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PDB: 3 results

6FQV
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BU of 6fqv by Molmil
2.60A BINARY COMPLEX OF S.AUREUS GYRASE with UNCLEAVED DNA
Descriptor: DNA (5'-D(*GP*AP*GP*CP*GP*TP*AP*CP*GP*GP*CP*CP*GP*TP*AP*CP*GP*CP*TP*T)-3'), DNA gyrase subunit A, DNA gyrase subunit B,DNA gyrase subunit B, ...
Authors:Bax, B.D, Germe, T, Basque, E, Maxwell, A.
Deposit date:2018-02-14
Release date:2018-04-04
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:A new class of antibacterials, the imidazopyrazinones, reveal structural transitions involved in DNA gyrase poisoning and mechanisms of resistance.
Nucleic Acids Res., 46, 2018
6FQM
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BU of 6fqm by Molmil
3.06A COMPLEX OF S.AUREUS GYRASE with imidazopyrazinone T1 AND DNA
Descriptor: 7-[(3~{S})-3-azanylpyrrolidin-1-yl]-5-cyclopropyl-8-fluoranyl-imidazo[1,2-a]quinoxalin-4-one, DNA (5'-D(*GP*AP*GP*AP*GP*TP*AP*T*GP*GP*CP*CP*AP*TP*AP*CP*TP*CP*T)-3'), DNA gyrase subunit A, ...
Authors:Bax, B.D, Germe, T, Basque, E, Maxwell, A.
Deposit date:2018-02-14
Release date:2018-04-04
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (3.06 Å)
Cite:A new class of antibacterials, the imidazopyrazinones, reveal structural transitions involved in DNA gyrase poisoning and mechanisms of resistance.
Nucleic Acids Res., 46, 2018
6FQS
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BU of 6fqs by Molmil
3.11A complex of S.Aureus gyrase with imidazopyrazinone T3 and DNA
Descriptor: 5-cyclopropyl-8-fluoranyl-7-pyridin-4-yl-imidazo[1,2-a]quinoxalin-4-one, DNA (5'-D(*GP*AP*GP*AP*GP*TP*AP*T*GP*GP*CP*CP*AP*TP*AP*CP*TP*CP*TP*T)-3'), DNA gyrase subunit A, ...
Authors:Bax, B.D, Germe, T, Basque, E, Maxwell, A.
Deposit date:2018-02-14
Release date:2018-04-04
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (3.11 Å)
Cite:A new class of antibacterials, the imidazopyrazinones, reveal structural transitions involved in DNA gyrase poisoning and mechanisms of resistance.
Nucleic Acids Res., 46, 2018

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