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PDB: 1 results

8CX5
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BU of 8cx5 by Molmil
Crystal Structure of small molecule alpha,beta-ketoamide 4 covalently bound to K-Ras(G12R)
Descriptor: GUANOSINE-5'-DIPHOSPHATE, Isoform 2B of GTPase KRas, MAGNESIUM ION, ...
Authors:Zhang, Z, Morstein, J, Ecker, A, Guiley, K.Z, Shokat, K.M.
Deposit date:2022-05-19
Release date:2022-08-31
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (1.72 Å)
Cite:Chemoselective Covalent Modification of K-Ras(G12R) with a Small Molecule Electrophile.
J.Am.Chem.Soc., 144, 2022

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