7X4N
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![BU of 7x4n by Molmil](/molmil-images/mine/7x4n) | Crystal Structure of C. elegans kinesin-4 KLP-12 complexed with tubulin and DARPin | 分子名称: | DARPin, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Taguchi, S, Imasaki, T, Saijo-Hamano, Y, Sakai, N, Nitta, R. | 登録日 | 2022-03-03 | 公開日 | 2022-09-21 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.88 Å) | 主引用文献 | Structural model of microtubule dynamics inhibition by kinesin-4 from the crystal structure of KLP-12 -tubulin complex. Elife, 11, 2022
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6JZT
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![BU of 6jzt by Molmil](/molmil-images/mine/6jzt) | |
6JF2
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![BU of 6jf2 by Molmil](/molmil-images/mine/6jf2) | |
6JZR
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7WEW
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![BU of 7wew by Molmil](/molmil-images/mine/7wew) | Structure of adenylation domain of epsilon-poly-L-lysine synthase | 分子名称: | ADENOSINE-5'-[LYSYL-PHOSPHATE], Epsilon-poly-L-lysine synthase, GLYCEROL, ... | 著者 | Okamoto, T, Yamanaka, K, Hamano, Y, Nagano, S, Hino, T. | 登録日 | 2021-12-24 | 公開日 | 2022-02-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of the adenylation domain from an epsilon-poly-l-lysine synthetase provides molecular mechanism for substrate specificity Biochem.Biophys.Res.Commun., 596, 2022
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6JT3
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![BU of 6jt3 by Molmil](/molmil-images/mine/6jt3) | Crystal Structure of BACE1 in complex with N-{3-[(4R,5R,6R)-2-amino-5-fluoro-4,6-dimethyl-5,6-dihydro-4H-1,3-thiazin-4-yl]-4-fluorophenyl}-5-(fluoromethoxy)pyrazine-2-carboxamide | 分子名称: | Beta-secretase 1, DIMETHYL SULFOXIDE, GLYCEROL, ... | 著者 | Tadano, G, Komano, K, Yoshida, S, Suzuki, S, Nakahara, K, Fuchino, K, Fujimoto, K, Matsuoka, E, Yamamoto, T, Asada, N, Ito, H, Sakaguchi, G, Kanegawa, N, Kido, Y, Ando, S, Fukushima, T, Teisman, A, Urmaliya, V, Dhuyvetter, D, Borghys, H, Bergh, A.V.D, Austin, N, Gijsen, H.J.M, Yamano, Y, Iso, Y, Kusakabe, K.I. | 登録日 | 2019-04-08 | 公開日 | 2019-10-30 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Discovery of an Extremely Potent Thiazine-Based beta-Secretase Inhibitor with Reduced Cardiovascular and Liver Toxicity at a Low Projected Human Dose. J.Med.Chem., 62, 2019
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6JT4
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![BU of 6jt4 by Molmil](/molmil-images/mine/6jt4) | Crystal Structure of BACE1 in complex with N-{3-[(4S,6S)-2-amino-4-methyl-6-(trifluoromethyl)-5,6-dihydro-4H-1,3-thiazin-4-yl]-4-fluorophenyl}-5-(fluoromethoxy)pyrazine-2-carboxamide | 分子名称: | Beta-secretase 1, GLYCEROL, IODIDE ION, ... | 著者 | Anan, K, Iso, Y, Oguma, T, Nakahara, K, Suzuki, S, Yamamoto, T, Matsuoka, E, Ito, H, Sakaguchi, G, Ando, S, Morimoto, K, Kanegawa, N, Kido, Y, Kawachi, T, Fukushima, T, Teisman, A, Urmaliya, V, Dhuyvetter, D, Borghys, H, Austin, N, Bergh, A.V.D, Verboven, P, Bischoff, F, Gijsen, H.J.M, Yamano, Y, Kusakabe, K.I. | 登録日 | 2019-04-08 | 公開日 | 2020-01-15 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Trifluoromethyl Dihydrothiazine-Based beta-Secretase (BACE1) Inhibitors with Robust Central beta-Amyloid Reduction and Minimal Covalent Binding Burden. Chemmedchem, 14, 2019
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3WVR
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![BU of 3wvr by Molmil](/molmil-images/mine/3wvr) | Structure of ATP grasp protein with AMP | 分子名称: | ADENOSINE MONOPHOSPHATE, GLYCEROL, PGM1, ... | 著者 | Matsui, T, Noike, M, Ooya, K, Sasaki, I, Hamano, Y, Maruyama, C, Ishikawa, J, Satoh, Y, Ito, H, Dairi, T, Morita, H. | 登録日 | 2014-06-04 | 公開日 | 2014-11-19 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2.175 Å) | 主引用文献 | A peptide ligase and the ribosome cooperate to synthesize the peptide pheganomycin. Nat.Chem.Biol., 11, 2015
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3WVQ
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![BU of 3wvq by Molmil](/molmil-images/mine/3wvq) | Structure of ATP grasp protein | 分子名称: | GLYCEROL, PGM1, SULFATE ION | 著者 | Matsui, T, Noike, M, Ooya, K, Sasaki, I, Hamano, Y, Maruyama, C, Ishikawa, J, Satoh, Y, Ito, H, Dairi, T, Morita, H. | 登録日 | 2014-06-04 | 公開日 | 2014-11-19 | 最終更新日 | 2014-12-31 | 実験手法 | X-RAY DIFFRACTION (1.955 Å) | 主引用文献 | A peptide ligase and the ribosome cooperate to synthesize the peptide pheganomycin. Nat.Chem.Biol., 11, 2015
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