Vii Secretion System. Biochem.J., 473, 2016
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2XDS
| Structure of HSP90 with small molecule inhibitor bound | 分子名称: | 1-CHLORO-4-METHYLPHTHALAZINE, DIMETHYL SULFOXIDE, HEAT SHOCK PROTEIN HSP 90-ALPHA | 著者 | Murray, C.W, Carr, M.G, Callaghan, O, Chessari, G, Congreve, M, Cowan, S, Coyle, J.E, Downham, R, Figueroa, E, Frederickson, M, Graham, B, McMenamin, R, OBrien, M.A, Patel, S, Phillips, T.R, Williams, G, Woodhead, A.J, Woolford, A.J.A. | 登録日 | 2010-05-07 | 公開日 | 2010-09-01 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Fragment-Based Drug Discovery Applied to Hsp90. Discovery of Two Lead Series with High Ligand Efficiency. J.Med.Chem., 53, 2010
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5FVL
| Crystal structure of Vps4-Vps20 complex from S.cerevisiae | 分子名称: | VACUOLAR PROTEIN SORTING-ASSOCIATED PROTEIN 20, VACUOLAR PROTEIN SORTING-ASSOCIATED PROTEIN 4 | 著者 | Kojima, R, Obita, T, Onoue, K, Mizuguchi, M. | 登録日 | 2016-02-09 | 公開日 | 2016-04-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.973 Å) | 主引用文献 | Structural Fine-Tuning of Mit Interacting Motif 2 (Mim2) and Allosteric Regulation of Escrt-III by Vps4 in Yeast. J.Mol.Biol., 428, 2016
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5FWS
| Wnt modulator Kremen crystal form I at 1.90A | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, KREMEN PROTEIN 1, ... | 著者 | Zebisch, M, Jackson, V.A, Jones, E.Y. | 登録日 | 2016-02-21 | 公開日 | 2016-07-20 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure of the Dual-Mode Wnt Regulator Kremen1 and Insight Into Ternary Complex Formation with Lrp6 and Dickkopf Structure, 24, 2016
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6Z1S
| Structure of Polyphenol Oxidase (mutant G292N) from Thermothelomyces thermophila | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Dimarogona, M, Nikolaivits, E, Valmas, A, Topakas, E. | 登録日 | 2020-05-14 | 公開日 | 2021-03-24 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Considerations Regarding Activity Determinants of Fungal Polyphenol Oxidases Based on Mutational and Structural Studies. Appl.Environ.Microbiol., 87, 2021
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2XEH
| Structural Determinants for Improved Thermal Stability of Designed Ankyrin Repeat Proteins With a Redesigned C-capping Module. | 分子名称: | NI3C MUT6, SULFATE ION | 著者 | Kramer, M, Wetzel, S.K, Pluckthun, A, Mittl, P, Grutter, M. | 登録日 | 2010-05-14 | 公開日 | 2010-08-18 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | Structural Determinants for Improved Thermal Stability of Designed Ankyrin Repeat Proteins with a Redesigned C-Capping Module. J.Mol.Biol., 404, 2010
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6Z8H
| Crystal structure of Variant Surface Glycoprotein VSG13 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, SULFATE ION, Variant surface glycoprotein MITat 1.13, ... | 著者 | Stebbins, C.E, Hempelmann, A, Van Straaten, M, Zeelen, J. | 登録日 | 2020-06-02 | 公開日 | 2021-03-17 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.38 Å) | 主引用文献 | Structure of trypanosome coat protein VSGsur and function in suramin resistance. Nat Microbiol, 6, 2021
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1JY7
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5K9L
| Beclin 2 CCD N187L mutant homodimer | 分子名称: | Beclin-2 | 著者 | Su, M, Sinha, S. | 登録日 | 2016-06-01 | 公開日 | 2017-03-08 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.52 Å) | 主引用文献 | BECN2 interacts with ATG14 through a metastable coiled-coil to mediate autophagy. Protein Sci., 26, 2017
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5K9X
| Crystal structure of Tryptophan synthase alpha chain from Legionella pneumophila subsp. pneumophila | 分子名称: | Tryptophan synthase alpha chain | 著者 | Chang, C, Hatzos-Skintges, C, Endres, M, ANDERSON, W.F, JOACHIMIAK, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2016-06-01 | 公開日 | 2016-06-15 | 実験手法 | X-RAY DIFFRACTION (2.016 Å) | 主引用文献 | Crystal structure of Tryptophan synthase alpha chain from Legionella pneumophila subsp. pneumophila To Be Published
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2NR1
| TRANSMEMBRANE SEGMENT 2 OF NMDA RECEPTOR NR1, NMR, 10 STRUCTURES | 分子名称: | NR1 M2 | 著者 | Gesell, J.J, Sun, W, Montal, M, Opella, S. | 登録日 | 1997-12-22 | 公開日 | 1998-04-29 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structures of the M2 channel-lining segments from nicotinic acetylcholine and NMDA receptors by NMR spectroscopy. Nat.Struct.Biol., 6, 1999
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5FYW
| Transcription initiation complex structures elucidate DNA opening (OC) | 分子名称: | DNA-DIRECTED RNA POLYMERASE II SUBUNIT RPB1, DNA-DIRECTED RNA POLYMERASE II SUBUNIT RPB11, DNA-DIRECTED RNA POLYMERASE II SUBUNIT RPB2, ... | 著者 | Plaschka, C, Hantsche, M, Dienemann, C, Burzinski, C, Plitzko, J, Cramer, P. | 登録日 | 2016-03-10 | 公開日 | 2016-05-18 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (4.35 Å) | 主引用文献 | Transcription Initiation Complex Structures Elucidate DNA Opening Nature, 533, 2016
