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PDB: 88675 件

7Z2P
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BU of 7z2p by Molmil
Tubulin-nocodazole complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Prota, A.E, Muehlethaler, T, Cavalli, A, Steinmetz, M.O.
登録日2022-02-28
公開日2022-08-31
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Novel fragment-derived colchicine-site binders as microtubule-destabilizing agents.
Eur.J.Med.Chem., 241, 2022
7OTS
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BU of 7ots by Molmil
Crystal structure of human Monoacylglycerol Lipase ABHD6 in complex with oleic acid and octyl glucoside
分子名称: GLYCEROL, Monoacylglycerol lipase ABHD6, OLEIC ACID, ...
著者Nawrotek, A, Talagas, A, Vuillard, L, Miallau, L.
登録日2021-06-10
公開日2021-06-23
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.792 Å)
主引用文献Crystal structure of human Monoacylglycerol Lipase ABHD6 in complex with oleic acid and octyl glucoside
To Be Published
6GIK
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BU of 6gik by Molmil
NMR structure of temporin B L1FK in SDS micelles
分子名称: temporinB_L1FK
著者Manzo, G, Mason, J.A.
登録日2018-05-12
公開日2018-06-13
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献Minor sequence modifications in temporin B cause drastic changes in antibacterial potency and selectivity by fundamentally altering membrane activity.
Sci Rep, 9, 2019
6Q2O
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BU of 6q2o by Molmil
Cryo-EM structure of RET/GFRa2/NRTN extracellular complex. The 3D refinement was applied with C2 symmetry.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, GDNF family receptor alpha-2, ...
著者Li, J, Shang, G.J, Chen, Y.J, Brautigam, C.A, Liou, J, Zhang, X.W, Bai, X.C.
登録日2019-08-08
公開日2019-10-02
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.65 Å)
主引用文献Cryo-EM analyses reveal the common mechanism and diversification in the activation of RET by different ligands.
Elife, 8, 2019
8Q79
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BU of 8q79 by Molmil
Structure of mBaoJin at pH 6.5
分子名称: CHLORIDE ION, mBaoJin
著者Samygina, V.R, Subach, O.M, Vlaskina, A.V, Nikolaeva, A.Y, Borshchevsky, V, Qin, W, Subach, F.V.
登録日2023-08-15
公開日2023-12-27
最終更新日2024-04-24
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Bright and stable monomeric green fluorescent protein derived from StayGold.
Nat.Methods, 21, 2024
7Z2N
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BU of 7z2n by Molmil
Tubulin-18-complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
著者Muehlethaler, T, Prota, A.E, Cavalli, A, Steinmetz, M.O.
登録日2022-02-28
公開日2022-08-31
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Novel fragment-derived colchicine-site binders as microtubule-destabilizing agents.
Eur.J.Med.Chem., 241, 2022
6H10
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BU of 6h10 by Molmil
Crystal Structure of KDM4D with tetrazolylhydrazide ligand NR073
分子名称: 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CHLORIDE ION, ...
著者Malecki, P.H, Weiss, M.S, Heinemann, U, Link, A.
登録日2018-07-10
公開日2020-01-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.104 Å)
主引用文献Crystal Structure of KDM4D with tetrazolylhydrazide ligand NR073
To be published
5LN4
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BU of 5ln4 by Molmil
Crystal structure of self-complemented PsaA, the major subunit of pH 6 antigen from Yersinia pests, in complex with choline
分子名称: CHOLINE ION, pH 6 antigen,pH 6 antigen
著者Pakharukova, N.A, Roy, S, Rahman, M.M, Tuitilla, M, Zavialov, A.V.
登録日2016-08-03
公開日2016-08-24
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.36 Å)
主引用文献Structural basis for Myf and Psa fimbriae-mediated tropism of pathogenic strains of Yersinia for host tissues.
Mol.Microbiol., 102, 2016
8Q4E
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BU of 8q4e by Molmil
Structure of Legionella pneumophila Lcl C-terminal domain
分子名称: HbP1
著者Rehman, S, Garnett, J.A.
登録日2023-08-06
公開日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The Legionella collagen-like protein employs a unique binding mechanism for the recognition of host glycosaminoglycans.
