6PVH
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![BU of 6pvh by Molmil](/molmil-images/mine/6pvh) | Crystal structure of PhqK in complex with paraherquamide K | 分子名称: | (7aS,12S,12aR,13aS)-3,3,12,14,14-pentamethyl-3,7,11,12,13,13a,14,15-octahydro-8H,10H-7a,12a-(epiminomethano)indolizino[6,7-h]pyrano[3,2-a]carbazol-16-one, FAD monooxygenase, FLAVIN-ADENINE DINUCLEOTIDE | 著者 | Fraley, A.E, Smith, J.L, Sherman, D.H. | 登録日 | 2019-07-20 | 公開日 | 2020-01-22 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Molecular Basis for Spirocycle Formation in the Paraherquamide Biosynthetic Pathway. J.Am.Chem.Soc., 142, 2020
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8IJ6
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![BU of 8ij6 by Molmil](/molmil-images/mine/8ij6) | Crystal structure of alcohol dehydrogenase from Burkholderia gladioli with NADP | 分子名称: | NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, Putative short-chain dehydrogenases/reductase family protein | 著者 | Han, X, Mei, Z.L, Liu, W.D, Sun, Z.T, Ma, J.A. | 登録日 | 2023-02-26 | 公開日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.28 Å) | 主引用文献 | Crystal structure of alcohol dehydrogenase from Burkholderia gladioli with NADP To Be Published
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8IJ8
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6PVB
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![BU of 6pvb by Molmil](/molmil-images/mine/6pvb) | The structure of NTMT1 in complex with compound 6 | 分子名称: | AMINO GROUP-()-(2~{S})-2-azanylpropanal-()-ISOLEUCINE-()-ARGININE-()-LYSINE-()-PROLINE-()-AMINO-ACETALDEHYDE-()-9-(5-{[(3S)-3-amino-3-carboxypropyl](pentyl)amino}-5-deoxy-beta-L-arabinofuranosyl)-9H-purin-6-amine, N-terminal Xaa-Pro-Lys N-methyltransferase 1, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Noinaj, N, Chen, D, Huang, R. | 登録日 | 2019-07-20 | 公開日 | 2020-08-19 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Probing the Plasticity in the Active Site of Protein N-terminal Methyltransferase 1 Using Bisubstrate Analogues. J.Med.Chem., 63, 2020
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6PVI
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![BU of 6pvi by Molmil](/molmil-images/mine/6pvi) | Crystal structure of PhqK in complex with paraherquamide L | 分子名称: | (8aS,13S,13aR,14aS)-4,4,13,15,15-pentamethyl-12,13,14,14a,15,16-hexahydro-4H,8H,9H,11H-8a,13a-(epiminomethano)[1,4]dioxepino[2,3-a]indolizino[6,7-h]carbazol-17-one, FAD monooxygenase, FLAVIN-ADENINE DINUCLEOTIDE | 著者 | Fraley, A.E, Smith, J.L, Sherman, D.H. | 登録日 | 2019-07-20 | 公開日 | 2020-01-22 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.093 Å) | 主引用文献 | Molecular Basis for Spirocycle Formation in the Paraherquamide Biosynthetic Pathway. J.Am.Chem.Soc., 142, 2020
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8IJ7
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8II9
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![BU of 8ii9 by Molmil](/molmil-images/mine/8ii9) | crystal structure of Hyp mutant from Hypoxylon sp. E7406B | 分子名称: | Terpene synthase | 著者 | Gao, J, Liu, W.D, Li, Q, Han, X, Wei, H.L, Dai, Z.J, Su, L.Q. | 登録日 | 2023-02-24 | 公開日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | crystal structure of Hyp to be published
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6Q1D
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![BU of 6q1d by Molmil](/molmil-images/mine/6q1d) | Holo YfeA reconstituted by zinc soaking | 分子名称: | Periplasmic chelated iron-binding protein YfeA, ZINC ION | 著者 | Radka, C.D, Labiuk, S.L, DeLucas, L.J, Aller, S.G. | 登録日 | 2019-08-03 | 公開日 | 2019-09-04 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Structures of the substrate-binding protein YfeA in apo and zinc-reconstituted holo forms. Acta Crystallogr D Struct Biol, 75, 2019
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4RIM
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2IOQ
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6Q7K
