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PDB: 1 results

5ZQU
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BU of 5zqu by Molmil
Crystal structure of tetrameric RXRalpha-LBD complexed with partial agonist CBt-PMN
Descriptor: 1-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)benzotriazole-5-carboxylic acid, BROMIDE ION, Retinoic acid receptor RXR-alpha
Authors:Miyashita, Y, Numoto, N, Arulmozhiraja, S, Nakano, S, Matsuo, N, Shimizu, K, Kakuta, H, Ito, S, Ikura, T, Ito, N, Tokiwa, H.
Deposit date:2018-04-20
Release date:2019-02-27
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (2.60038781 Å)
Cite:Dual conformation of the ligand induces the partial agonistic activity of retinoid X receptor alpha (RXR alpha ).
FEBS Lett., 593, 2019

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