Biorxiv, 2023
7Z73
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BU of 7z73 by Molmil
Crystal structure of p63 tetramerization domain in complex with darpin 8F1
分子名称: Darpin 8F1, Isoform 2 of Tumor protein 63
著者Chaikuad, A, Strubel, A, Doetsch, V, Knapp, S, Structural Genomics Consortium (SGC)
登録日2022-03-14
公開日2022-07-06
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.27 Å)
主引用文献Designed Ankyrin Repeat Proteins as a tool box for analyzing p63.
Cell Death Differ., 29, 2022
7PV2
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BU of 7pv2 by Molmil
GA1 bacteriophage portal protein
分子名称: Head-tail connector (Portal protein)
著者Javed, A, Villanueva, H, Orlova, E.V, Savva, R.
登録日2021-10-01
公開日2022-10-12
最終更新日2023-10-25
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Cryo-EM Structures of Two Bacteriophage Portal Proteins Provide Insights for Antimicrobial Phage Engineering.
Viruses, 13, 2021
8QK8
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BU of 8qk8 by Molmil
Structure of Legionella pneumophila Lcl C-terminal domain bound to sulphate
分子名称: HbP1, SULFATE ION
著者Rehman, S, Garnett, J.A.
登録日2023-09-14
公開日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The Legionella collagen-like protein employs a unique binding mechanism for the recognition of host glycosaminoglycans.
Biorxiv, 2023
7TZ4
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BU of 7tz4 by Molmil
Salicylate Adenylate PchD from Pseudomonas aeruginosa containing 4-cyanosalicyl-AMS
分子名称: 5'-O-[(4-cyano-2-hydroxybenzoyl)sulfamoyl]adenosine, Pyochelin biosynthesis salicyl-AMP ligase PchD
著者Shelton, C.L, Meneely, K.M, Lamb, A.L.
登録日2022-02-15
公開日2022-05-18
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Rational inhibitor design for Pseudomonas aeruginosa salicylate adenylation enzyme PchD.
J.Biol.Inorg.Chem., 27, 2022
8QDD
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BU of 8qdd by Molmil
Structure of mBaoJin at pH 8.5
分子名称: CHLORIDE ION, SULFATE ION, mBaoJin
著者Samygina, V.R, Vlaskina, A.V, Gabdulkhakov, A, Subach, O.M, Subach, F.V.
登録日2023-08-28
公開日2023-12-27
最終更新日2024-04-24
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Bright and stable monomeric green fluorescent protein derived from StayGold.
Nat.Methods, 21, 2024
7TYB
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BU of 7tyb by Molmil
Salicylate Adenylate PchD from Pseudomonas aeruginosa containing salicyl-AMS
分子名称: 5'-O-[(2-hydroxybenzoyl)sulfamoyl]adenosine, Pyochelin biosynthesis protein PchD
著者Meneely, K.M, Shelton, C.L, Lamb, A.L.
登録日2022-02-11
公開日2022-05-18
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献Rational inhibitor design for Pseudomonas aeruginosa salicylate adenylation enzyme PchD.
J.Biol.Inorg.Chem., 27, 2022
6NFD
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BU of 6nfd by Molmil
beta-lactamase SHV-11 from Klebsiella pneumoniae strain NTUH-K2044
分子名称: 1,2-ETHANEDIOL, PHOSPHATE ION, beta-lactamase SHV-11
著者Osipiuk, J, Welk, L, Endres, M, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID)
登録日2018-12-19
公開日2018-12-26
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.17 Å)
主引用文献beta-lactamase SHV-11 from Klebsiella pneumoniae strain NTUH-K2044
to be published
5KGA
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BU of 5kga by Molmil
X-ray structure of a glucosamine N-Acetyltransferase from Clostridium acetobutylicum, mutant D287N, in complex with N-acetylglucosamine
分子名称: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYL COENZYME *A, ...
著者Dopkins, B.J, Thoden, J.B, Tipton, P.A, Holden, H.M.
登録日2016-06-13
公開日2016-07-06
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Studies on a Glucosamine/Glucosaminide N-Acetyltransferase.
Biochemistry, 55, 2016
4WKN
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BU of 4wkn by Molmil
Crystal structure of Helicobacter pylori 5'-methylthioadenosine/S-adenosyl homocysteine nucleosidase (MTAN) complexed with methylthio-DADMe-Immucillin-A
分子名称: (3R,4S)-1-[(4-AMINO-5H-PYRROLO[3,2-D]PYRIMIDIN-7-YL)METHYL]-4-[(METHYLSULFANYL)METHYL]PYRROLIDIN-3-OL, Aminodeoxyfutalosine nucleosidase
著者Cameron, S.A, Wang, S, Almo, S.C, Schramm, V.L.
