3TBH
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3ZKY
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![BU of 3zky by Molmil](/molmil-images/mine/3zky) | Isopenicillin N synthase with substrate analogue AhCmC | 分子名称: | FE (III) ION, GLYCEROL, ISOPENICILLIN N SYNTHASE, ... | 著者 | Daruzzaman, A, Clifton, I.J, Rutledge, P.J. | 登録日 | 2013-01-25 | 公開日 | 2013-03-20 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | The Interaction of Isopenicillin N Synthase with Homologated Substrate Analogues Delta-(L-Alpha-Aminoadipoyl)-L-Homocysteinyl-D-Xaa Characterised by Protein Crystallography. Chembiochem, 14, 2013
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3ZLJ
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![BU of 3zlj by Molmil](/molmil-images/mine/3zlj) | CRYSTAL STRUCTURE OF FULL-LENGTH E.COLI DNA MISMATCH REPAIR PROTEIN MUTS D835R MUTANT IN COMPLEX WITH GT MISMATCHED DNA | 分子名称: | 5'-D(*AP*GP*CP*TP*GP*CP*CP*AP*GP*GP*CP*AP*CP*CP *AP*GP*TP*GP*TP*CP*AP)-3', 5'-D(*TP*GP*AP*CP*AP*CP*TP*GP*GP*TP*GP*CP*TP*TP *GP*GP*CP*AP*GP*CP*TP)-3', DNA MISMATCH REPAIR PROTEIN MUTS | 著者 | Groothuizen, F.S, Fish, A, Petoukhov, M.V, Reumer, A, Manelyte, L, Winterwerp, H.H.K, Marinus, M.G, Lebbink, J.H.G, Svergun, D.I, Friedhoff, P, Sixma, T.K. | 登録日 | 2013-02-01 | 公開日 | 2013-07-17 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Using Stable Muts Dimers and Tetramers to Quantitatively Analyze DNA Mismatch Recognition and Sliding Clamp Formation. Nucleic Acids Res., 41, 2013
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3SOP
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![BU of 3sop by Molmil](/molmil-images/mine/3sop) | Crystal Structure Of Human Septin 3 GTPase Domain | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Neuronal-specific septin-3 | 著者 | Marques, I.A, Macedo, J.N.A, Pereira, H.M, Valadares, N.F, Araujo, A.P.U, Garratt, R.C. | 登録日 | 2011-06-30 | 公開日 | 2012-11-28 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.885 Å) | 主引用文献 | The structure and properties of septin 3: a possible missing link in septin filament formation. Biochem.J., 450, 2013
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3UTC
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![BU of 3utc by Molmil](/molmil-images/mine/3utc) | Ec_IspH in complex with (E)-4-hydroxybut-3-enyl diphosphate | 分子名称: | (3E)-4-hydroxybut-3-en-1-yl trihydrogen diphosphate, 4-hydroxy-3-methylbut-2-enyl diphosphate reductase, IRON/SULFUR CLUSTER | 著者 | Span, I, Wang, K, Wang, W, Zhang, Y, Bacher, A, Eisenreich, W, Li, K, Schulz, C, Oldfield, E, Groll, M. | 登録日 | 2011-11-25 | 公開日 | 2012-09-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Discovery of acetylene hydratase activity of the iron-sulphur protein IspH. Nat Commun, 3, 2012
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3T4P
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3TEB
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![BU of 3teb by Molmil](/molmil-images/mine/3teb) | endonuclease/exonuclease/phosphatase family protein from Leptotrichia buccalis C-1013-b | 分子名称: | Endonuclease/exonuclease/phosphatase, MAGNESIUM ION | 著者 | Chang, C, Bigelow, L, Muniez, I, Bearden, J, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2011-08-12 | 公開日 | 2011-08-31 | 実験手法 | X-RAY DIFFRACTION (2.99 Å) | 主引用文献 | Crystal structure of endonuclease/exonuclease/phosphatase family protein from Leptotrichia buccalis C-1013-b To be Published
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3UVH
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![BU of 3uvh by Molmil](/molmil-images/mine/3uvh) | Crystal Structure Analysis of E81M mutant of human CLIC1 | 分子名称: | Chloride intracellular channel protein 1 | 著者 | Fanucchi, S, Achilonu, I.A, Fernandes, M.A, Legg-E'Silva, D.A, Stoychev, S.H, Dirr, H.W. | 登録日 | 2011-11-30 | 公開日 | 2011-12-14 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | Crystal Structure Analysis of E81M mutant of human CLIC1 To be Published
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3RXS
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![BU of 3rxs by Molmil](/molmil-images/mine/3rxs) | Crystal structure of Trypsin complexed with (3-methoxyphenyl)methanamine (F04 and A06, cocktail experiment) | 分子名称: | 1-(3-methoxyphenyl)methanamine, CALCIUM ION, Cationic trypsin, ... | 著者 | Yamane, J, Yao, M, Zhou, Y, Tanaka, I. | 登録日 | 2011-05-10 | 公開日 | 2011-08-24 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | In-crystal affinity ranking of fragment hit compounds reveals a relationship with their inhibitory activities J.Appl.Crystallogr., 44, 2011
