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1U8G
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Crystal structure of a HIV-1 Protease in complex with peptidomimetic inhibitor KI2-PHE-GLU-GLU-NH2
分子名称: PROTEASE RETROPEPSIN, peptidomimetic inhibitor KI2-PHE-GLU-GLU-NH2
著者Brynda, J, Rezacova, P, Fabry, M, Horejsi, M, Hradilek, M, Soucek, R, Stouracova, R, Konvalinka, J, Sedlacek, J.
登録日2004-08-06
公開日2004-11-02
最終更新日2018-02-14
実験手法X-RAY DIFFRACTION (2.201 Å)
主引用文献Inhibitor binding at the protein interface in crystals of a HIV-1 protease complex.
Acta Crystallogr.,Sect.D, 60, 2004
1MF2
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ANTI HIV1 PROTEASE FAB COMPLEX
分子名称: MONOCLONAL ANTIBODY F11.2.32
著者Lescar, J, Bentley, G.A.
登録日1996-12-27
公開日1997-12-31
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Three-dimensional structure of an Fab-peptide complex: structural basis of HIV-1 protease inhibition by a monoclonal antibody.
J.Mol.Biol., 267, 1997
1CL7
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ANTI HIV1 PROTEASE FAB
分子名称: PROTEIN (IGG1 ANTIBODY 1696 (constant heavy chain)), PROTEIN (IGG1 ANTIBODY 1696 (light chain)), PROTEIN (IGG1 ANTIBODY 1696 (variable heavy chain))
著者Lescar, J, Bentley, G.A.
登録日1999-05-06
公開日2000-01-12
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Inhibition of the HIV-1 and HIV-2 proteases by a monoclonal antibody.
Protein Sci., 8, 1999
2HRP
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ANTIGEN-ANTIBODY COMPLEX
分子名称: HIV-1 PROTEASE PEPTIDE, MONOCLONAL ANTIBODY F11.2.32
著者Lescar, J, Bentley, G.A.
登録日1996-12-27
公開日1997-12-31
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Three-dimensional structure of an Fab-peptide complex: structural basis of HIV-1 protease inhibition by a monoclonal antibody.
J.Mol.Biol., 267, 1997
1NH0
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1.03 A structure of HIV-1 protease: inhibitor binding inside and outside the active site
分子名称: BETA-MERCAPTOETHANOL, PROTEASE RETROPEPSIN, SULFATE ION, ...
著者Brynda, J, Rezacova, P, Fabry, M, Horejsi, M, Hradilek, M, Soucek, M, Konvalinka, J, Sedlacek, J.
登録日2002-12-18
公開日2004-04-13
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.03 Å)
主引用文献A Phenylnorstatine Inhibitor Binding to HIV-1 Protease: Geometry, Protonation, and Subsite-Pocket Interactions Analyzed at Atomic Resolution
J.Med.Chem., 47, 2004
2HKH
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Crystal structure of the Fab M75
分子名称: GLYCEROL, Immunoglobulin Heavy chain Fab fragment, Immunoglobulin Light chain Fab fragment
著者Kral, V, Mader, P, Stouracova, R, Fabry, M, Sedlacek, J, Brynda, J.
登録日2006-07-04
公開日2007-11-13
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Stabilization of antibody structure upon association to a human carbonic anhydrase IX epitope studied by X-ray crystallography, microcalorimetry, and molecular dynamics simulations.
Proteins, 71, 2008
2HKF
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Crystal structure of the Complex Fab M75- Peptide
分子名称: Carbonic anhydrase 9, Immunoglobulin Heavy chain Fab fragment, Immunoglobulin Light chain Fab fragment
著者Kral, V, Mader, P, Stouracova, R, Fabry, M, Horejsi, M, Brynda, J.
登録日2006-07-04
公開日2007-11-13
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Stabilization of antibody structure upon association to a human carbonic anhydrase IX epitope studied by X-ray crystallography, microcalorimetry, and molecular dynamics simulations.
Proteins, 71, 2008

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件を2024-05-15に公開中

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