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1NI4
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BU of 1ni4 by Molmil
HUMAN PYRUVATE DEHYDROGENASE
分子名称: MAGNESIUM ION, POTASSIUM ION, Pyruvate dehydrogenase E1 component: Alpha subunit, ...
著者Ciszak, E, Korotchkina, L.G, Dominiak, P.M, Sidhu, S, Patel, M.S.
登録日2002-12-20
公開日2003-06-17
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structural Basis for Flip-Flop Action of Thiamin Pyrophosphate-Dependent Enzymes Revealed by Human Pyruvate Dehydrogenase
J.Biol.Chem., 278, 2003
1ZY8
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BU of 1zy8 by Molmil
The crystal structure of dihydrolipoamide dehydrogenase and dihydrolipoamide dehydrogenase-binding protein (didomain) subcomplex of human pyruvate dehydrogenase complex.
分子名称: Dihydrolipoyl dehydrogenase, mitochondrial, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Ciszak, E.M, Makal, A, Hong, Y.S, Vettaikkorumakankauv, A.K, Korotchkina, L.G, Patel, M.S.
登録日2005-06-09
公開日2005-11-15
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.59 Å)
主引用文献How Dihydrolipoamide Dehydrogenase-binding Protein Binds Dihydrolipoamide Dehydrogenase in the Human Pyruvate Dehydrogenase Complex.
J.Biol.Chem., 281, 2006
2OZL
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BU of 2ozl by Molmil
Human pyruvate dehydrogenase S264E variant
分子名称: MAGNESIUM ION, POTASSIUM ION, Pyruvate dehydrogenase E1 component alpha subunit, ...
著者Ciszak, E.M, Dominiak, P.M, Patel, M.S, Korotchkina, L.G.
登録日2007-02-26
公開日2007-05-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Phosphorylation of Serine 264 Impedes Active Site Accessibility in the E1 Component of the Human Pyruvate Dehydrogenase Multienzyme Complex
Biochemistry, 46, 2007
6H60
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BU of 6h60 by Molmil
pseudo-atomic structural model of the E3BP component of the human pyruvate dehydrogenase multienzyme complex
分子名称: Pyruvate dehydrogenase protein X component, mitochondrial
著者Haselbach, D, Prajapati, S, Tittmann, K, Stark, H.
登録日2018-07-25
公開日2019-06-05
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (6 Å)
主引用文献Structural and Functional Analyses of the Human PDH Complex Suggest a "Division-of-Labor" Mechanism by Local E1 and E3 Clusters.
Structure, 27, 2019
6H55
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BU of 6h55 by Molmil
core of the human pyruvate dehydrogenase (E2)
分子名称: Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, mitochondrial
著者Haselbach, D, Prajapati, S, Tittmann, K, Stark, H.
登録日2018-07-23
公開日2019-06-05
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (6 Å)
主引用文献Structural and Functional Analyses of the Human PDH Complex Suggest a "Division-of-Labor" Mechanism by Local E1 and E3 Clusters.
Structure, 27, 2019
3II4
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BU of 3ii4 by Molmil
Structure of mycobacterial lipoamide dehydrogenase bound to a triazaspirodimethoxybenzoyl inhibitor
分子名称: Dihydrolipoyl dehydrogenase, FLAVIN-ADENINE DINUCLEOTIDE, N-[2-(2,4-dichlorophenyl)ethyl]-2-{8-[(2,4-dimethoxyphenyl)carbonyl]-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]dec-3-yl}acetamide
著者Lima, C.D.
登録日2009-07-31
公開日2010-01-26
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.42 Å)
主引用文献Triazaspirodimethoxybenzoyls as selective inhibitors of mycobacterial lipoamide dehydrogenase .
Biochemistry, 49, 2010
6CER
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BU of 6cer by Molmil
Human pyruvate dehydrogenase complex E1 component V138M mutation
分子名称: MAGNESIUM ION, Pyruvate dehydrogenase E1 component subunit alpha, somatic form, ...
著者Whitley, M.J, Arjunan, P, Furey, W.
登録日2018-02-12
公開日2018-07-11
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.69 Å)
主引用文献Pyruvate dehydrogenase complex deficiency is linked to regulatory loop disorder in the alpha V138M variant of human pyruvate dehydrogenase.
J. Biol. Chem., 293, 2018
6CFO
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BU of 6cfo by Molmil
HUMAN PYRUVATE DEHYDROGENASE E1 COMPONENT COMPLEX WITH COVALENT TDP ADDUCT ACETYL PHOSPHINATE
分子名称: 3-[(4-amino-2-methylpyrimidin-5-yl)methyl]-2-{(1S)-1-hydroxy-1-[(R)-hydroxy(oxo)-lambda~5~-phosphanyl]ethyl}-5-(2-{[(S)-hydroxy(phosphonooxy)phosphoryl]oxy}ethyl)-4-methyl-1,3-thiazol-3-ium, MAGNESIUM ION, Pyruvate dehydrogenase E1 component subunit alpha, ...
著者ARJUNAN, P, WHITLEY, M.J, FUREY, W.
登録日2018-02-15
公開日2018-07-11
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Pyruvate dehydrogenase complex deficiency is linked to regulatory loop disorder in the alpha V138M variant of human pyruvate dehydrogenase.
J. Biol. Chem., 293, 2018

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