3D7T
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![BU of 3d7t by Molmil](/molmil-images/mine/3d7t) | Structural basis for the recognition of c-Src by its inactivator Csk | Descriptor: | Proto-oncogene tyrosine-protein kinase Src, STAUROSPORINE, Tyrosine-protein kinase CSK | Authors: | Levinson, N.M, Seeliger, M.A, Cole, P.A, Kuriyan, J. | Deposit date: | 2008-05-21 | Release date: | 2008-08-05 | Last modified: | 2021-10-20 | Method: | X-RAY DIFFRACTION (2.899 Å) | Cite: | Structural basis for the recognition of c-Src by its inactivator Csk. Cell(Cambridge,Mass.), 134, 2008
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3D7U
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![BU of 3d7u by Molmil](/molmil-images/mine/3d7u) | Structural basis for the recognition of c-Src by its inactivator Csk | Descriptor: | Proto-oncogene tyrosine-protein kinase Src, Tyrosine-protein kinase CSK | Authors: | Levinson, N.M, Seeliger, M.A, Cole, P.A, Kuriyan, J. | Deposit date: | 2008-05-21 | Release date: | 2008-08-05 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (4.111 Å) | Cite: | Structural basis for the recognition of c-Src by its inactivator Csk. Cell(Cambridge,Mass.), 134, 2008
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2G2H
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![BU of 2g2h by Molmil](/molmil-images/mine/2g2h) | |
2G2F
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![BU of 2g2f by Molmil](/molmil-images/mine/2g2f) | |
2G1T
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![BU of 2g1t by Molmil](/molmil-images/mine/2g1t) | |
2G2I
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![BU of 2g2i by Molmil](/molmil-images/mine/2g2i) | |
4MXY
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![BU of 4mxy by Molmil](/molmil-images/mine/4mxy) | Src M314L T338M double mutant bound to kinase inhibitor bosutinib | Descriptor: | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile, Proto-oncogene tyrosine-protein kinase Src | Authors: | Levinson, N.M, Boxer, S.G. | Deposit date: | 2013-09-26 | Release date: | 2013-12-25 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.582 Å) | Cite: | A conserved water-mediated hydrogen bond network defines bosutinib's kinase selectivity. Nat.Chem.Biol., 10, 2014
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4MXX
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![BU of 4mxx by Molmil](/molmil-images/mine/4mxx) | Human Src A403T mutant bound to kinase inhibitor bosutinib | Descriptor: | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile, Proto-oncogene tyrosine-protein kinase Src | Authors: | Levinson, N.M, Boxer, S.G. | Deposit date: | 2013-09-26 | Release date: | 2013-12-04 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | A conserved water-mediated hydrogen bond network defines bosutinib's kinase selectivity. Nat.Chem.Biol., 10, 2014
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4MXZ
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![BU of 4mxz by Molmil](/molmil-images/mine/4mxz) | Src M314L T338M double mutant bound to kinase inhibitor bosutinib | Descriptor: | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile, Proto-oncogene tyrosine-protein kinase Src | Authors: | Levinson, N.M, Boxer, S.G. | Deposit date: | 2013-09-26 | Release date: | 2013-12-04 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.582 Å) | Cite: | A conserved water-mediated hydrogen bond network defines bosutinib's kinase selectivity. Nat.Chem.Biol., 10, 2014
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4MXO
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![BU of 4mxo by Molmil](/molmil-images/mine/4mxo) | human Src kinase bound to kinase inhibitor bosutinib | Descriptor: | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile, Proto-oncogene tyrosine-protein kinase Src | Authors: | Levinson, N.M, Boxer, S.G. | Deposit date: | 2013-09-26 | Release date: | 2013-12-04 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.105 Å) | Cite: | A conserved water-mediated hydrogen bond network defines bosutinib's kinase selectivity. Nat.Chem.Biol., 10, 2014
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3UE4
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![BU of 3ue4 by Molmil](/molmil-images/mine/3ue4) | |