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2SKD
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PYRIDOXAL PHOSPHORYLASE B IN COMPLEX WITH PHOSPHATE, GLUCOSE AND INOSINE-5'-MONOPHOSPHATE
分子名称: INOSINIC ACID, PHOSPHATE ION, PYRIDOXAL PHOSPHORYLASE B, ...
著者Oikonomakos, N.G, Zographos, S.E, Tsitsanou, K.E, Johnson, L.N, Acharya, K.R.
登録日1998-12-11
公開日1998-12-16
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Activator anion binding site in pyridoxal phosphorylase b: the binding of phosphite, phosphate, and fluorophosphate in the crystal.
Protein Sci., 5, 1996
2VFZ
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CRYSTAL STRUCTURE OF ALPHA-1,3 GALACTOSYLTRANSFERASE (R365K) IN COMPLEX WITH UDP-2F-GALACTOSE
分子名称: MANGANESE (II) ION, N-ACETYLLACTOSAMINIDE ALPHA-1,3-GALACTOSYL TRANSFERASE, URIDINE-5'-DIPHOSPHATE-2-DEOXY-2-FLUOROGALACTOSE
著者Jamaluddin, H, Tumbale, P, Withers, S.G, Acharya, K.R, Brew, K.
登録日2007-11-06
公開日2007-11-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Conformational Changes Induced by Binding Udp-2F-Galactose to Alpha-1,3 Galactosyltransferase-Implications for Catalysis
J.Mol.Biol., 369, 2007
1C5D
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THE CRYSTAL STRUCTURE OF THE FAB FRAGMENT OF A RAT MONOCLONAL ANTIBODY AGAINST THE MAIN IMMUNOGENIC REGION OF THE HUMAN MUSCLE ACETYLCHOLINE RECEPTOR
分子名称: MONOCLONAL ANTIBODY AGAINST THE MAIN IMMUNOGENIC REGION OF THE HUMAN MUSCLE ACETYLCHOLINE RECEPTOR
著者Kontou, M, Leonidas, D.D, Vatzaki, E.H, Tsantili, P, Mamalaki, A, Oikonomakos, N.G, Acharya, K.R, Tzartos, S.J.
登録日1999-11-17
公開日1999-12-03
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The crystal structure of the Fab fragment of a rat monoclonal antibody against the main immunogenic region of the human muscle acetylcholine receptor.
Eur.J.Biochem., 267, 2000
2VS5
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THE BINDING OF UDP-GALACTOSE BY AN ACTIVE SITE MUTANT OF alpha-1,3 GALACTOSYLTRANSFERASE (alpha3GT)
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, GALACTOSE-URIDINE-5'-DIPHOSPHATE, MANGANESE (II) ION, ...
著者Tumbale, P, Jamaluddin, H, Thiyagarajan, N, Brew, K, Acharya, K.R.
登録日2008-04-18
公開日2008-07-15
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献Structural Basis of Udp-Galactose Binding by Alpha- 1,3-Galactosyltransferase (Alpha3Gt): Role of Negative Charge on Aspartic Acid 316 in Structure and Activity.
Biochemistry, 47, 2008
2VS3
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THE BINDING OF UDP-GALACTOSE BY AN ACTIVE SITE MUTANT OF alpha-1,3 GALACTOSYLTRANSFERASE (alpha3GT)
分子名称: MANGANESE (II) ION, N-ACETYLLACTOSAMINIDE ALPHA-1,3-GALACTOSYLTRANSFERASE, URIDINE-5'-DIPHOSPHATE, ...
著者Tumbale, P, Jamaluddin, H, Thiyagarajan, N, Brew, K, Acharya, K.R.
登録日2008-04-18
公開日2008-07-15
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural Basis of Udp-Galactose Binding by Alpha- 1,3-Galactosyltransferase (Alpha3Gt): Role of Negative Charge on Aspartic Acid 316 in Structure and Activity.
