3D7T
| Structural basis for the recognition of c-Src by its inactivator Csk | 分子名称: | Proto-oncogene tyrosine-protein kinase Src, STAUROSPORINE, Tyrosine-protein kinase CSK | 著者 | Levinson, N.M, Seeliger, M.A, Cole, P.A, Kuriyan, J. | 登録日 | 2008-05-21 | 公開日 | 2008-08-05 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (2.899 Å) | 主引用文献 | Structural basis for the recognition of c-Src by its inactivator Csk. Cell(Cambridge,Mass.), 134, 2008
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3D7U
| Structural basis for the recognition of c-Src by its inactivator Csk | 分子名称: | Proto-oncogene tyrosine-protein kinase Src, Tyrosine-protein kinase CSK | 著者 | Levinson, N.M, Seeliger, M.A, Cole, P.A, Kuriyan, J. | 登録日 | 2008-05-21 | 公開日 | 2008-08-05 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (4.111 Å) | 主引用文献 | Structural basis for the recognition of c-Src by its inactivator Csk. Cell(Cambridge,Mass.), 134, 2008
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4MXX
| Human Src A403T mutant bound to kinase inhibitor bosutinib | 分子名称: | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile, Proto-oncogene tyrosine-protein kinase Src | 著者 | Levinson, N.M, Boxer, S.G. | 登録日 | 2013-09-26 | 公開日 | 2013-12-04 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | A conserved water-mediated hydrogen bond network defines bosutinib's kinase selectivity. Nat.Chem.Biol., 10, 2014
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4MXZ
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4MXO
| human Src kinase bound to kinase inhibitor bosutinib | 分子名称: | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile, Proto-oncogene tyrosine-protein kinase Src | 著者 | Levinson, N.M, Boxer, S.G. | 登録日 | 2013-09-26 | 公開日 | 2013-12-04 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.105 Å) | 主引用文献 | A conserved water-mediated hydrogen bond network defines bosutinib's kinase selectivity. Nat.Chem.Biol., 10, 2014
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4MXY
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2G2H
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2G2F
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2G1T
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2G2I
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3UE4
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