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PDB: 2 results

6M1U
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BU of 6m1u by Molmil
Crystal structure of the vertebrate conserved region (VCR) of human METTL16
Descriptor: RNA N6-adenosine-methyltransferase METTL16,RNA N6-adenosine-methyltransferase METTL16
Authors:Aoyama, T, Yamashita, S, Tomita, K.
Deposit date:2020-02-26
Release date:2020-04-01
Last modified:2024-03-27
Method:X-RAY DIFFRACTION (2.791 Å)
Cite:Mechanistic insights into m6A modification of U6 snRNA by human METTL16.
Nucleic Acids Res., 48, 2020
7WOX
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BU of 7wox by Molmil
PPARgamma antagonist (MMT-160)- PPARgamma LBD complex
Descriptor: N-[[5-(3-phenylprop-2-ynoylamino)-2-propoxy-phenyl]methyl]-4-pyrimidin-2-yl-benzamide, Peroxisome proliferator-activated receptor gamma
Authors:Yoshizawa, M, Aoyama, T, Itoh, T, Miyachi, H.
Deposit date:2022-01-22
Release date:2022-04-13
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:Arylalkynyl amide-type peroxisome proliferator-activated receptor gamma (PPAR gamma )-selective antagonists covalently bind to the PPAR gamma ligand binding domain with a unique binding mode.
Bioorg.Med.Chem.Lett., 64, 2022

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PDB entries from 2024-05-01

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