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PDB: 5 results

1LYB
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BU of 1lyb by Molmil
CRYSTAL STRUCTURES OF NATIVE AND INHIBITED FORMS OF HUMAN CATHEPSIN D: IMPLICATIONS FOR LYSOSOMAL TARGETING AND DRUG DESIGN
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CATHEPSIN D, PEPSTATIN, ...
Authors:Baldwin, E.T, Bhat, T.N, Gulnik, S, Erickson, J.W.
Deposit date:1993-04-22
Release date:1994-01-31
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Crystal structures of native and inhibited forms of human cathepsin D: implications for lysosomal targeting and drug design.
Proc.Natl.Acad.Sci.USA, 90, 1993
1LYA
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BU of 1lya by Molmil
CRYSTAL STRUCTURES OF NATIVE AND INHIBITED FORMS OF HUMAN CATHEPSIN D: IMPLICATIONS FOR LYSOSOMAL TARGETING AND DRUG DESIGN
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CATHEPSIN D, alpha-D-mannopyranose-(1-6)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose
Authors:Baldwin, E.T, Bhat, T.N, Gulnik, S, Erickson, J.W.
Deposit date:1993-04-22
Release date:1994-01-31
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Crystal structures of native and inhibited forms of human cathepsin D: implications for lysosomal targeting and drug design.
Proc.Natl.Acad.Sci.USA, 90, 1993
1M43
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BU of 1m43 by Molmil
Crystal structure of PMII in complex with pepstatin a to 2.4 A
Descriptor: Pepstatin, plasmepsin II
Authors:Asojo, O.A, Silva, A.M, Gulnik, S.
Deposit date:2002-07-02
Release date:2002-07-24
Last modified:2021-10-27
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Novel uncomplexed and complex structures of PM II, an aspartic protease from P. falciparum
To be Published
4FE6
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Crystal Structure of HIV-1 Protease in Complex with an enamino-oxindole inhibitor
Descriptor: (3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl {(2S,3R)-3-hydroxy-4-[({(3Z)-3-[1-(methylamino)ethylidene]-2-oxo-2,3-dihydro-1H-indol-5-yl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate, HIV protease
Authors:Silva, A.M, Eissenstat, M, Guerassina, T, Gulnik, S, Afonina, E, Yu, B, Erickson, J, Ludke, D, Yokoe, H.
Deposit date:2012-05-29
Release date:2012-07-18
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2 Å)
Cite:Enamino-oxindole HIV protease inhibitors.
Bioorg.Med.Chem.Lett., 22, 2012
1UQR
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Type II 3-dehydroquinate dehydratase (DHQase) from Actinobacillus pleuropneumoniae
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3-DEHYDROQUINATE DEHYDRATASE, SULFATE ION
Authors:Maes, D, Gonzalez-Ramirez, L.A, Lopez-Jaramillo, J, Yu, B, De Bondt, H, Zegers, I, Afonina, E, Garcia-Ruiz, J.M, Gulnik, S.
Deposit date:2003-10-16
Release date:2003-10-30
Last modified:2019-07-24
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Structural Study of the Type II 3-Dehydroquinate Dehydratase from Actinobacillus Pleuropneumoniae
Acta Crystallogr.,Sect.D, 60, 2004

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