登録日2014-10-02
公開日2015-11-25
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献New Antibiotic Candidates against Helicobacter pylori.
J.Am.Chem.Soc., 137, 2015
5KGJ
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BU of 5kgj by Molmil
X-ray structure of a glucosamine N-Acetyltransferase from Clostridium acetobutylicum in complex with galactosamine
分子名称: 1,2-ETHANEDIOL, 2-amino-2-deoxy-alpha-D-galactopyranose, 3-[4-(2-HYDROXYETHYL)PIPERAZIN-1-YL]PROPANE-1-SULFONIC ACID, ...
著者Dopkins, B.J, Thoden, J.B, Tipton, P.A, Holden, H.M.
登録日2016-06-13
公開日2016-07-06
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Studies on a Glucosamine/Glucosaminide N-Acetyltransferase.
Biochemistry, 55, 2016
5D91
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BU of 5d91 by Molmil
Structure of a phosphatidylinositolphosphate (PIP) synthase from Renibacterium Salmoninarum
分子名称: AF2299 protein,Phosphatidylinositol synthase, MAGNESIUM ION, Octadecane, ...
著者Clarke, O.B, Tomasek, D.T, Jorge, C.D, Belcher Dufrisne, M, Kim, M, Banerjee, S, Rajashankar, K.R, Hendrickson, W.A, Santos, H, Mancia, F.
登録日2015-08-18
公開日2015-11-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.501 Å)
主引用文献Structural basis for phosphatidylinositol-phosphate biosynthesis.
Nat Commun, 6, 2015
6GRG
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BU of 6grg by Molmil
E. coli Microcin synthetase McbBCD complex with pro-MccB17, ADP and phosphate bound
分子名称: 1,2-ETHANEDIOL, ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ...
著者Ghilarov, D, Stevenson, C.E.M, Travin, D.Y, Piskunova, J, Serebryakova, M, Maxwell, A, Lawson, D.M, Severinov, K.
登録日2018-06-11
公開日2019-01-30
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Architecture of Microcin B17 Synthetase: An Octameric Protein Complex Converting a Ribosomally Synthesized Peptide into a DNA Gyrase Poison.
Mol. Cell, 73, 2019
8UW3
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BU of 8uw3 by Molmil
Human LINE-1 retrotransposon ORF2 protein engaged with template RNA in elongation state
分子名称: Complementary DNA, LINE-1 retrotransposable element ORF2 protein, THYMIDINE-5'-TRIPHOSPHATE, ...
著者Thawani, A, Florez Ariza, A.J, Collins, K, Nogales, E.
登録日2023-11-06
公開日2023-12-20
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Template and target-site recognition by human LINE-1 in retrotransposition.
Nature, 626, 2024
8URW
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BU of 8urw by Molmil
Cyanobacterial RNA polymerase elongation complex with NusG and CTP
分子名称: CYTIDINE-5'-TRIPHOSPHATE, DNA (40-MER), DNA-directed RNA polymerase subunit alpha, ...
著者Qayyum, M.Z, Imashimizu, M, Leanca, M, Vishwakarma, R.K, Bradley Riaz, A, Yuzenkova, Y, Murakami, K.S.
登録日2023-10-26
公開日2023-12-27
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (2.79 Å)
主引用文献Structure and function of the Si3 insertion integrated into the trigger loop/helix of cyanobacterial RNA polymerase.
Proc.Natl.Acad.Sci.USA, 121, 2024
5JYT
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BU of 5jyt by Molmil
NMR structure of foldswitch-stablized KaiB from Thermosynechococcus elongatus
分子名称: Circadian clock protein KaiB
著者Tseng, R.D, LiWang, A.L.
登録日2016-05-15
公開日2017-03-29
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural basis of the day-night transition in a bacterial circadian clock.
Science, 355, 2017
8Q7Y
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BU of 8q7y by Molmil
ESIBD structure of beta-galactosidase
分子名称: Beta-galactosidase
著者Esser, T, Boehning, J, Bharat, T.A.M, Rauschenbach, S.
登録日2023-08-17
公開日2024-01-10
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (2.6 Å)
主引用文献Cryo-EM of soft-landed beta-galactosidase: Gas-phase and native structures are remarkably similar.
Sci Adv, 10, 2024

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