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PDB: 5 件

2AW2
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BU of 2aw2 by Molmil
Crystal structure of the human BTLA-HVEM complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, B and T lymphocyte attenuator, NICKEL (II) ION, ...
著者Compaan, D.M, Gonzalez, L.C, Tom, I, Loyet, K.M, Eaton, D, Hymowitz, S.G.
登録日2005-08-31
公開日2005-09-27
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Attenuating Lymphocyte Activity: the crystal structure of the BTLA-HVEM complex
J.Biol.Chem., 280, 2005
7UFG
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BU of 7ufg by Molmil
Cryo-EM structure of PAPP-A in complex with IGFBP5
分子名称: Insulin-like growth factor-binding protein 5, Pappalysin-1, ZINC ION
著者Judge, R.A, Jain, R, Hao, Q, Ouch, C, Sridar, J, Smith, C.L, Wang, J.C.K, Eaton, D.
登録日2022-03-22
公開日2022-09-28
実験手法ELECTRON MICROSCOPY (3.28 Å)
主引用文献Structure of the PAPP-ABP5 complex reveals mechanism of substrate recognition
Nat Commun, 13, 2022
8D8O
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Cryo-EM structure of substrate unbound PAPP-A
分子名称: Pappalysin-1, ZINC ION
著者Judge, R.A, Jain, R, Hao, Q, Ouch, C, Sridar, J, Smith, C.L, Wang, J.C.K, Eaton, D.
登録日2022-06-08
公開日2022-09-28
実験手法ELECTRON MICROSCOPY (3.35 Å)
主引用文献Structure of the PAPP-ABP5 complex reveals mechanism of substrate recognition
Nat Commun, 13, 2022
8SL1
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Cryo-EM structure of PAPP-A2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Judge, R.A, Stoll, V.S, Eaton, D, Hao, Q, Bratkowski, M.A.
登録日2023-04-20
公開日2023-11-08
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.13 Å)
主引用文献Cryo-EM structure of human PAPP-A2 and mechanism of substrate recognition.
Commun Chem, 6, 2023
4XJS
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Human CD38 complexed with inhibitor 1 [6-fluoro-2-methyl-4-[(2,3,6-trichlorobenzyl)amino]quinoline-8-carboxamide]
分子名称: 5-O-phosphono-alpha-D-ribofuranose, 6-fluoro-2-methyl-4-[(2,3,6-trichlorobenzyl)amino]quinoline-8-carboxamide, ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
著者Shewchuk, L.M, Deaton, D, Stewart, E.
登録日2015-01-09
公開日2015-08-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Discovery of 4-Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38.
J.Med.Chem., 58, 2015

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件を2024-07-03に公開中

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