2QR7
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![BU of 2qr7 by Molmil](/molmil-images/mine/2qr7) | |
3KN5
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![BU of 3kn5 by Molmil](/molmil-images/mine/3kn5) | |
3KN6
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![BU of 3kn6 by Molmil](/molmil-images/mine/3kn6) | |
2QR8
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![BU of 2qr8 by Molmil](/molmil-images/mine/2qr8) | |
4N0S
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![BU of 4n0s by Molmil](/molmil-images/mine/4n0s) | Complex of ERK2 with caffeic acid | Descriptor: | CAFFEIC ACID, DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, ... | Authors: | Kurinov, I, Malakhova, M. | Deposit date: | 2013-10-02 | Release date: | 2014-08-27 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.7992 Å) | Cite: | Caffeic Acid Directly Targets ERK1/2 to Attenuate Solar UV-Induced Skin Carcinogenesis. Cancer Prev Res (Phila), 7, 2014
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3SA0
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![BU of 3sa0 by Molmil](/molmil-images/mine/3sa0) | Complex of ERK2 with norathyriol | Descriptor: | Mitogen-activated protein kinase 1, SULFATE ION, norathyriol | Authors: | Kurinov, I, Malakhova, M. | Deposit date: | 2011-06-02 | Release date: | 2011-12-14 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (1.5947 Å) | Cite: | Norathyriol Suppresses Skin Cancers Induced by Solar Ultraviolet Radiation by Targeting ERK Kinases. Cancer Res., 72, 2012
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5WP1
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![BU of 5wp1 by Molmil](/molmil-images/mine/5wp1) | Complex of ERK2 with 5,7-dihydroxychromone | Descriptor: | 5,7-dihydroxy-4H-1-benzopyran-4-one, BENZOIC ACID, Mitogen-activated protein kinase 1, ... | Authors: | Kurinov, I, Malakhova, M. | Deposit date: | 2017-08-03 | Release date: | 2018-08-08 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (1.4 Å) | Cite: | Multiple phytochemicals at low doses accumulatively inhibit one key protein in cancers To Be Published
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4ZXT
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![BU of 4zxt by Molmil](/molmil-images/mine/4zxt) | Complex of ERK2 with catechol | Descriptor: | AMMONIUM ION, CATECHOL, Mitogen-activated protein kinase 1, ... | Authors: | Kurinov, I, Malakhova, M. | Deposit date: | 2015-05-20 | Release date: | 2016-05-25 | Last modified: | 2016-10-05 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | A natural small molecule, catechol, induces c-Myc degradation by directly targeting ERK2 in lung cancer. Oncotarget, 7, 2016
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1SBX
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![BU of 1sbx by Molmil](/molmil-images/mine/1sbx) | Crystal structure of the Dachshund-homology domain of human SKI | Descriptor: | Ski oncogene | Authors: | Wilson, J.J, Malakhova, M, Zhang, R, Joachimiak, A, Hegde, R.S. | Deposit date: | 2004-02-11 | Release date: | 2004-05-25 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (1.65 Å) | Cite: | Crystal Structure of the Dachshund Homology Domain of human SKI Structure, 12, 2004
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3G51
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![BU of 3g51 by Molmil](/molmil-images/mine/3g51) | |