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Novel Inhibitors of Bacterial Methionine Aminopeptidase with Broad-Spectrum Biochemical Activity
Descriptor:	MANGANESE (II) ION, Methionine aminopeptidase, N~2~-[(3,5-difluorophenyl)acetyl]-N-[(3S,7R)-1-methyl-2-oxo-7-phenyl-2,3,4,7-tetrahydro-1H-azepin-3-yl]-L-alaninamide
Authors:	Rose, J.A, Lahiri, S.D, McKinney, D.C, Albert, R, Morningstar, M, Shapiro, A.B, Fisher, S.F, Fleming, P.R.
Deposit date:	2015-04-07
Release date:	2016-04-13
Last modified:	2024-03-06
Method:	X-RAY DIFFRACTION (1.43 Å)
Cite:	Novel Inhibitors of Bacterial Methionine Aminopeptidase with Broad-Spectrum Biochemical Activity To be Published

Crystal structure of Helicobacter pylori glutamate racemase in complex with D-Glutamate and an inhibitor
Descriptor:	1-[(3S)-5-PHENYL-3-THIOPHEN-2-YL-3H-1,4-BENZODIAZEPIN-2-YL]AZETIDIN-3-OL, D-GLUTAMIC ACID, GLUTAMATE RACEMASE
Authors:	Lundqvist, T.
Deposit date:	2008-11-25
Release date:	2008-12-09
Last modified:	2023-12-13
Method:	X-RAY DIFFRACTION (1.87 Å)
Cite:	Potent and selective inhibitors of Helicobacter pylori glutamate racemase (MurI): pyridodiazepine amines. Bioorg. Med. Chem. Lett., 19, 2009

GlmU in complex with a Quinazoline Compound
Descriptor:	Bifunctional protein GlmU, N-{4-[(7-hydroxy-6-methoxyquinazolin-4-yl)amino]phenyl}benzamide, SULFATE ION, ...
Authors:	Larsen, N.A, Doig, P.
Deposit date:	2012-03-06
Release date:	2013-05-29
Last modified:	2024-02-28
Method:	X-RAY DIFFRACTION (2 Å)
Cite:	An aminoquinazoline inhibitor of the essential bacterial cell wall synthetic enzyme GlmU has a unique non-protein-kinase-like binding mode. Biochem.J., 446, 2012