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PDB: 7 件

4X2K
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BU of 4x2k by Molmil
Selection of fragments for kinase inhibitor design: decoration is key
分子名称: 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6H)-one, SULFATE ION, TGF-beta receptor type-1
著者Czodrowski, P, Hoelzemann, G, Barnickel, G, Greiner, H, Musil, D.
登録日2014-11-26
公開日2014-12-24
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Selection of fragments for kinase inhibitor design: decoration is key.
J.Med.Chem., 58, 2015
4X3J
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BU of 4x3j by Molmil
Selection of fragments for kinase inhibitor design: decoration is key
分子名称: 1-[4-(4-amino-5-oxopyrido[2,3-d]pyrimidin-8(5H)-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea, Angiopoietin-1 receptor
著者Czodrowski, P, Hoelzemann, G, Barnickel, G, Greiner, H, Musil, D.
登録日2014-11-30
公開日2014-12-24
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Selection of fragments for kinase inhibitor design: decoration is key.
J.Med.Chem., 58, 2015
4X2F
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BU of 4x2f by Molmil
Selection of fragments for kinase inhibitor design: decoration is key
分子名称: 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8H)-one, SULFATE ION, TGF-beta receptor type-1
著者Czodrowski, P, Hoelzemann, G, Barnickel, G, Greiner, H, Musil, D.
登録日2014-11-26
公開日2015-10-28
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Selection of fragments for kinase inhibitor design: decoration is key.
J.Med.Chem., 58, 2015
4X2N
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BU of 4x2n by Molmil
Selection of fragments for kinase inhibitor design: decoration is key
分子名称: SULFATE ION, TGF-beta receptor type-1
著者Czodrowski, P, Hoelzemann, G, Barnickel, G, Greiner, H, Musil, D.
登録日2014-11-26
公開日2014-12-24
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Selection of fragments for kinase inhibitor design: decoration is key.
J.Med.Chem., 58, 2015
4X2G
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BU of 4x2g by Molmil
Selection of fragments for kinase inhibitor design: decoration is key
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6H)-one, SULFATE ION, ...
著者Czodrowski, P, Hoelzemann, G, Barnickel, G, Greiner, H, Musil, D.
登録日2014-11-26
公開日2015-08-12
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献Selection of fragments for kinase inhibitor design: decoration is key.
J.Med.Chem., 58, 2015
4X2J
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BU of 4x2j by Molmil
Selection of fragments for kinase inhibitor design: decoration is key
分子名称: 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8H)-one, SULFATE ION, TGF-beta receptor type-1
著者Czodrowski, P, Hoelzemann, G, Barnickel, G, Greiner, H, Musil, D.
登録日2014-11-26
公開日2014-12-24
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Selection of fragments for kinase inhibitor design: decoration is key.
J.Med.Chem., 58, 2015
4X0M
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BU of 4x0m by Molmil
Selection of fragments for kinase inhibitor design: decoration is key
分子名称: 4-aminopyrido[2,3-d]pyrimidin-5(8H)-one, SULFATE ION, TGF-beta receptor type-1
著者Czodrowski, P, Hoelzemann, G, Barnickel, G, Greiner, H, Musil, D.
登録日2014-11-21
公開日2014-12-24
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献Selection of fragments for kinase inhibitor design: decoration is key.
J.Med.Chem., 58, 2015

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件を2024-05-08に公開中

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