Biochemistry, 47, 2008
2VS4
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THE BINDING OF UDP-GALACTOSE BY AN ACTIVE SITE MUTANT OF alpha-1,3 GALACTOSYLTRANSFERASE (alpha3GT)
分子名称: GLYCEROL, MANGANESE (II) ION, N-ACETYLLACTOSAMINIDE ALPHA-1,3-GALACTOSYLTRANSFERASE, ...
著者Tumbale, P, Jamaluddin, H, Thiyagarajan, N, Brew, K, Acharya, K.R.
登録日2008-04-18
公開日2008-07-15
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Structural Basis of Udp-Galactose Binding by Alpha- 1,3-Galactosyltransferase (Alpha3Gt): Role of Negative Charge on Aspartic Acid 316 in Structure and Activity.
Biochemistry, 47, 2008
2W5G
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RNASE A-5'-ATP COMPLEX
分子名称: ADENOSINE-5'-TRIPHOSPHATE, RIBONUCLEASE PANCREATIC
著者Chavali, G.B, Holloway, D.E, Baker, M.D, Acharya, K.R.
登録日2008-12-10
公開日2009-02-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Influence of Naturally-Occurring 5'-Pyrophosphate- Linked Substituents on the Binding of Adenylic Inhibitors to Ribonuclease A: An X-Ray Crystallographic Study.
Biopolymers, 91, 2009
2WD2
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A chimeric microtubule disruptor with efficacy on a taxane resistant cell line
分子名称: 7-methoxy-2-(3-methoxybenzyl)-1,2,3,4-tetrahydroisoquinolin-6-yl sulfamate, CARBONIC ANHYDRASE 2, FORMIC ACID, ...
著者Leese, M.P, Jourdan, F.L, Kimberley, M.R, Cozier, G.E, Regis-Lydi, S, Foster, P.A, Newman, S.P, Thiyagarajan, N, Acharya, K.R, Ferrandis, E, Purohit, A, Reed, M.J, Potter, B.V.L.
登録日2009-03-19
公開日2010-03-31
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Chimeric Microtubule Disruptors.
Chem.Commun.(Camb.), 46, 2010
2WGZ
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Crystal structure of alpha-1,3 galactosyltransferase (alpha3GT) in a complex with p-nitrophenyl-beta-galactoside (pNP-beta-Gal)
分子名称: 4-nitrophenyl beta-D-galactopyranoside, GLYCEROL, MANGANESE (II) ION, ...
著者Jamaluddin, H, Tumbale, P, Ferns, T.A, Thiyagarajan, N, Brew, K, Acharya, K.R.
登録日2009-04-28
公開日2009-06-16
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Crystal Structure of Alpha-1,3 Galactosyltransferase (Alpha3Gt) in a Complex with P-Nitrophenyl-Beta-Galactoside (Pnpbetagal).
Biochem.Biophys.Res.Commun., 385, 2009
2W2D
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Crystal Structure of a Catalytically Active, Non-toxic Endopeptidase Derivative of Clostridium botulinum Toxin A
分子名称: ACETATE ION, BOTULINUM NEUROTOXIN A HEAVY CHAIN, BOTULINUM NEUROTOXIN A LIGHT CHAIN, ...
著者Masuyer, G, Thiyagarajan, N, James, P.L, Marks, P.M.H, Chaddock, J.A, Acharya, K.R.
登録日2008-10-29
公開日2009-03-24
最終更新日2022-05-04
実験手法X-RAY DIFFRACTION (2.59 Å)
主引用文献Crystal Structure of a Catalytically Active, Non-Toxic Endopeptidase Derivative of Clostridium Botulinum Toxin A.
Biochem.Biophys.Res.Commun., 381, 2009
2W5L
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RNASE A-NADP COMPLEX
分子名称: NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, RIBONUCLEASE PANCREATIC
著者Chavali, G.B, Holloway, D.E, Baker, M.D, Acharya, K.R.
登録日2008-12-10
公開日2009-02-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Influence of Naturally-Occurring 5'-Pyrophosphate-Linked Substituents on the Binding of Adenylic Inhibitors to Ribonuclease A: An X-Ray Crystallographic Study.