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3ZII
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![BU of 3zii by Molmil](/molmil-images/mine/3zii) | Bacillus subtilis SepF G109K, C-terminal domain | 分子名称: | CELL DIVISION PROTEIN SEPF | 著者 | Duman, R, Ishikawa, S, Celik, I, Ogasawara, N, Lowe, J, Hamoen, L.W. | 登録日 | 2013-01-09 | 公開日 | 2013-11-27 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural and Genetic Analyses Reveal the Protein Sepf as a New Membrane Anchor for the Z Ring. Proc.Natl.Acad.Sci.USA, 110, 2013
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3RXE
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![BU of 3rxe by Molmil](/molmil-images/mine/3rxe) | Crystal structure of Trypsin complexed with benzamide | 分子名称: | BENZAMIDINE, CALCIUM ION, Cationic trypsin, ... | 著者 | Yamane, J, Yao, M, Zhou, Y, Tanaka, I. | 登録日 | 2011-05-10 | 公開日 | 2011-08-24 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | In-crystal affinity ranking of fragment hit compounds reveals a relationship with their inhibitory activities J.Appl.Crystallogr., 44, 2011
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3S0F
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![BU of 3s0f by Molmil](/molmil-images/mine/3s0f) | Apis mellifera OBP14 native apo, crystal form 2 | 分子名称: | OBP14 | 著者 | Spinelli, S, Lagarde, A, Iovinella, I, Tegoni, M, Pelosi, P, Cambillau, C. | 登録日 | 2011-05-13 | 公開日 | 2011-11-30 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Crystal structure of Apis mellifera OBP14, a C-minus odorant-binding protein, and its complexes with odorant molecules. Insect Biochem.Mol.Biol., 42, 2012
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3ZW3
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![BU of 3zw3 by Molmil](/molmil-images/mine/3zw3) | Fragment based discovery of a novel and selective PI3 Kinase inhibitor | 分子名称: | N-{6-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]imidazo[1,2-a]pyridin-2-yl}acetamide, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT GAMMA ISOFORM | 著者 | Brown, D.G, Hughes, S.J, Milan, D.S, Kilty, I.C, Lewthwaite, R.A, Mathias, J.P, O'Reilly, M.A, Pannifer, A, Phelan, A, Baldock, D.A. | 登録日 | 2011-07-28 | 公開日 | 2011-09-28 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Fragment based discovery of a novel and selective PI3 kinase inhibitor. Bioorg. Med. Chem. Lett., 21, 2011
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3ZVV
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![BU of 3zvv by Molmil](/molmil-images/mine/3zvv) | Fragment Bound to PI3Kinase gamma | 分子名称: | 5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-amine, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT GAMMA ISOFORM | 著者 | Hughes, S.J, Milan, D.S, Kilty, I.C, Lewthwaite, R.A, Mathias, J.P, O'Reilly, M.A, Phelan, A, Baldock, D.A, Brown, D.G. | 登録日 | 2011-07-27 | 公開日 | 2011-09-28 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Fragment based discovery of a novel and selective PI3 kinase inhibitor. Bioorg. Med. Chem. Lett., 21, 2011
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4A3O
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![BU of 4a3o by Molmil](/molmil-images/mine/4a3o) | Crystal structure of the USP15 DUSP-UBL monomer | 分子名称: | GLYCEROL, UBIQUITIN CARBOXYL-TERMINAL HYDROLASE 15 | 著者 | Elliott, P.R, Liu, H, Pastok, M.W, Grossmann, G.J, Rigden, D.J, Clague, M.J, Urbe, S, Barsukov, I.L. | 登録日 | 2011-10-03 | 公開日 | 2011-11-16 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural Variability of the Ubiquitin Specific Protease Dusp-Ubl Double Domains. FEBS Lett., 585, 2011
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3SJZ
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![BU of 3sjz by Molmil](/molmil-images/mine/3sjz) | The structure of aIF2gamma subunit delta 41-45 from archaeon Sulfolobus solfataricus complexed with GDP and GDPNP | 分子名称: | BETA-MERCAPTOETHANOL, GUANOSINE-5'-DIPHOSPHATE, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, ... | 著者 | Arkhipova, V.I, Lazopulo, S.M, Lazopulo, A.M, Nikonov, O.S, Stolboushkina, E.A, Gabdoulkhakov, A.G, Garber, M.B, Nikonov, S.V. | 登録日 | 2011-06-22 | 公開日 | 2012-07-04 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | HOLD FOR PUBLICATION To be Published
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3SM8
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3X0Q
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![BU of 3x0q by Molmil](/molmil-images/mine/3x0q) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ESMM-state at reaction time of 20 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.14 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X06
