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PDB: 42507 件

1I94
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CRYSTAL STRUCTURES OF THE SMALL RIBOSOMAL SUBUNIT WITH TETRACYCLINE, EDEINE AND IF3
分子名称: 16S RRNA, 30S RIBOSOMAL PROTEIN S10, 30S RIBOSOMAL PROTEIN S11, ...
著者Pioletti, M, Schluenzen, F, Harms, J, Zarivach, R, Gluehmann, M, Avila, H, Bartels, H, Jacobi, C, Hartsch, T, Yonath, A, Franceschi, F.
登録日2001-03-18
公開日2001-04-12
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Crystal structures of complexes of the small ribosomal subunit with tetracycline, edeine and IF3.
EMBO J., 20, 2001
8DVN
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Crystal structure of LRP6 E3E4 in complex with disulfide constrained peptide E3.10
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Thakur, A.K, Liau, N.P.D, Sudhamsu, J, Hannoush, R.N.
登録日2022-07-29
公開日2023-03-29
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.53 Å)
主引用文献Synthetic Multivalent Disulfide-Constrained Peptide Agonists Potentiate Wnt1/ beta-Catenin Signaling via LRP6 Coreceptor Clustering.
Acs Chem.Biol., 18, 2023
1XX5
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Crystal Structure of Natrin from Naja atra snake venom
分子名称: ETHANOL, Natrin 1
著者Wang, J, Shen, B, Lou, X.H, Guo, M, Teng, M.K, Niu, L.W.
登録日2004-11-04
公開日2005-06-14
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Blocking effect and crystal structure of natrin toxin, a cysteine-rich secretory protein from Naja atra venom that targets the BKCa channel
Biochemistry, 44, 2005
8DVL
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Crystal structure of LRP6 E3E4 in complex with disulfide constrained peptide E3.18
分子名称: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Thakur, A.K, Liau, N.P.D, Sudhamsu, J, Hannoush, R.N.
登録日2022-07-29
公開日2023-03-29
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Synthetic Multivalent Disulfide-Constrained Peptide Agonists Potentiate Wnt1/ beta-Catenin Signaling via LRP6 Coreceptor Clustering.
Acs Chem.Biol., 18, 2023
8E7Y
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RsTSPO A138F with two heme bound
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, PROTOPORPHYRIN IX CONTAINING FE, Tryptophan-rich sensory protein
著者Liu, J, Hiser, C, Li, F, Garavito, R, Ferguson-Miller, S.
登録日2022-08-25
公開日2023-03-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献New TSPO Crystal Structures of Mutant and Heme-Bound Forms with Altered Flexibility, Ligand Binding, and Porphyrin Degradation Activity.
Biochemistry, 62, 2023
8DVM
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Crystal structure of LRP6 E3E4 in complex with disulfide constrained peptide E3.6
分子名称: 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Thakur, A.K, Liau, N.P.D, Sudhamsu, J, Hannoush, R.N.
登録日2022-07-29
公開日2023-03-29
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Synthetic Multivalent Disulfide-Constrained Peptide Agonists Potentiate Wnt1/ beta-Catenin Signaling via LRP6 Coreceptor Clustering.
Acs Chem.Biol., 18, 2023
5HXH
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Structural mechanisms of extracellular ion exchange and induced binding-site occlusion in the sodium-calcium exchanger NCX_Mj soaked with zero Na+ and Ca2+
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, CALCIUM ION, PENTADECANE, ...
著者Liao, J, Jiang, Y.X, Faraldo-Gomez, J.D.
登録日2016-01-30
公開日2016-05-11
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.804 Å)
主引用文献Mechanism of extracellular ion exchange and binding-site occlusion in a sodium/calcium exchanger
Nat.Struct.Mol.Biol., 23, 2016
1I9B
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X-RAY STRUCTURE OF ACETYLCHOLINE BINDING PROTEIN (ACHBP)
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ACETYLCHOLINE BINDING PROTEIN, CALCIUM ION
著者Brejc, K, van Dijk, W.J, Klaassen, R, Schuurmans, M, van der Oost, J, Smit, A.B, Sixma, T.K.
