1A0O
| CHEY-BINDING DOMAIN OF CHEA IN COMPLEX WITH CHEY | 分子名称: | CHEA, CHEY, MANGANESE (II) ION | 著者 | Chinardet, N, Welch, M, Mourey, L, Birck, C, Samama, J.P. | 登録日 | 1997-12-05 | 公開日 | 1998-12-30 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Structure of the CheY-binding domain of histidine kinase CheA in complex with CheY. Nat.Struct.Biol., 5, 1998
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5M2E
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7OO1
| Structure, function and characterization of a second pyruvate kinase isozyme in Pseudomonas aeruginosa. | 分子名称: | Pyruvate kinase | 著者 | Abdelhamid, Y, Wang, M, Parkhill, S, Brear, P, Welch, M. | 登録日 | 2021-05-26 | 公開日 | 2021-11-03 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (3.01 Å) | 主引用文献 | Structure, Function and Regulation of a Second Pyruvate Kinase Isozyme in Pseudomonas aeruginosa Front Microbiol, 12, 2021
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6ZU0
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5OAS
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1FFS
| CHEY-BINDING DOMAIN OF CHEA IN COMPLEX WITH CHEY FROM CRYSTALS SOAKED IN ACETYL PHOSPHATE | 分子名称: | CHEMOTAXIS PROTEIN CHEA, CHEMOTAXIS PROTEIN CHEY, MANGANESE (II) ION | 著者 | Gouet, P, Chinardet, N, Welch, M, Guillet, V, Birck, C, Mourey, L, Samama, J.-P. | 登録日 | 2000-07-26 | 公開日 | 2001-01-17 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Further insights into the mechanism of function of the response regulator CheY from crystallographic studies of the CheY--CheA(124--257) complex. Acta Crystallogr.,Sect.D, 57, 2001
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1FFG
| CHEY-BINDING DOMAIN OF CHEA IN COMPLEX WITH CHEY AT 2.1 A RESOLUTION | 分子名称: | CHEMOTAXIS PROTEIN CHEA, CHEMOTAXIS PROTEIN CHEY, MANGANESE (II) ION | 著者 | Gouet, P, Chinardet, N, Welch, M, Guillet, V, Birck, C, Mourey, L, Samama, J.-P. | 登録日 | 2000-07-25 | 公開日 | 2001-01-17 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Further insights into the mechanism of function of the response regulator CheY from crystallographic studies of the CheY--CheA(124--257) complex. Acta Crystallogr.,Sect.D, 57, 2001
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1FFW
| CHEY-BINDING DOMAIN OF CHEA IN COMPLEX WITH CHEY WITH A BOUND IMIDO DIPHOSPHATE | 分子名称: | CHEMOTAXIS PROTEIN CHEA, CHEMOTAXIS PROTEIN CHEY, IMIDO DIPHOSPHATE, ... | 著者 | Gouet, P, Chinardet, N, Welch, M, Guillet, V, Birck, C, Mourey, L, Samama, J.-P. | 登録日 | 2000-07-26 | 公開日 | 2001-01-17 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Further insights into the mechanism of function of the response regulator CheY from crystallographic studies of the CheY--CheA(124--257) complex. Acta Crystallogr.,Sect.D, 57, 2001
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6G1O
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6G3U
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6T5M
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6T4V
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6QXL
| Crystal Structure of Pyruvate Kinase II (PykA) from Pseudomonas aeruginosa in complex with sodium malonate, magnesium and glucose-6-phosphate | 分子名称: | 6-O-phosphono-alpha-D-glucopyranose, GLYCEROL, MAGNESIUM ION, ... | 著者 | Abdelhamid, Y, Brear, P, Welch, M. | 登録日 | 2019-03-07 | 公開日 | 2019-09-11 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.43 Å) | 主引用文献 | Evolutionary plasticity in the allosteric regulator-binding site of pyruvate kinase isoform PykA fromPseudomonas aeruginosa. J.Biol.Chem., 294, 2019
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6S62
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6S87
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6S6F
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2GFS
