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STRUCTURE OF A RETRO-BINDING PEPTIDE INHIBITOR COMPLEXED WITH HUMAN ALPHA-THROMBIN
Descriptor:	ALPHA-THROMBIN, HIRUGEN PEPTIDE, methyl N-(4-carbamimidamidobutanoyl)-L-phenylalanyl-L-allothreonyl-L-phenylalaninate
Authors:	Tabernero, L, Sack, J.
Deposit date:	1994-07-25
Release date:	1995-10-15
Last modified:	2012-12-12
Method:	X-RAY DIFFRACTION (2.6 Å)
Cite:	Structure of a retro-binding peptide inhibitor complexed with human alpha-thrombin. J.Mol.Biol., 246, 1995

CRYSTAL STRUCTURE OF RAR-RELATED ORPHAN RECEPTOR C (NHIS-RORGT(244-487)-L6-SRC1(6T78-692) IN COMPLEX WITH A TRICYCLIC SULFONE RORGT INVERSE AGONIST
Descriptor:	Nuclear receptor ROR-gamma, trans-4-[(3aR,9bR)-8-cyano-9b-[(4-fluorophenyl)sulfonyl]-7-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-1,2,3a,4,5,9b-hexahydro-3H-benzo[e]indole-3-carbonyl]cyclohexane-1-carboxylic acid
Authors:	Sack, J.S.
Deposit date:	2020-08-18
Release date:	2020-09-16
Last modified:	2023-10-18
Method:	X-RAY DIFFRACTION (2.43 Å)
Cite:	Tricyclic sulfones as potent, selective and efficacious ROR gamma t inverse agonists - Exploring C6 and C8 SAR using late-stage functionalization. Bioorg.Med.Chem.Lett., 30, 2020