登録日2001-03-18
公開日2001-05-16
最終更新日2018-03-07
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors.
Nature, 411, 2001
1XGA
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ALPHA CONOTOXIN GI: 2-7;3-13 (NATIVE) DISULFIDE BOND ISOMER, NMR, 35 STRUCTURES
分子名称: ALPHA-CONOTOXIN GI
著者Gehrmann, J, Alewood, P.F, Craik, D.J.
登録日1998-01-18
公開日1999-02-16
最終更新日2024-06-05
実験手法SOLUTION NMR
主引用文献Structure determination of the three disulfide bond isomers of alpha-conotoxin GI: a model for the role of disulfide bonds in structural stability.
J.Mol.Biol., 278, 1998
8E7W
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RsTSPO A139T with Heme
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, (2S)-3-{[{[(2S)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-2-[(6E)-HEXADEC-6-ENOYLOXY]PROPYL (8E)-OCTADEC-8-ENOATE, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Liu, J, Hiser, C, Li, F, Garavito, R, Ferguson-Miller, S.
登録日2022-08-25
公開日2023-03-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献New TSPO Crystal Structures of Mutant and Heme-Bound Forms with Altered Flexibility, Ligand Binding, and Porphyrin Degradation Activity.
Biochemistry, 62, 2023
8E84
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Human PCNA mutant- C148S
分子名称: Proliferating cell nuclear antigen
著者Magrino, J, Page, B, Gaubitz, C, Kelch, B.A.
登録日2022-08-25
公開日2023-04-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献A thermosensitive PCNA allele underlies an ataxia-telangiectasia-like disorder.
J.Biol.Chem., 299, 2023
8EBU
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XPC release from Core7-XPA-DNA (Cy5)
分子名称: DNA repair protein complementing XP-A cells, DNA repair protein complementing XP-C cells, DNA1, ...
著者Kim, J, Yang, W.
登録日2022-08-31
公開日2023-04-19
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Lesion recognition by XPC, TFIIH and XPA in DNA excision repair.
Nature, 617, 2023
8EBS
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Initial DNA-lesion (Cy5) binding by XPC and TFIIH
分子名称: CALCIUM ION, Centrin-2, DNA, ...
著者Kim, J, Yang, W.
登録日2022-08-31
公開日2023-04-19
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Lesion recognition by XPC, TFIIH and XPA in DNA excision repair.
Nature, 617, 2023
8EBT
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XPA repositioning Core7 of TFIIH relative to XPC-DNA lesion (Cy5)
分子名称: CALCIUM ION, Centrin-2, DNA, ...
著者Kim, J, Yang, W.
登録日2022-08-31
公開日2023-04-19
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Lesion recognition by XPC, TFIIH and XPA in DNA excision repair.
Nature, 617, 2023
8EBY
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XPC release from Core7-XPA-DNA (AP)
分子名称: DNA, DNA repair protein complementing XP-A cells, DNA repair protein complementing XP-C cells, ...
著者Kim, J, Yang, W.
登録日2022-08-31
公開日2023-04-19
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Lesion recognition by XPC, TFIIH and XPA in DNA excision repair.
Nature, 617, 2023
1L8F
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Structure of 20K-endoglucanase from Melanocarpus albomyces at 1.8 A
分子名称: Endoglucanase
著者Valjakka, J, Rouvinen, J.
登録日2002-03-20
公開日2003-04-01
最終更新日2018-04-04
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure of 20K endoglucanase from Melanocarpus albomyces at 1.8 A resolution.
Acta Crystallogr.,Sect.D, 59, 2003
8DV3
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Crystal structure of human CD1b presenting Phosphatidylinositol C34:1
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOINOSITOL, 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Farquhar, R, Rossjohn, J, Shahine, A.
登録日2022-07-28
公開日2023-04-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献alpha beta T-cell receptor recognition of self-phosphatidylinositol presented by CD1b.
