6S4F
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![BU of 6s4f by Molmil](/molmil-images/mine/6s4f) | Structure of human MTHFD2 in complex with TH9619 | 分子名称: | (E,4S)-4-[[5-[2-[2,6-bis(azanyl)-4-oxidanylidene-1H-pyrimidin-5-yl]ethanoylamino]-3-fluoranyl-pyridin-2-yl]carbonylamino]pent-2-enedioic acid, ADENOSINE-5'-DIPHOSPHATE, Bifunctional methylenetetrahydrofolate dehydrogenase/cyclohydrolase, ... | 著者 | Scaletti, E.R, Gustafsson, R, Bonagas, N, Gustafsson, N.M, Henriksson, M, Abdurakhmanov, E, Andersson, Y, Bengtsson, C, Borhade, S, Desroses, M, Farnegardh, K, Garg, N, Gokturk, C, Haraldsson, M, Iliev, P, Jarvius, M, Jemth, A.S, Kalderen, C, Karsten, S, Klingegard, F, Koolmeister, T, Martens, U, Llona-Minguez, S, Loseva, O, Marttila, P, Michel, M, Moulson, R, Nordstrom, H, Paulin, C, Pham, T, Pudelko, L, Rasti, A, Roos, A.K, Sarno, A, Sandberg, L, Scobie, M, Sjoberg, B, Svensson, R, Unterlass, J.E, Vallin, K, Vo, D, Wiita, E, Warpman-Berglund, U, Homan, E.J, Helleday, T, Stenmark, P. | 登録日 | 2019-06-27 | 公開日 | 2021-07-07 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Pharmacological targeting of MTHFD2 suppresses acute myeloid leukemia by inducing thymidine depletion and replication stress. Nat Cancer, 3, 2022
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6S4E
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![BU of 6s4e by Molmil](/molmil-images/mine/6s4e) | Structure of human MTHFD2 in complex with TH7299 | 分子名称: | (2S)-2-[[4-[[2,4-bis(azanyl)-6-oxidanylidene-1H-pyrimidin-5-yl]carbamoylamino]phenyl]carbonylamino]pentanedioic acid, Bifunctional methylenetetrahydrofolate dehydrogenase/cyclohydrolase, mitochondrial, ... | 著者 | Gustafsson, R, Scaletti, E.R, Bonagas, N, Gustafsson, N.M, Henriksson, M, Abdurakhmanov, E, Andersson, Y, Bengtsson, C, Borhade, S, Desroses, M, Farnegardh, K, Garg, N, Gokturk, C, Haraldsson, M, Iliev, P, Jarvius, M, Jemth, A.S, Kalderen, C, Karsten, S, Klingegard, F, Koolmeister, T, Martens, U, Llona-Minguez, S, Loseva, O, Marttila, P, Michel, M, Moulson, R, Nordstrom, H, Paulin, C, Pham, T, Pudelko, L, Rasti, A, Roos, A.K, Sarno, A, Sandberg, L, Scobie, M, Sjoberg, B, Svensson, R, Unterlass, J.E, Vallin, K, Vo, D, Wiita, E, Warpman-Berglund, U, Homan, E.J, Helleday, T, Stenmark, P. | 登録日 | 2019-06-27 | 公開日 | 2021-07-07 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Pharmacological targeting of MTHFD2 suppresses acute myeloid leukemia by inducing thymidine depletion and replication stress. Nat Cancer, 3, 2022
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1GXD
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![BU of 1gxd by Molmil](/molmil-images/mine/1gxd) | proMMP-2/TIMP-2 complex | 分子名称: | 72 KDA TYPE IV COLLAGENASE, CALCIUM ION, METALLOPROTEINASE INHIBITOR 2, ... | 著者 | Morgunova, E, Tuuttila, A, Bergmann, U, Tryggvason, K. | 登録日 | 2002-04-02 | 公開日 | 2002-07-09 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structural Insight Into the Complex Formation of Latent Matrix Metalloproteinase 2 with Tissue Inhibitor of Metalloproteinase 2 Proc.Natl.Acad.Sci.USA, 99, 2002
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1PNE
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![BU of 1pne by Molmil](/molmil-images/mine/1pne) | CRYSTALLIZATION AND STRUCTURE DETERMINATION OF BOVINE PROFILIN AT 2.0 ANGSTROMS RESOLUTION | 分子名称: | PROFILIN | 著者 | Cedergren-Zeppezauer, E.S, Goonesekere, N.C.W, Rozycki, M.D, Myslik, J.C, Dauter, Z, Lindberg, U, Schutt, C.E. | 登録日 | 1995-05-05 | 公開日 | 1995-07-31 | 最終更新日 | 2017-11-29 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystallization and structure determination of bovine profilin at 2.0 A resolution. J.Mol.Biol., 240, 1994
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2OAN
