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PDB: 16 件

4GUX
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BU of 4gux by Molmil
Crystal structure of trypsin:MCoTi-II complex
分子名称: ACETATE ION, CALCIUM ION, Cationic trypsin, ...
著者King, G.J, Daly, N.L, Thorstholm, L, Greenwood, K.P, Rosengren, K.J, Heras, B, Craik, D.J, Martin, J.L.
登録日2012-08-30
公開日2013-09-04
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.803 Å)
主引用文献Structural insights into the role of the cyclic backbone in a squash trypsin inhibitor
J.Biol.Chem., 288, 2013
6VXY
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BU of 6vxy by Molmil
Triazole bridged SFTI1 inhibitor in complex with beta-trypsin
分子名称: 1-methyl-1H-1,2,3-triazole, CALCIUM ION, Cationic trypsin, ...
著者White, A.M, King, G.J, Durek, T, Craik, D.J.
登録日2020-02-25
公開日2020-07-01
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.398 Å)
主引用文献Application and Structural Analysis of Triazole-Bridged Disulfide Mimetics in Cyclic Peptides.
Angew.Chem.Int.Ed.Engl., 2020
4TTO
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BU of 4tto by Molmil
Quasi-racemic structure of [V25A] kalata B1
分子名称: D-kalata B1, Kalata-B1
著者Wang, C.K, King, G.J, Craik, D.J.
登録日2014-06-22
公開日2014-09-10
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.3002 Å)
主引用文献Racemic and Quasi-Racemic X-ray Structures of Cyclic Disulfide-Rich Peptide Drug Scaffolds.
Angew.Chem.Int.Ed.Engl., 53, 2014
4TTM
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BU of 4ttm by Molmil
Racemic structure of kalata B1 (kB1)
分子名称: D-kalata B1, Kalata-B1
著者Wang, C.K, King, G.J, Craik, D.J.
登録日2014-06-22
公開日2014-09-10
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9001 Å)
主引用文献Racemic and Quasi-Racemic X-ray Structures of Cyclic Disulfide-Rich Peptide Drug Scaffolds.
Angew.Chem.Int.Ed.Engl., 53, 2014
4TTL
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BU of 4ttl by Molmil
Racemic structure of cyclic Vc1.1 (cVc1.1-1)
分子名称: Alpha-conotoxin Vc1A
著者Wang, C.K, King, G.J, Craik, D.J.
登録日2014-06-22
公開日2014-09-10
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.7004 Å)
主引用文献Racemic and Quasi-Racemic X-ray Structures of Cyclic Disulfide-Rich Peptide Drug Scaffolds.
Angew.Chem.Int.Ed.Engl., 53, 2014
4TTK
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BU of 4ttk by Molmil
Racemic structure of Sunflower Trypsin Inhibitor-1 (SFTI-1)
分子名称: Sunflower Trypsin Inhibitor-1 (SFTI-1) (D-form)
著者Wang, C.K, King, G.J, Craik, D.J.
登録日2014-06-22
公開日2014-09-10
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.2502 Å)
主引用文献Racemic and Quasi-Racemic X-ray Structures of Cyclic Disulfide-Rich Peptide Drug Scaffolds.
Angew.Chem.Int.Ed.Engl., 53, 2014
4TTN
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BU of 4ttn by Molmil
Quasi-racemic structure of [G6A]kalata B1
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, D-kalata B1, Kalata-B1
著者Wang, C.K, King, G.J, Craik, D.J.
登録日2014-06-22
公開日2014-09-10
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.2507 Å)
主引用文献Racemic and Quasi-Racemic X-ray Structures of Cyclic Disulfide-Rich Peptide Drug Scaffolds.
Angew.Chem.Int.Ed.Engl., 53, 2014
5INZ
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BU of 5inz by Molmil
Racemic structure of baboon theta defensin-2
分子名称: 1,2-ETHANEDIOL, SULFATE ION, Theta defensin-2, ...
著者Wang, C.K, King, G.J, Conibear, A.C, Ramos, M.C, Craik, D.J.
登録日2016-03-08
公開日2016-04-27
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.447 Å)
主引用文献Mirror Images of Antimicrobial Peptides Provide Reflections on Their Functions and Amyloidogenic Properties.
J.Am.Chem.Soc., 138, 2016
4GXZ
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BU of 4gxz by Molmil