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![BU of 6q7k by Molmil](/molmil-images/mine/6q7k) | ERK2 mini-fragment binding | 分子名称: | 1H-imidazol-2-amine, Mitogen-activated protein kinase 1, SULFATE ION | 著者 | O'Reilly, M, Cleasby, A, Davies, T.G, Hall, R, Ludlow, F, Murray, C.W, Tisi, D, Jhoti, H. | 登録日 | 2018-12-13 | 公開日 | 2019-03-27 | 最終更新日 | 2019-05-22 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | Crystallographic screening using ultra-low-molecular-weight ligands to guide drug design. Drug Discov Today, 24, 2019
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2IJF
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8IHA
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6QEG
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![BU of 6qeg by Molmil](/molmil-images/mine/6qeg) | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX WITH AN INHIBITOR 2-Oxo-1-phenyl-pyrrolidine-3-carboxylic acid (2-thiophen-2-yl-ethyl)-amide | 分子名称: | (3~{S})-3-oxidanyl-2-oxidanylidene-1-phenyl-~{N}-(2-thiophen-2-ylethyl)pyrrolidine-3-carboxamide, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Musil, D, Heinrich, T, Lehmann, M. | 登録日 | 2019-01-07 | 公開日 | 2019-05-01 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | Discovery and Structure-Based Optimization of Next-Generation Reversible Methionine Aminopeptidase-2 (MetAP-2) Inhibitors. J.Med.Chem., 62, 2019
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2IYT
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![BU of 2iyt by Molmil](/molmil-images/mine/2iyt) | Shikimate kinase from Mycobacterium tuberculosis in unliganded state, open LID (conf. A) | 分子名称: | CHLORIDE ION, SHIKIMATE KINASE | 著者 | Hartmann, M.D, Bourenkov, G.P, Oberschall, A, Strizhov, N, Bartunik, H.D. | 登録日 | 2006-07-22 | 公開日 | 2006-10-11 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Mechanism of Phosphoryl Transfer Catalyzed by Shikimate Kinase from Mycobacterium Tuberculosis. J.Mol.Biol., 364, 2006
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5KSY
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![BU of 5ksy by Molmil](/molmil-images/mine/5ksy) | hMiro1 C-domain GDP Complex P41212 Crystal Form | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, Mitochondrial Rho GTPase 1 | 著者 | Klosowiak, J.L, Focia, P.J, Rice, S.E, Freymann, D.M. | 登録日 | 2016-07-10 | 公開日 | 2016-09-21 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.482 Å) | 主引用文献 | Structural insights into Parkin substrate lysine targeting from minimal Miro substrates. Sci Rep, 6, 2016
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4RR2
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![BU of 4rr2 by Molmil](/molmil-images/mine/4rr2) | Crystal structure of human primase | 分子名称: | DNA primase large subunit, DNA primase small subunit, IRON/SULFUR CLUSTER, ... | 著者 | Baranovskiy, A.G, Gu, J, Suwa, Y, Babayeva, N.D, Tahirov, T.H. | 登録日 | 2014-11-05 | 公開日 | 2015-01-21 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Crystal structure of the human primase. J.Biol.Chem., 290, 2015
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2J6B
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![BU of 2j6b by Molmil](/molmil-images/mine/2j6b) | crystal structure of AFV3-109, a highly conserved protein from crenarchaeal viruses | 分子名称: | AFV3-109 | 著者 | Keller, J, Leulliot, N, Cambillau, C, Campanacci, V, Porciero, S, Prangishvili, D, Cortez, D, Quevillon-Cheruel, S, Van Tilbeurgh, H. | 登録日 | 2006-09-27 | 公開日 | 2007-02-20 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Crystal Structure of Afv3-109, a Highly Conserved Protein from Crenarchaeal Viruses. Virol J., 4, 2007
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4RWH
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![BU of 4rwh by Molmil](/molmil-images/mine/4rwh) | Crystal structure of T cell costimulatory ligand B7-1 (CD80) | 分子名称: | T-lymphocyte activation antigen CD80 | 著者 | Fedorov, A.A, Fedorov, E.V, Samanta, D, Hillerich, B, Seidel, R.D, Almo, S.C. | 登録日 | 2014-12-04 | 公開日 | 2014-12-17 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.802 Å) | 主引用文献 | Crystal structure of T cell costimulatory ligand B7-1 (CD80) To be Published