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![BU of 2oan by Molmil](/molmil-images/mine/2oan) | Structure of oxidized beta-actin | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Actin, cytoplasmic 1, ... | 著者 | Schmitzberger, F, Lassing, I, Nordlund, P, Lindberg, U. | 登録日 | 2006-12-16 | 公開日 | 2007-05-01 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.606 Å) | 主引用文献 | Molecular and Structural Basis for Redox Regulation of beta-Actin. J.Mol.Biol., 370, 2007
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1F7S
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![BU of 1f7s by Molmil](/molmil-images/mine/1f7s) | CRYSTAL STRUCTURE OF ADF1 FROM ARABIDOPSIS THALIANA | 分子名称: | ACTIN DEPOLYMERIZING FACTOR (ADF), LAURYL DIMETHYLAMINE-N-OXIDE | 著者 | Bowman, G.D, Nodelman, I.M, Lindberg, U, Chua, N.H, Schutt, C.E. | 登録日 | 2000-06-27 | 公開日 | 2000-11-15 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | A comparative structural analysis of the ADF/cofilin family. Proteins, 41, 2000
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6J7W
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![BU of 6j7w by Molmil](/molmil-images/mine/6j7w) | Crystal Structure of Human BCMA in complex with UniAb(TM) VH | 分子名称: | Tumor necrosis factor receptor superfamily member 17, UniAb | 著者 | Clarke, S.C, Ma, B, Trinklein, N.D, Schellenberger, U, Osborn, M, Ouisse, L, Boudreau, A, Davison, L, Harris, K.E, Ugamraj, H, Balasubramani, A, Dang, K, Jorgensen, B, Ogana, H, Pham, D, Pratap, P, Sankaran, P, Anegon, I, van Schooten, W, Bruggemann, M, Buelow, R, Force Aldred, S. | 登録日 | 2019-01-18 | 公開日 | 2019-02-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Multispecific Antibody Development Platform Based on Human Heavy Chain Antibodies Front Immunol, 9, 2018
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5E7Y
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![BU of 5e7y by Molmil](/molmil-images/mine/5e7y) | Crystal structure of P450 BM3 heme domain M7 variant | 分子名称: | Bifunctional P-450/NADPH-P450 reductase, GLYCEROL, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Panneerselvm, S, Shehzad, A, Bocola, M, Mueller-Dieckmann, J, Schwaneberg, U. | 登録日 | 2015-10-13 | 公開日 | 2017-01-25 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of P450 BM3 heme domain M7 variant To Be Published
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1TJ7
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![BU of 1tj7 by Molmil](/molmil-images/mine/1tj7) | Structure determination and refinement at 2.44 A resolution of Argininosuccinate lyase from E. coli | 分子名称: | Argininosuccinate lyase, GLYCEROL, PHOSPHATE ION | 著者 | Bhaumik, P, Koski, M.K, Bergman, U, Wierenga, R.K. | 登録日 | 2004-06-03 | 公開日 | 2004-10-26 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.44 Å) | 主引用文献 | Structure determination and refinement at 2.44 A resolution of argininosuccinate lyase from Escherichia coli. Acta Crystallogr.,Sect.D, 60, 2004
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5NGS
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![BU of 5ngs by Molmil](/molmil-images/mine/5ngs) | Crystal structure of human MTH1 in complex with inhibitor 6-[(2-phenylethyl)sulfanyl]-7H-purin-2-amine | 分子名称: | 6-(2-phenylethylsulfanyl)-7~{H}-purin-2-amine, 7,8-dihydro-8-oxoguanine triphosphatase, ACETATE ION, ... | 著者 | Gustafsson, R, Rudling, A, Almlof, I, Homan, E, Scobie, M, Warpman Berglund, U, Helleday, T, Carlsson, J, Stenmark, P. | 登録日 | 2017-03-20 | 公開日 | 2017-10-04 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Fragment-Based Discovery and Optimization of Enzyme Inhibitors by Docking of Commercial Chemical Space. J. Med. Chem., 60, 2017
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5NGR