Crystal structure of a periplasmic thioredoxin-like protein from Salmonella enterica serovar Typhimurium
分子名称: Suppression of copper sensitivity protein
著者Shepherd, M, Heras, B, King, G.J, Argente, M.P, Achard, M.E.S, King, N.P, McEwan, A.G, Schembri, M.A.
登録日2012-09-04
公開日2013-07-17
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.04 Å)
主引用文献Structural and functional characterization of ScsC, a periplasmic thioredoxin-like protein from Salmonella enterica serovar Typhimurium
Antioxid Redox Signal, 19, 2013
6U22
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BU of 6u22 by Molmil
Crystal structure of SFTI-triazole inhibitor in complex with beta-trypsin
分子名称: 1-methyl-1H-1,2,3-triazole, CALCIUM ION, Cationic trypsin, ...
著者White, A.M, King, G.J, Durek, T, Craik, D.J.
登録日2019-08-19
公開日2020-07-01
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Application and Structural Analysis of Triazole-Bridged Disulfide Mimetics in Cyclic Peptides.
Angew.Chem.Int.Ed.Engl., 59, 2020
4H8S
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BU of 4h8s by Molmil
Crystal structure of human APPL2BARPH domain
分子名称: DCC-interacting protein 13-beta
著者Martin, J.L, King, G.J.
登録日2012-09-23
公開日2012-10-17
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Membrane Curvature Protein Exhibits Interdomain Flexibility and Binds a Small GTPase.
J.Biol.Chem., 287, 2012
6DL1
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BU of 6dl1 by Molmil
Racemic structure of jatrophidin, an orbitide from Jatropha curcas
分子名称: jatrophidin
著者Wang, C.K, King, G.J, Ramalho, S.D.
登録日2018-05-31
公開日2018-11-14
最終更新日2020-01-01
実験手法X-RAY DIFFRACTION (1.029 Å)
主引用文献Synthesis, Racemic X-ray Crystallographic, and Permeability Studies of Bioactive Orbitides from Jatropha Species.
J. Nat. Prod., 81, 2018
6DL0
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BU of 6dl0 by Molmil
Crystal structure of pohlianin C, an orbitide from Jatropha pohliana
分子名称: pohlianin C
著者Wang, C.K, King, G.J, Ramalho, S.D.
登録日2018-05-31
公開日2018-11-07
最終更新日2023-07-26
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Synthesis, Racemic X-ray Crystallographic, and Permeability Studies of Bioactive Orbitides from Jatropha Species.
J. Nat. Prod., 81, 2018
6DKZ
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BU of 6dkz by Molmil
Racemic structure of ribifolin, an orbitide from Jatropha ribifolia
分子名称: ribifolin
著者Wang, C.K, King, G.J, Ramalho, S.D.
登録日2018-05-31
公開日2018-11-14
最終更新日2020-01-01
実験手法X-RAY DIFFRACTION (0.99 Å)
主引用文献Synthesis, Racemic X-ray Crystallographic, and Permeability Studies of Bioactive Orbitides from Jatropha Species.
J. Nat. Prod., 81, 2018
6DKY
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BU of 6dky by Molmil
Crystal structure of ribifolin, an orbitide from Jatropha ribifolia
分子名称: ILE-LEU-GLY-SER-ILE-ILE-LEU-GLY
著者Wang, C.K, Ramalho, S.D, King, G.J, Craik, D.J.
登録日2018-05-31
公開日2018-11-07
最終更新日2020-01-01
実験手法X-RAY DIFFRACTION (1.239 Å)
主引用文献Synthesis, Racemic X-ray Crystallographic, and Permeability Studies of Bioactive Orbitides from Jatropha Species.
J. Nat. Prod., 81, 2018
6EEZ
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BU of 6eez by Molmil
Crystal Structure of the thiol-disulfide exchange protein alpha-DsbA2 from Wolbachia pipientis
分子名称: DsbA-like disulfide oxidoreductase
著者Walden, P.M, Lakshmanane, P, King, G.J, Martin, J.L.
登録日2018-08-15
公開日2019-04-17
最終更新日2020-01-01
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献The atypical thiol-disulfide exchange protein alpha-DsbA2 from Wolbachia pipientis is a homotrimeric disulfide isomerase.
Acta Crystallogr D Struct Biol, 75, 2019

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件を2024-07-24に公開中

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