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PDB: 6 件

4NJN
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BU of 4njn by Molmil
Crystal Structure of E.coli GlpG at pH 4.5
分子名称: Rhomboid protease GlpG
著者Dickey, S.W, Baker, R.P, Cho, S, Urban, S.
登録日2013-11-11
公開日2013-12-25
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Proteolysis inside the Membrane Is a Rate-Governed Reaction Not Driven by Substrate Affinity.
Cell(Cambridge,Mass.), 155, 2013
4NJP
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BU of 4njp by Molmil
Proteolysis inside the membrane is a rate-governed reaction not Driven by substrate affinity
分子名称: Rhomboid protease GlpG
著者Dickey, S.W, Baker, R.P, Cho, S, Urban, S.
登録日2013-11-11
公開日2013-12-25
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Proteolysis inside the Membrane Is a Rate-Governed Reaction Not Driven by Substrate Affinity.
Cell(Cambridge,Mass.), 155, 2013
5F5B
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BU of 5f5b by Molmil
Structure of E.Coli GlpG complexed with peptidic inhibitor Ac-VRMA-CHO
分子名称: Rhomboid protease GlpG, peptidic derivative of Gurken: ACE-VAL-ARG-MET-ALA-aldehyde
著者Urban, S, Cho, S, Dickey, S.W.
登録日2015-12-04
公開日2016-02-17
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis.
Mol.Cell, 61, 2016
5F5D
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BU of 5f5d by Molmil
Crystal structures and Inhibition kinetics reveal a two-state catalytic mechanism with drug design implications for rhomboid proteolysis
分子名称: Rhomboid protease GlpG
著者Urban, S, Cho, S, Dickey, S.W.
登録日2015-12-04
公開日2016-02-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis.
Mol.Cell, 61, 2016
5F5G
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BU of 5f5g by Molmil
Structure of E.Coli GlpG Y205F mutant complexed with peptidic inhibitor Ac-RMA-CHO in the DMPC/CHAPSO bicelle
分子名称: ACE-ARG-MET-ALA-aldehyde, Rhomboid protease GlpG
著者Urban, S, Cho, S, Dickey, S.W.
登録日2015-12-04
公開日2016-04-06
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis.
Mol.Cell, 61, 2016
5F5K
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BU of 5f5k by Molmil
E.Coli GlpG Y205F mutant complexed with aldehyde inhibitor in DMPC/CHAPSO bicelle
分子名称: Peptidic derivative of Gurken: ACE-ARG-LYS-VAL-ARG-MET-ALA-aldehyde, Rhomboid protease GlpG
著者Urban, S, Cho, S, Dickey, S.W.
登録日2015-12-04
公開日2016-02-10
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis.
Mol.Cell, 61, 2016

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件を2024-07-24に公開中

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