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5NOB
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BU of 5nob by Molmil
Crystal structure of human tankyrase 2 in complex with OD336
分子名称: 1-[3-[4-(2-chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxidanylidene-3~{H}-benzimidazole-5-carbonitrile, Tankyrase-2, ZINC ION
著者Ignatev, A, Lehtio, L.
登録日2017-04-11
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach.
J. Med. Chem., 60, 2017
3CPH
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BU of 3cph by Molmil
Crystal structure of Sec4 in complex with Rab-GDI
分子名称: GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Rab GDP-dissociation inhibitor, ...
著者Kravchenko, S, Ignatev, A, Goody, R.S, Rak, A, Pylypenko, O.
登録日2008-03-31
公開日2008-05-06
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献A structural model of the GDP dissociation inhibitor rab membrane extraction mechanism.
J.Biol.Chem., 283, 2008
3CPJ
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BU of 3cpj by Molmil
Crystal structure of Ypt31 in complex with yeast Rab-GDI
分子名称: CHLORIDE ION, GTP-binding protein YPT31/YPT8, GUANOSINE-5'-DIPHOSPHATE, ...
著者Kravchenko, S, Ignatev, A, Goody, R.S, Rak, A, Pylypenko, O.
登録日2008-03-31
公開日2008-05-06
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献A structural model of the GDP dissociation inhibitor rab membrane extraction mechanism.
J.Biol.Chem., 283, 2008
3CPI
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BU of 3cpi by Molmil
Crystal structure of yeast Rab-GDI
分子名称: Rab GDP-dissociation inhibitor
著者Kravchenko, S, Ignatev, A, Goody, R.S, Rak, A, Pylypenko, O.
登録日2008-03-31
公開日2008-05-06
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献A structural model of the GDP dissociation inhibitor rab membrane extraction mechanism.
J.Biol.Chem., 283, 2008
5AEH
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BU of 5aeh by Molmil
Crystal structure of human tankyrase 2 in complex with OD332
分子名称: N-{4-[(2-chlorophenyl)(pyrimidin-4-yl)carbamoyl]phenyl}-4-methoxybenzamide, TANKYRASE-2, ZINC ION
著者Ignatev, A, Lehtio, L.
登録日2015-08-31
公開日2016-01-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Development and Structural Analysis of Adenosine Site Binding Tankyrase Inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016
4CBW
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BU of 4cbw by Molmil
Crystal structure of Plasmodium berghei actin I with D-loop from muscle actin
分子名称: 1,4-DIETHYLENE DIOXIDE, ACTIN, ALPHA SKELETAL MUSCLE, ...
著者Vahokoski, J, Bhargav, S.P, Desfosses, A, Andreadaki, M, Kumpula, E.P, Ignatev, A, Munico Martinez, S, Lepper, S, Frischknecht, F, Siden-Kiamos, I, Sachse, C, Kursula, I.
登録日2013-10-17
公開日2014-04-30
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.501 Å)
主引用文献Structural Differences Explain Diverse Functions of Plasmodium Actins.
Plos Pathog., 10, 2014
4CBU
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BU of 4cbu by Molmil
Crystal structure of Plasmodium falciparum actin I
分子名称: ACTIN-1, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ...
著者Vahokoski, J, Bhargav, S.P, Desfosses, A, Andreadaki, M, Kumpula, E.P, Ignatev, A, Munico Martinez, S, Lepper, S, Frischknecht, F, Siden-Kiamos, I, Sachse, C, Kursula, I.
登録日2013-10-16
公開日2014-04-30
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Structural Differences Explain Diverse Functions of Plasmodium Actins.
Plos Pathog., 10, 2014
4CBX
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BU of 4cbx by Molmil
Crystal structure of Plasmodium berghei actin II
分子名称: ACTIN-2, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ...
著者Vahokoski, J, Bhargav, S.P, Desfosses, A, Andreadaki, M, Kumpula, E.P, Ignatev, A, Munico Martinez, S, Lepper, S, Frischknecht, F, Siden-Kiamos, I, Sachse, C, Kursula, I.
登録日2013-10-17
公開日2014-04-30
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural Differences Explain Diverse Functions of Plasmodium Actins.
Plos Pathog., 10, 2014
5NSP
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BU of 5nsp by Molmil
Crystal structure of TNKS2 in complex with OD334
分子名称: 1-[4-[4-(2-chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]phenyl]-2-oxidanylidene-3~{H}-benzimidazole-5-carbonitrile, BICARBONATE ION, GLYCEROL, ...
著者Nkizinkiko, Y, Haikarainen, T, Lehtio, L.
登録日2017-04-26
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach.
J. Med. Chem., 60, 2017
5ADT
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BU of 5adt by Molmil
Crystal structure of human tankyrase 2 in complex with OD73
分子名称: BICARBONATE ION, N-[3-chloranyl-4-[[4-(4-methoxyphenyl)oxan-4-yl]methylcarbamoyl]phenyl]-2-methyl-1,3-oxazole-5-carboxamide, SULFATE ION, ...
著者Haikarainen, T, Lehtio, L.
登録日2015-08-24
公開日2016-01-13
最終更新日2016-01-20
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Development and Structural Analysis of Adenosine Site Binding Tankyrase Inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016
5ADS
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BU of 5ads by Molmil
Crystal structure of human tankyrase 2 in complex with OD39
分子名称: BICARBONATE ION, DI(HYDROXYETHYL)ETHER, GLYCEROL, ...
著者Haikarainen, T, Lehtio, L.
登録日2015-08-24
公開日2016-01-13
最終更新日2016-01-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Development and Structural Analysis of Adenosine Site Binding Tankyrase Inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016
5ADR
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BU of 5adr by Molmil
Crystal structure of human tankyrase 2 in complex with OD38
分子名称: BICARBONATE ION, N-(4-(((4-(4-methoxyphenyl)oxan-4- yl)methyl)carbamoyl)phenyl)-5-methylfuran-2-carboxamide, SULFATE ION, ...
著者Haikarainen, T, Lehtio, L.
登録日2015-08-24
公開日2016-01-13
最終更新日2016-01-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Development and Structural Analysis of Adenosine Site Binding Tankyrase Inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016
5ADQ
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BU of 5adq by Molmil
Crystal structure of human tankyrase 2 in complex with JW55
分子名称: BICARBONATE ION, GLYCEROL, N-(4-(((4-(4-methoxyphenyl)oxan-4- yl)methyl)carbamoyl)phenyl)furan-2-carboxamide, ...
著者Haikarainen, T, Lehtio, L.
登録日2015-08-24
公開日2016-01-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Development and Structural Analysis of Adenosine Site Binding Tankyrase Inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016

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件を2024-04-24に公開中

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