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2Y0T
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3WA6
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4FE1
| Improving the Accuracy of Macromolecular Structure Refinement at 7 A Resolution | 分子名称: | 1,2-DIPALMITOYL-PHOSPHATIDYL-GLYCEROLE, 1,2-DISTEAROYL-MONOGALACTOSYL-DIGLYCERIDE, BETA-CAROTENE, ... | 著者 | Fromme, R, Adams, P.D, Fromme, P, Levitt, M, Schroeder, G.F, Brunger, A.T. | 登録日 | 2012-05-29 | 公開日 | 2012-08-15 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (4.9228 Å) | 主引用文献 | Improving the accuracy of macromolecular structure refinement at 7 A resolution. Structure, 20, 2012
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2XP1
| Structure of the tandem SH2 domains from Antonospora locustae transcription elongation factor Spt6 | 分子名称: | CHLORIDE ION, SPT6, SULFATE ION | 著者 | Diebold, M.-L, Koch, M, Cavarelli, J, Romier, C. | 登録日 | 2010-08-24 | 公開日 | 2010-09-29 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Noncanonical Tandem Sh2 Enables Interaction of Elongation Factor Spt6 with RNA Polymerase II. J.Biol.Chem., 285, 2010
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8P0L
| Crystal structure of human O-GlcNAcase in complex with an S-linked CKII peptide | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CYSTEINE, Protein O-GlcNAcase, ... | 著者 | Males, A, Davies, G.J, Calvelo, M, Alteen, M.G, Vocadlo, D.J, Rovira, C. | 登録日 | 2023-05-10 | 公開日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Human O -GlcNAcase Uses a Preactivated Boat-skew Substrate Conformation for Catalysis. Evidence from X-ray Crystallography and QM/MM Metadynamics. Acs Catalysis, 13, 2023
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5JQQ
| Crystal structure of glucosyl-3-phosphoglycerate synthase from Mycobacterium tuberculosis - apo form | 分子名称: | GLYCEROL, Glucosyl-3-phosphoglycerate synthase | 著者 | Albesa-Jove, D, Urresti, S, Gest, P.M, van der Woerd, M, Jackson, M, Guerin, M.E. | 登録日 | 2016-05-05 | 公開日 | 2016-12-21 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structure of glucosyl-3-phosphoglycerate synthase from Mycobacterium tuberculosis - apo form To Be Published
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2XDU
| Structure of HSP90 with small molecule inhibitor bound | 分子名称: | 1-CHLORO-4-METHYLPHTHALAZINE, DIMETHYL SULFOXIDE, HEAT SHOCK PROTEIN HSP 90-ALPHA, ... | 著者 | Murray, C.W, Carr, M.G, Callaghan, O, Chessari, G, Congreve, M, Cowan, S, Coyle, J.E, Downham, R, Figueroa, E, Frederickson, M, Graham, B, McMenamin, R, OBrien, M.A, Patel, S, Phillips, T.R, Williams, G, Woodhead, A.J, Woolford, A.J.A. | 登録日 | 2010-05-07 | 公開日 | 2010-09-01 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Fragment-Based Drug Discovery Applied to Hsp90. Discovery of Two Lead Series with High Ligand Efficiency. J.Med.Chem., 53, 2010
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8P35
| Mutant human titin immunoglobulin-like 21 domain - C3575S | 分子名称: | Titin | 著者 | Martinez-Martin, I, Crousilles, A, Mortensen, S.A, Alegre-Cebollada, J, Wilmanns, M. | 登録日 | 2023-05-17 | 公開日 | 2023-11-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Titin domains with reduced core hydrophobicity cause dilated cardiomyopathy. Cell Rep, 42, 2023
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8P49
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5JRB
| Rad52(1-212) K102A/K133A/E202A mutant | 分子名称: | DNA repair protein RAD52 homolog | 著者 | Saotome, M, Saito, K, Kurumizaka, H, Kagawa, W. | 登録日 | 2016-05-06 | 公開日 | 2016-08-10 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.405 Å) | 主引用文献 | Structure of the human DNA-repair protein RAD52 containing surface mutations. Acta Crystallogr.,Sect.F, 72, 2016
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5FAO
| CTX-M-15 in complex with FPI-1465 | 分子名称: | Beta-lactamase, [[(3~{R},6~{S})-1-methanoyl-6-[[(3~{S})-pyrrolidin-3-yl]oxycarbamoyl]piperidin-3-yl]amino] hydrogen sulfate | 著者 | King, A.M, King, D.T, French, S, Brouillette, E, Asli, A, Alexander, A.N, Vuckovic, M, Maiti, S.N, Parr, T.R, Brown, E.D, Malouin, F, Strynadka, N.C.J, Wright, G.D. | 登録日 | 2015-12-11 | 公開日 | 2016-02-17 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.01 Å) | 主引用文献 | Structural and Kinetic Characterization of Diazabicyclooctanes as Dual Inhibitors of Both Serine-beta-Lactamases and Penicillin-Binding Proteins. Acs Chem.Biol., 11, 2016
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5JRO
| The crystal structure of azoreductase from Yersinia pestis CO92 in its Apo form | 分子名称: | FMN-dependent NADH-azoreductase, GLYCEROL | 著者 | Tan, K, Gu, M, Kwon, K, Anderson, W.F, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2016-05-06 | 公開日 | 2016-06-15 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.54 Å) | 主引用文献 | The crystal structure of azoreductase from Yersinia pestis CO92 in its Apo form To Be Published
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