Biopolymers, 91, 2009
2VWE
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Crystal Structure of Vascular Endothelial Growth Factor-B in Complex with a Neutralizing Antibody Fab Fragment
分子名称: ANTI-VEGF-B MONOCLONAL ANTIBODY, VASCULAR ENDOTHELIAL GROWTH FACTOR B
著者Leonard, P, Scotney, P.D, Jabeen, T, Iyer, S, Fabri, L.J, Nash, A.D, Acharya, K.R.
登録日2008-06-23
公開日2008-11-04
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Crystal Structure of Vascular Endothelial Growth Factor-B in Complex with a Neutralising Antibody Fab Fragment.
J.Mol.Biol., 384, 2008
2R3Z
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Crystal structure of mouse IP-10
分子名称: Small-inducible cytokine B10
著者Jabeen, T, Leonard, P, Jamaluddin, H, Acharya, K.R.
登録日2007-08-30
公開日2008-08-12
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structure of mouse IP-10, a chemokine
Acta Crystallogr.,Sect.D, 64, 2008
2VQ8
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RNASE ZF-1A
分子名称: CHLORIDE ION, RNASE ZF-1A
著者Kazakou, K, Holloway, D.E, Prior, S.H, Subramanian, V, Acharya, K.R.
登録日2008-03-12
公開日2008-06-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Ribonuclease A Homologues of the Zebrafish: Polymorphism, Crystal Structures of Two Representatives and Their Evolutionary Implications.
J.Mol.Biol., 380, 2008
2VXL
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Screening a Limited Structure-based Library Identifies UDP-GalNAc- Specific Mutants of alpha-1,3 Galactosyltransferase
分子名称: MANGANESE (II) ION, N-ACETYLLACTOSAMINIDE ALPHA-1,3-GALACTOSYLTRANSFERASE, URIDINE-5'-DIPHOSPHATE
著者Tumbale, P, Jamaluddin, H, Thiyagarajan, N, Acharya, K.R, Brew, K.
登録日2008-07-07
公開日2008-09-23
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Screening a Limited Structure-Based Library Identifies Udp-Galnac-Specific Mutants of {Alpha}-1,3-Galactosyltransferase.
Glycobiology, 18, 2008
2VQ9
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RNASE ZF-3E
分子名称: CHLORIDE ION, RNASE 1
著者Kazakou, K, Holloway, D.E, Prior, S.H, Subramanian, V, Acharya, K.R.
登録日2008-03-12
公開日2008-06-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Ribonuclease A Homologues of the Zebrafish: Polymorphism, Crystal Structures of Two Representatives and Their Evolutionary Implications
J.Mol.Biol., 380, 2008
2W5K
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RNASE A-NADPH COMPLEX
分子名称: NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, RIBONUCLEASE PANCREATIC
著者Chavali, G.B, Holloway, D.E, Baker, M.D, Acharya, K.R.
登録日2008-12-10
公開日2009-02-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Influence of Naturally-Occurring 5'-Pyrophosphate-Linked Substituents on the Binding of Adenylic Inhibitors to Ribonuclease A: An X-Ray Crystallographic Study.
Biopolymers, 91, 2009
1DT2
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CRYSTAL STRUCTURE OF EXFOLIATIVE TOXIN B
分子名称: EXFOLIATIVE TOXIN B
著者Papageorgiou, A.C, Plano, L.R.W, Collins, C.M, Acharya, K.R.
登録日2000-01-11
公開日2003-01-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural similarities and differences in Staphylococcus aureus exfoliative toxins A and B as revealed by their crystal structures.
Protein Sci., 9, 2000
1DUA
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CRYSTAL STRUCTURE OF EXFOLIATIVE TOXIN A
分子名称: EXFOLIATIVE TOXIN A
著者Papageorgiou, A.C, Plano, L.R.W, Collins, C.M, Acharya, K.R.