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![BU of 3x06 by Molmil](/molmil-images/mine/3x06) | Crystal structure of PIP4KIIBETA T201M complex with GMP | 分子名称: | GUANOSINE-5'-MONOPHOSPHATE, Phosphatidylinositol 5-phosphate 4-kinase type-2 beta | 著者 | Takeuchi, K, Lo, Y.H, Sumita, K, Senda, M, Terakawa, J, Dimitoris, A, Locasale, J.W, Sasaki, M, Yoshino, H, Zhang, Y, Kahoud, E.R, Takano, T, Yokota, T, Emerling, B, Asara, J.A, Ishida, T, Shimada, I, Daikoku, T, Cantley, L.C, Senda, T, Sasaki, A.T. | 登録日 | 2014-10-09 | 公開日 | 2015-10-14 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | The Lipid Kinase PI5P4K beta Is an Intracellular GTP Sensor for Metabolism and Tumorigenesis Mol.Cell, 61, 2016
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3X2O
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![BU of 3x2o by Molmil](/molmil-images/mine/3x2o) | Neutron and X-ray joint refined structure of PcCel45A apo form at 298K. | 分子名称: | Endoglucanase V-like protein | 著者 | Nakamura, A, Ishida, T, Kusaka, K, Yamada, T, Tanaka, I, Niimura, N, Samejima, M, Igarashi, K. | 登録日 | 2014-12-22 | 公開日 | 2015-10-07 | 最終更新日 | 2019-12-18 | 実験手法 | NEUTRON DIFFRACTION (1.5 Å), X-RAY DIFFRACTION | 主引用文献 | "Newton's cradle" proton relay with amide-imidic acid tautomerization in inverting cellulase visualized by neutron crystallography. Sci Adv, 1, 2015
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3S92
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![BU of 3s92 by Molmil](/molmil-images/mine/3s92) | Crystal Structure of the second bromodomain of human BRD3 in complex with the inhibitor JQ1 | 分子名称: | (6S)-6-(2-tert-butoxy-2-oxoethyl)-4-(4-chlorophenyl)-2,3,9-trimethyl-6,7-dihydrothieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-10-ium, 1,2-ETHANEDIOL, Bromodomain-containing protein 3 | 著者 | Filippakopoulos, P, Picaud, S, Qi, J, Keates, T, Felletar, I, Fedorov, O, Muniz, J, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Weigelt, J, Bountra, C, Bradner, J.E, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2011-05-31 | 公開日 | 2011-06-29 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.36 Å) | 主引用文献 | Crystal Structure of the second bromodomain of human BRD3 in complex with the inhibitor JQ1 To be Published
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3X0K
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![BU of 3x0k by Molmil](/molmil-images/mine/3x0k) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ES-state at 0.97 angstrom resolution | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, [(2R,3S,4R,5R)-5-(6-AMINOPURIN-9-YL)-3,4-DIHYDROXY-OXOLAN-2-YL]METHYL [HYDROXY-[[(2R,3S,4R,5S)-3,4,5-TRIHYDROXYOXOLAN-2-YL]METHOXY]PHOSPHORYL] HYDROGEN PHOSPHATE | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-16 | 公開日 | 2016-04-27 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (0.97 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0I
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![BU of 3x0i by Molmil](/molmil-images/mine/3x0i) | ADP ribose pyrophosphatase in apo state at 0.91 angstrom resolution | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, SULFATE ION | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-16 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (0.91 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X2P
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![BU of 3x2p by Molmil](/molmil-images/mine/3x2p) | Neutron and X-ray joint refined structure of PcCel45A with cellopentaose at 298K. | 分子名称: | Endoglucanase V-like protein, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose-(1-4)-beta-D-glucopyranose-(1-4)-beta-D-glucopyranose-(1-4)-beta-D-glucopyranose | 著者 | Nakamura, A, Ishida, T, Kusaka, K, Yamada, T, Tanaka, I, Niimura, N, Samejima, M, Igarashi, K. | 登録日 | 2014-12-22 | 公開日 | 2015-10-14 | 最終更新日 | 2020-07-29 | 実験手法 | NEUTRON DIFFRACTION (1.518 Å), X-RAY DIFFRACTION | 主引用文献 | "Newton's cradle" proton relay with amide-imidic acid tautomerization in inverting cellulase visualized by neutron crystallography. Sci Adv, 1, 2015
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3X0M
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![BU of 3x0m by Molmil](/molmil-images/mine/3x0m) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ESM-state at reaction time of 3 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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