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![BU of 5ngr by Molmil](/molmil-images/mine/5ngr) | Crystal structure of human MTH1 in complex with fragment inhibitor 8-(methylsulfanyl)-7H-purin-6-amine | 分子名称: | 7,8-dihydro-8-oxoguanine triphosphatase, 8-methylsulfanyl-7~{H}-purin-6-amine, SULFATE ION | 著者 | Gustafsson, R, Rudling, A, Almlof, I, Homan, E, Scobie, M, Warpman Berglund, U, Helleday, T, Carlsson, J, Stenmark, P. | 登録日 | 2017-03-20 | 公開日 | 2017-10-04 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Fragment-Based Discovery and Optimization of Enzyme Inhibitors by Docking of Commercial Chemical Space. J. Med. Chem., 60, 2017
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4TNL
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![BU of 4tnl by Molmil](/molmil-images/mine/4tnl) | 1.8 A resolution room temperature structure of Thermolysin recorded using an XFEL | 分子名称: | CALCIUM ION, Thermolysin, ZINC ION | 著者 | Kern, J, Tran, R, Alonso-Mori, R, Koroidov, S, Echols, N, Hattne, J, Ibrahim, M, Gul, S, Laksmono, H, Sierra, R.G, Gildea, R.J, Han, G, Hellmich, J, Lassalle-Kaiser, B, Chatterjee, R, Brewster, A, Stan, C.A, Gloeckner, C, Lampe, A, DiFiore, D, Milathianaki, D, Fry, A.R, Seibert, M.M, Koglin, J.E, Gallo, E, Uhlig, J, Sokaras, D, Weng, T.-C, Zwart, P.H, Skinner, D.E, Bogan, M.J, Messerschmidt, M, Glatzel, P, Williams, G.J, Boutet, S, Adams, P.D, Zouni, A, Messinger, J, Sauter, N.K, Bergmann, U, Yano, J, Yachandra, V.K. | 登録日 | 2014-06-04 | 公開日 | 2014-07-09 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Taking snapshots of photosynthetic water oxidation using femtosecond X-ray diffraction and spectroscopy. Nat Commun, 5, 2014
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5NGT
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![BU of 5ngt by Molmil](/molmil-images/mine/5ngt) | Crystal structure of human MTH1 in complex with inhibitor 7-(furan-2-yl)-5-methyl-1,3-benzoxazol-2-amine | 分子名称: | 7,8-dihydro-8-oxoguanine triphosphatase, 7-(furan-2-yl)-5-methyl-1,3-benzoxazol-2-amine, SULFATE ION | 著者 | Gustafsson, R, Rudling, A, Almlof, I, Homan, E, Scobie, M, Warpman Berglund, U, Helleday, T, Carlsson, J, Stenmark, P. | 登録日 | 2017-03-20 | 公開日 | 2017-10-04 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Fragment-Based Discovery and Optimization of Enzyme Inhibitors by Docking of Commercial Chemical Space. J. Med. Chem., 60, 2017
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1BKO
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![BU of 1bko by Molmil](/molmil-images/mine/1bko) | |
1BKP
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![BU of 1bkp by Molmil](/molmil-images/mine/1bkp) | |
1BR9
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![BU of 1br9 by Molmil](/molmil-images/mine/1br9) | HUMAN TISSUE INHIBITOR OF METALLOPROTEINASE-2 | 分子名称: | METALLOPROTEINASE-2 INHIBITOR | 著者 | Tuuttila, A, Morgunova, E, Bergmann, U, Lindqvist, Y, Tryggvason, K, Schneider, G. | 登録日 | 1998-08-28 | 公開日 | 1999-05-04 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Three-dimensional structure of human tissue inhibitor of metalloproteinases-2 at 2.1 A resolution. J.Mol.Biol., 284, 1998
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1BSP
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![BU of 1bsp by Molmil](/molmil-images/mine/1bsp) | THERMOSTABLE THYMIDYLATE SYNTHASE A FROM BACILLUS SUBTILIS | 分子名称: | PHOSPHATE ION, THYMIDYLATE SYNTHASE A | 著者 | Stout, T.J, Schellenberger, U, Santi, D.V, Stroud, R.M. | 登録日 | 1998-07-09 | 公開日 | 1999-02-16 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structures of a unique thermal-stable thymidylate synthase from Bacillus subtilis. Biochemistry, 37, 1998
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1BSF
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1CK7
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![BU of 1ck7 by Molmil](/molmil-images/mine/1ck7) | GELATINASE A (FULL-LENGTH) | 分子名称: | CALCIUM ION, CHLORIDE ION, PROTEIN (GELATINASE A), ... | 著者 | Morgunova, E, Tuuttila, A, Bergmann, U, Isupov, M, Lindqvist, Y, Schneider, G, Tryggvason, K. | 登録日 | 1999-04-28 | 公開日 | 1999-08-25 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structure of human pro-matrix metalloproteinase-2: activation mechanism revealed. Science, 284, 1999