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6JD2
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![BU of 6jd2 by Molmil](/molmil-images/mine/6jd2) | Crystal structure of Sulfolobus solfataricus ketol-acid reductoisomerase (Sso-KARI) in complex with Mg2+ at pH8.5 | 分子名称: | BETA-MERCAPTOETHANOL, MAGNESIUM ION, Putative ketol-acid reductoisomerase 2 | 著者 | Chen, C.Y, Chang, Y.C, Lin, K.F, Huang, C.H, Lin, B.L, Ko, T.P, Hsieh, D.L, Tsai, M.D. | 登録日 | 2019-01-30 | 公開日 | 2019-08-14 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.53 Å) | 主引用文献 | Use of Cryo-EM To Uncover Structural Bases of pH Effect and Cofactor Bispecificity of Ketol-Acid Reductoisomerase. J.Am.Chem.Soc., 141, 2019
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6JFV
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![BU of 6jfv by Molmil](/molmil-images/mine/6jfv) | The crystal structure of 2B-2B complex from keratins 5 and 14 (C367A mutant of K14) | 分子名称: | Keratin, type I cytoskeletal 14, type II cytoskeletal 5 | 著者 | Kim, M.S, Lee, C.H, Coulombe, P.A, Leahy, D.J. | 登録日 | 2019-02-12 | 公開日 | 2020-01-22 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structure-Function Analyses of a Keratin Heterotypic Complex Identify Specific Keratin Regions Involved in Intermediate Filament Assembly. Structure, 28, 2020
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7B5K
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![BU of 7b5k by Molmil](/molmil-images/mine/7b5k) | E. coli 70S containing suppressor tRNA in the A-site stabilized by a Negamycin analogue and P-site tRNA-nascent chain. | 分子名称: | 16S rRNA, 2-[[[(3~{R},5~{R})-3-azanyl-6-(3-azanylpropylamino)-5-oxidanyl-hexanoyl]amino]-methyl-amino]ethanoic acid, 23S rRNA, ... | 著者 | Albers, S, Beckert, B, Matthies, M, Schuster, R, Riedner, M, Seuring, C, Sanyal, S, Torda, A, Wilson, N.D, Ignatova, Z. | 登録日 | 2020-12-03 | 公開日 | 2021-05-26 | 最終更新日 | 2024-04-24 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Harnessing evolutionarily flexibility in tRNAs to maximize nonsense suppression activities Nat Commun, 2021
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1SVL
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![BU of 1svl by Molmil](/molmil-images/mine/1svl) | Co-crystal structure of SV40 large T antigen helicase domain and ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ZINC ION, ... | 著者 | Gai, D, Zhao, R, Finkielstein, C.V, Chen, X.S. | 登録日 | 2004-03-29 | 公開日 | 2004-10-19 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Mechanisms of conformational change for a replicative hexameric helicase of SV40 large tumor antigen. Cell(Cambridge,Mass.), 119, 2004
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4R4P
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![BU of 4r4p by Molmil](/molmil-images/mine/4r4p) | Crystal Structure of the VS ribozyme-A756G mutant | 分子名称: | MAGNESIUM ION, VS ribozyme RNA | 著者 | Piccirilli, J.A, Suslov, N.B, Dasgupta, S, Huang, H, Lilley, D.M.J, Rice, P.A. | 登録日 | 2014-08-19 | 公開日 | 2015-09-30 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.07 Å) | 主引用文献 | Crystal structure of the Varkud satellite ribozyme. Nat.Chem.Biol., 11, 2015
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6IDS
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![BU of 6ids by Molmil](/molmil-images/mine/6ids) | Crystal structure of Vibrio cholerae MATE transporter VcmN D35N mutant | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, MATE family efflux transporter | 著者 | Kusakizako, T, Claxton, D.P, Tanaka, Y, Maturana, A.D, Kuroda, T, Ishitani, R, Mchaourab, H.S, Nureki, O. | 登録日 | 2018-09-11 | 公開日 | 2019-01-16 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.79 Å) | 主引用文献 | Structural Basis of H+-Dependent Conformational Change in a Bacterial MATE Transporter. Structure, 27, 2019
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