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PDB: 2 results

8PJ8
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BU of 8pj8 by Molmil
FKBP51FK1 F67E/K60Orn (i, i+7) in complex with SAFit1
Descriptor: 2-[3-[(1~{R})-1-[(2~{S})-1-[(2~{S})-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)ethanoyl]piperidin-2-yl]carbonyloxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]ethanoic acid, Peptidyl-prolyl cis-trans isomerase FKBP5
Authors:Meyners, C, Charalampidou, A, Hausch, F.
Deposit date:2023-06-23
Release date:2024-03-06
Last modified:2024-04-10
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Automated Flow Peptide Synthesis Enables Engineering of Proteins with Stabilized Transient Binding Pockets.
Acs Cent.Sci., 10, 2024
8PJA
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BU of 8pja by Molmil
FKBP51FK1 F67E/K58 (i, i+9) in complex with SAFit1
Descriptor: 2-[3-[(1~{R})-1-[(2~{S})-1-[(2~{S})-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)ethanoyl]piperidin-2-yl]carbonyloxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]ethanoic acid, Peptidyl-prolyl cis-trans isomerase FKBP5
Authors:Meyners, C, Charalampidou, A, Hausch, F.
Deposit date:2023-06-23
Release date:2024-03-06
Last modified:2024-04-10
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Automated Flow Peptide Synthesis Enables Engineering of Proteins with Stabilized Transient Binding Pockets.
Acs Cent.Sci., 10, 2024

219140

PDB entries from 2024-05-01

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