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5E78
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![BU of 5e78 by Molmil](/molmil-images/mine/5e78) | Crystal structure of P450 BM3 heme domain variant complexed with Co(III)Sep | 分子名称: | 1,3,6,8,10,13,16,19-octaazabicyclo[6.6.6]icosane, Bifunctional P-450/NADPH-P450 reductase, CHLORIDE ION, ... | 著者 | Panneerselvm, S, Shehzad, A, Bocola, M, Mueller-Dieckmann, J, Schwaneberg, U. | 登録日 | 2015-10-12 | 公開日 | 2016-09-28 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystallographic insights into a cobalt (III) sepulchrate based alternative cofactor system of P450 BM3 monooxygenase. Biochim. Biophys. Acta, 1866, 2018
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1D1J
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![BU of 1d1j by Molmil](/molmil-images/mine/1d1j) | CRYSTAL STRUCTURE OF HUMAN PROFILIN II | 分子名称: | 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 1-METHOXY-2-[2-(2-METHOXY-ETHOXY]-ETHANE, PROFILIN II, ... | 著者 | Nodelman, I.M, Bowman, G.D, Lindberg, U, Schutt, C.E. | 登録日 | 1999-09-17 | 公開日 | 2000-12-22 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | X-ray structure determination of human profilin II: A comparative structural analysis of human profilins. J.Mol.Biol., 294, 1999
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7VKE
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![BU of 7vke by Molmil](/molmil-images/mine/7vke) | Crystal structure of human CD38 ECD in complex with UniDab(TM) F11A | 分子名称: | 1,2-ETHANEDIOL, ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1, CHLORIDE ION, ... | 著者 | Schooten, W.V, Schellenberger, U, Ugamraj, H.S, Manicka, S, Bijpuria, S, Gondu, R.K. | 登録日 | 2021-09-29 | 公開日 | 2022-08-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | TNB-738, a biparatopic antibody, boosts intracellular NAD+ by inhibiting CD38 ecto-enzyme activity. Mabs, 14, 2022
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1TJC
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![BU of 1tjc by Molmil](/molmil-images/mine/1tjc) | Crystal structure of peptide-substrate-binding domain of human type I collagen prolyl 4-hydroxylase | 分子名称: | Prolyl 4-hydroxylase alpha-1 subunit | 著者 | Pekkala, M, Hieta, R, Bergmann, U, Kivirikko, K.I, Wierenga, R.K, Myllyharju, J. | 登録日 | 2004-06-04 | 公開日 | 2004-10-12 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The Peptide-Substrate-binding Domain of Collagen Prolyl 4-Hydroxylases Is a Tetratricopeptide Repeat Domain with Functional Aromatic Residues. J.Biol.Chem., 279, 2004
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1JS5
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![BU of 1js5 by Molmil](/molmil-images/mine/1js5) | Solution Structure of dAAUAA DNA Bulge | 分子名称: | 5'-D(*CP*GP*TP*AP*GP*CP*CP*GP*AP*TP*GP*C)-3', 5'-D(*GP*CP*AP*TP*CP*GP*AP*AP*UP*AP*AP*GP*CP*TP*AP*CP*G)-3' | 著者 | Gollmick, F.A, Lorenz, M, Dornberger, U, von Langen, J, Diekmann, S, Fritzsche, H. | 登録日 | 2001-08-16 | 公開日 | 2002-08-28 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of dAATAA and dAAUAA DNA bulges. Nucleic Acids Res., 30, 2002
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1JS7
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![BU of 1js7 by Molmil](/molmil-images/mine/1js7) | Solution Structure of dAAUAA DNA Bulge | 分子名称: | 5'-D(*CP*GP*TP*AP*GP*CP*CP*GP*AP*TP*GP*C)-3', 5'-D(*GP*CP*AP*TP*CP*GP*AP*AP*UP*AP*AP*GP*CP*TP*AP*CP*G)-3' | 著者 | Gollmick, F.A, Lorenz, M, Dornberger, U, von Langen, J, Diekmann, S, Fritzsche, H. | 登録日 | 2001-08-16 | 公開日 | 2002-06-19 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of dAATAA and dAAUAA DNA bulges. Nucleic Acids Res., 30, 2002
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