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Crystal structure of EphA4 kinase domain
Descriptor:	EPHRIN TYPE-A RECEPTOR 4, GLYCEROL
Authors:	Farenc, C.J.A, Celie, P.H.N, Siegal, G.
Deposit date:	2011-01-25
Release date:	2011-11-02
Last modified:	2023-12-20
Method:	X-RAY DIFFRACTION (1.7 Å)
Cite:	Crystal Structure of the Epha4 Protein Tyrosine Kinase Domain in the Apo- and Dasatinib-Bound State. FEBS Lett., 585, 2011

Crystal structure of EphA4 kinase domain in complex with Dasatinib.
Descriptor:	EPHRIN TYPE-A RECEPTOR 4, N-(2-CHLORO-6-METHYLPHENYL)-2-({6-[4-(2-HYDROXYETHYL)PIPERAZIN-1-YL]-2-METHYLPYRIMIDIN-4-YL}AMINO)-1,3-THIAZOLE-5-CARBOXAMIDE
Authors:	Farenc, C.J.A, Celie, P.H.N, Siegal, G.
Deposit date:	2011-01-25
Release date:	2011-11-02
Last modified:	2023-12-20
Method:	X-RAY DIFFRACTION (1.543 Å)
Cite:	Crystal Structure of the Epha4 Protein Tyrosine Kinase Domain in the Apo- and Dasatinib-Bound State. FEBS Lett., 585, 2011

Crystal structure of EphA4 kinase domain in complex with VUF 12058
Descriptor:	5-(5-FLUORO-2-METHYLPHENYL)-6,7,8,9-TETRAHYDRO-3H-PYRAZOLO[3,4-C]ISOQUINOLIN-1-AMINE, EPHRIN TYPE-A RECEPTOR 4,, GLYCEROL
Authors:	Farenc, C.J.A, Celie, P.H.N, vanLinden, O.P.J, Siegal, G.
Deposit date:	2010-11-19
Release date:	2011-11-30
Last modified:	2023-12-20
Method:	X-RAY DIFFRACTION (2.117 Å)
Cite:	Fragment Based Lead Discovery of Small Molecule Inhibitors for the Epha4 Receptor Tyrosine Kinase. Eur.J.Med.Chem., 47, 2012