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PDB: 54 件

4IU8
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Crystal structure of a membrane transporter (selenomethionine derivative)
分子名称: NITRATE ION, Nitrite extrusion protein 2
著者Yan, H, Huang, W, Yan, C, Gong, X, Jiang, S, Zhao, Y, Wang, J, Shi, Y.
登録日2013-01-20
公開日2013-04-17
実験手法X-RAY DIFFRACTION (3.11 Å)
主引用文献Structure and mechanism of a nitrate transporter.
Cell Rep, 3, 2013
7DY7
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Discovery of Novel Small-molecule Inhibitors of PD-1/PD-L1 Axis that Promotes PD-L1 Internalization and Degradation
分子名称: 2-[[3-[[5-(2-methyl-3-phenyl-phenyl)-1,3,4-oxadiazol-2-yl]amino]phenyl]methylamino]ethanol, Programmed cell death 1 ligand 1
著者Cheng, Y, Wang, T.Y, Lu, M.L, Jiang, S, Xiao, Y.B.
登録日2021-01-20
公開日2022-01-26
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.42 Å)
主引用文献Discovery of Small-Molecule Inhibitors of the PD-1/PD-L1 Axis That Promote PD-L1 Internalization and Degradation.
J.Med.Chem., 65, 2022
2JNR
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Discovery and optimization of a natural HIV-1 entry inhibitor targeting the gp41 fusion peptide
分子名称: ENV polyprotein, VIR165
著者Munch, J, Standker, L, Adermann, K, Schulz, A, Pohlmann, S, Chaipan, C, Biet, T, Peters, T, Meyer, B, Wilhelm, D, Lu, H, Jing, W, Jiang, S, Forssmann, W, Kirchhoff, F.
登録日2007-02-01
公開日2007-05-08
最終更新日2023-12-20
実験手法SOLUTION NMR
主引用文献Discovery and Optimization of a Natural HIV-1 Entry Inhibitor Targeting the gp41 Fusion Peptide.
Cell(Cambridge,Mass.), 129, 2007
7XTP
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eIF4E in Complex with a Disulphide-Free Autonomous VH Domain
分子名称: Eukaryotic translation initiation factor 4E, VH-S4ss, [[(2R,3S,4R,5R)-5-(6-AMINO-3-METHYL-4-OXO-5H-IMIDAZO[4,5-C]PYRIDIN-1-YL)-3,4-DIHYDROXY-OXOLAN-2-YL]METHOXY-HYDROXY-PHOSPHORYL] PHOSPHONO HYDROGEN PHOSPHATE
著者Brown, C.J, Frosi, Y, Jiang, S, Lin, Y.C.
登録日2022-05-17
公開日2022-07-27
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.828 Å)
主引用文献Engineering an autonomous VH domain to modulate intracellular pathways and to interrogate the eIF4F complex.
Nat Commun, 13, 2022
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