| P38 Kinase Crystal Structure in complex with RO3201195 | 分子名称: | Mitogen-Activated Protein Kinase 14, [5-AMINO-1-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL](3-{[(2R)-2,3-DIHYDROXYPROPYL]OXY}PHENYL)METHANONE | 著者 | Harris, S.F, Bertrand, J, Villasenor, A. | 登録日 | 2006-03-23 | 公開日 | 2006-04-18 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.752 Å) | 主引用文献 | Discovery of S-[5-Amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(2,3-dihydroxypropoxy)phenyl]-methanone (RO3201195), and Orally Bioavailable and Highly Selective Inhibitor of p38 Map Kinase J.Med.Chem., 49, 2006
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3D4Q
| Pyrazole-based inhibitors of B-Raf kinase | 分子名称: | (1E)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1H-pyrazol-4-yl)-2,3-dihydro-1H-inden-1-one oxime, B-Raf proto-oncogene serine/threonine-protein kinase | 著者 | Morales, T, Vigers, G.P.A, Brandhuber, B.J. | 登録日 | 2008-05-14 | 公開日 | 2008-08-19 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Potent and selective pyrazole-based inhibitors of B-Raf kinase. Bioorg.Med.Chem.Lett., 18, 2008
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3PSD
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3PSB
| Furo[2,3-c]pyridine-based Indanone Oximes as Potent and Selective B-Raf Inhibitors | 分子名称: | B-RAF PROTO-ONCOGENE SERINE/THREONINE-PROTEIN KINASE, ethyl 3-{[1-(hydroxyamino)-2H-inden-5-yl]amino}thieno[2,3-c]pyridine-2-carboxylate | 著者 | Morales, T, Vigers, G.P.A, Brandhuber, B.J. | 登録日 | 2010-12-01 | 公開日 | 2011-01-19 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | The Discovery of furo[2,3-c]pyridine-based indanone oximes as potent and selective B-Raf inhibitors. Bioorg.Med.Chem.Lett., 21, 2011
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1OZ1
| P38 MITOGEN-ACTIVATED KINASE IN COMPLEX WITH 4-AZAINDOLE INHIBITOR | 分子名称: | 3-(4-FLUOROPHENYL)-2-PYRIDIN-4-YL-1H-PYRROLO[3,2-B]PYRIDIN-1-OL, Mitogen-activated protein kinase 14 | 著者 | Lovejoy, B, Villasenor, A, Browner, M, Dunten, P. | 登録日 | 2003-04-07 | 公開日 | 2003-09-23 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Design and synthesis of 4-azaindoles as inhibitors of p38 MAP kinase. J.Med.Chem., 46, 2003
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1FFZ
| LARGE RIBOSOMAL SUBUNIT COMPLEXED WITH R(CC)-DA-PUROMYCIN | 分子名称: | 23S RIBOSOMAL RNA, R(P*CP*C*)-D(P*A)-R(P*(PU)) | 著者 | Nissen, P, Hansen, J, Ban, N, Moore, P.B, Steitz, T.A. | 登録日 | 2000-07-26 | 公開日 | 2000-08-28 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | The structural basis of ribosome activity in peptide bond synthesis. Science, 289, 2000
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8RQO
| Human thyroid hormone receptor alpha ligand binding domain in complex with beta-selective agonist ALG-055009 | 分子名称: | 6-azanyl-2-[3,5-bis(chloranyl)-4-[(6-oxidanylidene-5-propan-2-yl-1~{H}-pyridazin-3-yl)oxy]phenyl]-1,2,4-triazine-3,5-dione, Isoform Alpha-1 of Thyroid hormone receptor alpha, SULFATE ION | 著者 | Lammens, A, Maskos, K, Stoycheva, A.D, McGowan, D.C. | 登録日 | 2024-01-18 | 公開日 | 2024-09-11 | 実験手法 | X-RAY DIFFRACTION (2.74 Å) | 主引用文献 | Discovery and Preclinical Profile of ALG-055009, a Potent and Selective Thyroid Hormone Receptor Beta (THR-beta ) Agonist for the Treatment of MASH. J.Med.Chem., 2024
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8RQN
| Human thyroid hormone receptor beta ligand binding domain in complex with beta-selective agonist ALG-055009 | 分子名称: | 6-azanyl-2-[3,5-bis(chloranyl)-4-[(6-oxidanylidene-5-propan-2-yl-1~{H}-pyridazin-3-yl)oxy]phenyl]-1,2,4-triazine-3,5-dione, Thyroid hormone receptor beta | 著者 | Lammens, A, Maskos, K, Stoycheva, A.D, McGowan, D.C. | 登録日 | 2024-01-18 | 公開日 | 2024-09-11 | 実験手法 | X-RAY DIFFRACTION (2.88 Å) | 主引用文献 | Discovery and Preclinical Profile of ALG-055009, a Potent and Selective Thyroid Hormone Receptor Beta (THR-beta ) Agonist for the Treatment of MASH. J.Med.Chem., 2024
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