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4DG4
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BU of 4dg4 by Molmil
Human mesotrypsin-S39Y complexed with bovine pancreatic trypsin inhibitor (BPTI)
Descriptor: CALCIUM ION, PRSS3 protein, Pancreatic trypsin inhibitor, ...
Authors:Salameh, M.A, Soares, A.S, Radisky, E.S.
Deposit date:2012-01-24
Release date:2012-09-12
Last modified:2018-01-24
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:Presence versus absence of hydrogen bond donor Tyr-39 influences interactions of cationic trypsin and mesotrypsin with protein protease inhibitors.
Protein Sci., 21, 2012
3L3T
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BU of 3l3t by Molmil
Human mesotrypsin complexed with amyloid precursor protein inhibitor variant (APPIR15K)
Descriptor: CALCIUM ION, FORMIC ACID, PRSS3 protein, ...
Authors:Salameh, M.A, Soares, A.S, Radisky, E.S.
Deposit date:2009-12-17
Release date:2010-09-22
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.378 Å)
Cite:Determinants of affinity and proteolytic stability in interactions of Kunitz family protease inhibitors with mesotrypsin.
J.Biol.Chem., 285, 2010
3L33
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BU of 3l33 by Molmil
Human mesotrypsin complexed with amyloid precursor protein inhibitor(APPI)
Descriptor: Amyloid beta A4 protein, CALCIUM ION, FORMIC ACID, ...
Authors:Salameh, M.A, Soares, A.S, Radisky, E.S.
Deposit date:2009-12-16
Release date:2010-09-22
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.48 Å)
Cite:Determinants of affinity and proteolytic stability in interactions of Kunitz family protease inhibitors with mesotrypsin.
J.Biol.Chem., 285, 2010
3P92
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BU of 3p92 by Molmil
Human mesotrypsin complexed with bovine pancreatic trypsin inhibitor variant (BPTI-K15R/R17G)
Descriptor: CALCIUM ION, PRSS3 protein, Pancreatic trypsin inhibitor
Authors:Salameh, M.A, Soares, A.S, Radisky, E.S.
Deposit date:2010-10-15
Release date:2011-08-31
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.5992 Å)
Cite:The P2' residue is a key determinant of mesotrypsin specificity: engineering a high-affinity inhibitor with anticancer activity.
Biochem.J., 440, 2011
3P95
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BU of 3p95 by Molmil
Human mesotrypsin complexed with bovine pancreatic trypsin inhibitor variant (BPTI-K15R/R17D)
Descriptor: CALCIUM ION, PRSS3 protein, Pancreatic trypsin inhibitor
Authors:Salameh, M.A, Soares, A.S, Radisky, E.S.
Deposit date:2010-10-15
Release date:2011-08-31
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.2991 Å)
Cite:The P2' residue is a key determinant of mesotrypsin specificity: engineering a high-affinity inhibitor with anticancer activity.
Biochem.J., 440, 2011
2RA3
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BU of 2ra3 by Molmil
Human cationic trypsin complexed with bovine pancreatic trypsin inhibitor (BPTI)
Descriptor: CALCIUM ION, Pancreatic trypsin inhibitor, SULFATE ION, ...
Authors:Salameh, M.A, Soares, A.S, Radisky, E.S.
Deposit date:2007-09-14
Release date:2007-12-11
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (1.46 Å)
Cite:Structural Basis for Accelerated Cleavage of Bovine Pancreatic Trypsin Inhibitor (BPTI) by Human Mesotrypsin.
J.Biol.Chem., 283, 2008
2R9P
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BU of 2r9p by Molmil
Human mesotrypsin complexed with bovine pancreatic trypsin inhibitor(BPTI)
Descriptor: Pancreatic trypsin inhibitor, SULFATE ION, Trypsin-3
Authors:Salameh, M.A, Soares, A.S, Radisky, E.S.
Deposit date:2007-09-13
Release date:2007-12-11
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:Structural Basis for Accelerated Cleavage of Bovine Pancreatic Trypsin Inhibitor (BPTI) by Human Mesotrypsin.
J.Biol.Chem., 283, 2008

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