登録日2000-01-17
公開日2003-01-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural similarities and differences in Staphylococcus aureus exfoliative toxins A and B as revealed by their crystal structures.
Protein Sci., 9, 2000
2W5M
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RNASE A-PYROPHOSPHATE ION COMPLEX
分子名称: PYROPHOSPHATE 2-, RIBONUCLEASE PANCREATIC
著者Chavali, G.B, Holloway, D.E, Baker, M.D, Acharya, K.R.
登録日2008-12-10
公開日2009-02-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Influence of Naturally-Occurring 5'-Pyrophosphate-Linked Substituents on the Binding of Adenylic Inhibitors to Ribonuclease A: An X-Ray Crystallographic Study.
Biopolymers, 91, 2009
2VXM
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Screening a Limited Structure-based Library Identifies UDP-GalNAc- Specific Mutants of alpha-1,3 Galactosyltransferase
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, GLYCEROL, N-ACETYLLACTOSAMINIDE ALPHA-1,3-GALACTOSYLTRANSFERASE
著者Tumbale, P, Jamaluddin, H, Thiyagarajan, N, Acharya, K.R, Brew, K.
登録日2008-07-07
公開日2008-09-23
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.82 Å)
主引用文献Screening a Limited Structure-Based Library Identifies Udp-Galnac-Specific Mutants of {Alpha}-1,3-Galactosyltransferase.
Glycobiology, 18, 2008
2WD3
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Highly Potent First Examples of Dual Aromatase-Steroid Sulfatase Inhibitors based on a Biphenyl Template
分子名称: 3-CHLORO-2'-CYANO-5'-(1H-1,2,4-TRIAZOL-1-YLMETHYL)BIPHENYL-4-YL SULFAMATE, CARBONIC ANHYDRASE 2, ZINC ION
著者Woo, L.W.L, Jackson, T, Putey, A, Cozier, G, Leonard, P, Acharya, K.R, Chander, S.K, Purohit, A, Reed, M.J, Potter, B.V.L.
登録日2009-03-19
公開日2010-02-23
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Highly Potent First Examples of Dual Aromatase-Steroid Sulfatase Inhibitors Based on a Biphenyl Template.
J.Med.Chem., 53, 2010
2W5I
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RNASE A-AP3A COMPLEX
分子名称: ADENOSINE-5'-TRIPHOSPHATE, RIBONUCLEASE PANCREATIC
著者Chavali, G.B, Holloway, D.E, Baker, M.D, Acharya, K.R.
登録日2008-12-10
公開日2009-02-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Influence of Naturally-Occurring 5'-Pyrophosphate-Linked Substituents on the Binding of Adenylic Inhibitors to Ribonuclease A: An X-Ray Crystallographic Study.
Biopolymers, 91, 2009
2X93
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Crystal structure of AnCE-trandolaprilat complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ANGIOTENSIN CONVERTING ENZYME, ...
著者Akif, M, Georgiadis, D, Mahajan, A, Dive, V, Sturrock, E.D, Isaac, R.E, Acharya, K.R.
登録日2010-03-14
公開日2010-06-02
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献High Resolution Crystal Structures of Drosophila Melanogaster Angiotensin Converting Enzyme in Complex with Novel Inhibitors and Anti- Hypertensive Drugs.
J.Mol.Biol., 400, 2010
1FZV
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THE CRYSTAL STRUCTURE OF HUMAN PLACENTA GROWTH FACTOR-1 (PLGF-1), AN ANGIOGENIC PROTEIN AT 2.0A RESOLUTION
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, PLACENTA GROWTH FACTOR
著者Iyer, S, Leonidas, D.D, Swaminathan, G.J, Maglione, D, Battisti, M, Tucci, M, Persico, M.G, Acharya, K.R.
登録日2000-10-04
公開日2001-05-09
最終更新日2022-12-21
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The crystal structure of human placenta growth factor-1 (PlGF-1), an angiogenic protein, at 2.0 A resolution.
J.Biol.Chem., 276, 2001

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