J.Biol.Chem., 299, 2023
8EBV
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Initial DNA-lesion (AP) binding by XPC and TFIIH complex 1
分子名称: CALCIUM ION, Centrin-2, DNA, ...
著者Kim, J, Yang, W.
登録日2022-08-31
公開日2023-04-19
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (7.1 Å)
主引用文献Lesion recognition by XPC, TFIIH and XPA in DNA excision repair.
Nature, 617, 2023
6MEP
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Crystal structure of the catalytic domain of the proto-oncogene tyrosine-protein kinase MER in complex with inhibitor UNC3437
分子名称: CHLORIDE ION, MAGNESIUM ION, Tyrosine-protein kinase Mer, ...
著者Da, C, Zhang, D, Stashko, M.A, Cheng, A, Hunter, D, Norris-Drouin, J, Graves, L, Machius, M, Miley, M.J, DeRyckere, D, Earp, H.S, Graham, D.K, Frye, S.V, Wang, X, Kireev, D.
登録日2018-09-06
公開日2019-09-11
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.893 Å)
主引用文献Data-Driven Construction of Antitumor Agents with Controlled Polypharmacology.
J.Am.Chem.Soc., 141, 2019
8DV4
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Crystal structure of the BC8B TCR-CD1b-PI complex
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOINOSITOL, 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Farquhar, R, Rossjohn, J, Shahine, A.
登録日2022-07-28
公開日2023-04-19
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献alpha beta T-cell receptor recognition of self-phosphatidylinositol presented by CD1b.
J.Biol.Chem., 299, 2023
8EBW
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Initial DNA-lesion (AP) binding by XPC and TFIIH complex2
分子名称: CALCIUM ION, Centrin-2, DNA, ...
著者Kim, J, Yang, W.
登録日2022-08-31
公開日2023-04-19
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (5.6 Å)
主引用文献Lesion recognition by XPC, TFIIH and XPA in DNA excision repair.
Nature, 617, 2023
8EBX
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XPA repositioning Core7 of TFIIH relative to XPC-DNA lesion (AP)
分子名称: CALCIUM ION, Centrin-2, DNA, ...
著者Kim, J, Yang, W.
登録日2022-08-31
公開日2023-04-19
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Lesion recognition by XPC, TFIIH and XPA in DNA excision repair.
Nature, 617, 2023
6LKE
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in meso full-length rat KMO in complex with an inhibitor identified via DNA-encoded chemical library screening
分子名称: 4-chloranyl-2-[[5-chloranyl-2-(5-methoxy-1,3-dihydroisoindol-2-yl)-1,3-thiazol-4-yl]carbonyl-methyl-amino]-5-fluoranyl-benzoic acid, CHLORIDE ION, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Mimasu, S, Yamagishi, H, Kiyohara, M, Hupp, D.C, Liu, J, Kakefuda, K, Okuda, T.
登録日2019-12-19
公開日2020-12-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Full-length in meso structure and mechanism of rat kynurenine 3-monooxygenase inhibition.
Commun Biol, 4, 2021
8E0P
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Crystal structure of mouse APCDD1 in fusion with engineered MBP
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3-[BENZYL(DIMETHYL)AMMONIO]PROPANE-1-SULFONATE, CHLORIDE ION, ...
著者Hsieh, F.L, Chang, T.H, Gabelli, S.B, Nathans, J.
登録日2022-08-09
公開日2023-05-03
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献Structure of WNT inhibitor adenomatosis polyposis coli down-regulated 1 (APCDD1), a cell-surface lipid-binding protein.
Proc.Natl.Acad.Sci.USA, 120, 2023
4ABB
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Fragments bound to bovine trypsin for the SAMPL challenge
分子名称: 1,2-ETHANEDIOL, 1-(1-BENZOTHIOPHEN-3-YL)METHANAMINE, CALCIUM ION, ...
著者Newman, J, Peat, T.S.
登録日2011-12-08
公開日2012-02-08
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献The Dingo Dataset: A Comprehensive Set of Data for the Sampl Challenge.
J.Comput.Aided Mol.Des., 26, 2012

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件を2024-08-14に公開中

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