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2Z5B
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BU of 2z5b by Molmil
Crystal Structure of a Novel Chaperone Complex for Yeast 20S Proteasome Assembly
分子名称: Protein YPL144W, Uncharacterized protein YLR021W
著者Yashiroda, H, Mizushima, T, Okamoto, K, Kameyama, T, Hayashi, H, Kishimoto, T, Kasahara, M, Kurimoto, E, Sakata, E, Suzuki, A, Hirano, Y, Murata, S, Kato, K, Yamane, T, Tanaka, K.
登録日2007-07-03
公開日2008-01-22
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Crystal structure of a chaperone complex that contributes to the assembly of yeast 20S proteasomes
Nat.Struct.Mol.Biol., 15, 2008
2Z5C
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BU of 2z5c by Molmil
Crystal Structure of a Novel Chaperone Complex for Yeast 20S Proteasome Assembly
分子名称: Proteasome component PUP2, Protein YPL144W, Uncharacterized protein YLR021W
著者Yashiroda, H, Mizushima, T, Okamoto, K, Kameyama, T, Hayashi, H, Kishimoto, T, Kasahara, M, Kurimoto, E, Sakata, E, Suzuki, A, Hirano, Y, Murata, S, Kato, K, Yamane, T, Tanaka, K.
登録日2007-07-03
公開日2008-01-22
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of a chaperone complex that contributes to the assembly of yeast 20S proteasomes
Nat.Struct.Mol.Biol., 15, 2008
3WXR
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BU of 3wxr by Molmil
Yeast 20S proteasome with a mutation of alpha7 subunit
分子名称: Probable proteasome subunit alpha type-7, Proteasome subunit alpha type-1, Proteasome subunit alpha type-2, ...
著者Yashiroda, H, Toda, Y, Otsu, S, Takagi, K, Mizushima, T, Murata, S.
登録日2014-08-06
公開日2014-10-22
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献N-terminal alpha 7 deletion of the proteasome 20S core particle substitutes for yeast PI31 function
Mol.Cell.Biol., 35, 2015
3VW6
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BU of 3vw6 by Molmil
Crystal structure of human apoptosis signal-regulating kinase 1 (ASK1) with imidazopyridine inhibitor
分子名称: 4-tert-butyl-N-[6-(1H-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide, Mitogen-activated protein kinase kinase kinase 5
著者Terao, Y, Suzuki, H, Yoshikawa, M, Yashiro, H, Takekawa, S, Fujitani, Y, Okada, K, Inoue, Y, Yamamoto, Y, Nakagawa, H, Yao, S, Kawamoto, T, Uchikawa, O.
登録日2012-08-06
公開日2012-10-31
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Design and biological evaluation of imidazo[1,2-a]pyridines as novel and potent ASK1 inhibitors.
Bioorg. Med. Chem. Lett., 22, 2012
3WWG
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BU of 3wwg by Molmil
Crystal structure of the N-glycan-deficient variant N448A of isopullulanase complexed with isopanose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Isopullulanase, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ...
著者Miyazaki, T, Yashiro, H, Nishikawa, A, Tonozuka, T.
登録日2014-06-17
公開日2014-11-12
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The side chain of a glycosylated asparagine residue is important for the stability of isopullulanase
J.Biochem., 157, 2015
2Z5E
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BU of 2z5e by Molmil
Crystal Structure of Proteasome Assembling Chaperone 3
分子名称: Proteasome Assembling Chaperone 3
著者Okamoto, K, Kurimoto, E, Sakata, E, Suzuki, A, Yamane, T, Hirano, Y, Murata, S, Tanaka, K, Kato, K.
登録日2007-07-06
公開日2008-02-19
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of a chaperone complex that contributes to the assembly of yeast 20S proteasomes
Nat.Struct.Mol.Biol., 15, 2008
3O95
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BU of 3o95 by Molmil
Crystal Structure of Human DPP4 Bound to TAK-100
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Yano, J.K, Aertgeerts, K.
登録日2010-08-03
公開日2011-01-26
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Discovery of a 3-Pyridylacetic Acid Derivative (TAK-100) as a Potent, Selective and Orally Active Dipeptidyl Peptidase IV (DPP-4) Inhibitor.
J.Med.Chem., 53, 2011
3O9V
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BU of 3o9v by Molmil
Crystal Structure of Human DPP4 Bound to TAK-986
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-(aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-methylpropyl)pyridine-3-carboxic acid, ...
著者Yano, J.K, Aertgeerts, K.
登録日2010-08-04
公開日2011-02-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Discovery of a 3-Pyridylacetic Acid Derivative (TAK-100) as a Potent, Selective and Orally Active Dipeptidyl Peptidase IV (DPP-4) Inhibitor.
J.Med.Chem., 53, 2011

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件を2024-05-01に公開中

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