8JT9
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![BU of 8jt9 by Molmil](/molmil-images/mine/8jt9) | Human VMAT2 complex with ketanserin | Descriptor: | 3-[2-[4-(4-fluorophenyl)carbonylpiperidin-1-yl]ethyl]-1~{H}-quinazoline-2,4-dione, Synaptic vesicular amine transporter | Authors: | Jiang, D.H, Wu, D. | Deposit date: | 2023-06-21 | Release date: | 2023-11-29 | Last modified: | 2024-02-21 | Method: | ELECTRON MICROSCOPY (2.97 Å) | Cite: | Transport and inhibition mechanisms of human VMAT2. Nature, 626, 2024
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8JTC
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![BU of 8jtc by Molmil](/molmil-images/mine/8jtc) | Human VMAT2 complex with reserpine | Descriptor: | Synaptic vesicular amine transporter, reserpine | Authors: | Jiang, D.H, Wu, D. | Deposit date: | 2023-06-21 | Release date: | 2023-11-29 | Last modified: | 2024-02-21 | Method: | ELECTRON MICROSCOPY (3.52 Å) | Cite: | Transport and inhibition mechanisms of human VMAT2. Nature, 626, 2024
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7X3U
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![BU of 7x3u by Molmil](/molmil-images/mine/7x3u) | cryo-EM structure of human TRiC-ADP | Descriptor: | ADENOSINE-5'-DIPHOSPHATE, T-complex protein 1 subunit alpha, T-complex protein 1 subunit beta, ... | Authors: | Cong, Y, Liu, C.X. | Deposit date: | 2022-03-01 | Release date: | 2023-06-07 | Last modified: | 2024-06-26 | Method: | ELECTRON MICROSCOPY (3.3 Å) | Cite: | Pathway and mechanism of tubulin folding mediated by TRiC/CCT along its ATPase cycle revealed using cryo-EM. Commun Biol, 6, 2023
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7X3J
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![BU of 7x3j by Molmil](/molmil-images/mine/7x3j) | Cryo-EM structure of human TRiC-tubulin-S2 | Descriptor: | ADENOSINE-5'-TRIPHOSPHATE, T-complex protein 1 subunit alpha, T-complex protein 1 subunit beta, ... | Authors: | Cong, Y, Liu, C.X. | Deposit date: | 2022-03-01 | Release date: | 2023-06-07 | Last modified: | 2023-07-05 | Method: | ELECTRON MICROSCOPY (4.2 Å) | Cite: | Pathway and mechanism of tubulin folding mediated by TRiC/CCT along its ATPase cycle revealed using cryo-EM. Commun Biol, 6, 2023
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7X6Q
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![BU of 7x6q by Molmil](/molmil-images/mine/7x6q) | cryo-EM structure of human TRiC-ATP-closed state | Descriptor: | T-complex protein 1 subunit alpha, T-complex protein 1 subunit beta, T-complex protein 1 subunit delta, ... | Authors: | Cong, Y, Liu, C.X. | Deposit date: | 2022-03-08 | Release date: | 2023-06-07 | Last modified: | 2024-06-26 | Method: | ELECTRON MICROSCOPY (4.5 Å) | Cite: | Pathway and mechanism of tubulin folding mediated by TRiC/CCT along its ATPase cycle revealed using cryo-EM. Commun Biol, 6, 2023
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7X7Y
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![BU of 7x7y by Molmil](/molmil-images/mine/7x7y) | Cryo-EM structure of Human TRiC-ATP-open state | Descriptor: | T-complex protein 1 subunit alpha, T-complex protein 1 subunit beta, T-complex protein 1 subunit delta, ... | Authors: | Cong, Y, Liu, C.X. | Deposit date: | 2022-03-10 | Release date: | 2023-06-07 | Last modified: | 2024-06-26 | Method: | ELECTRON MICROSCOPY (3.8 Å) | Cite: | Pathway and mechanism of tubulin folding mediated by TRiC/CCT along its ATPase cycle revealed using cryo-EM. Commun Biol, 6, 2023
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7X0V
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![BU of 7x0v by Molmil](/molmil-images/mine/7x0v) | cryo-EM structure of human TRiC-ADP-AlFx | Descriptor: | ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MAGNESIUM ION, ... | Authors: | Cong, Y, Liu, C.X. | Deposit date: | 2022-02-22 | Release date: | 2023-04-12 | Last modified: | 2024-06-26 | Method: | ELECTRON MICROSCOPY (3.2 Å) | Cite: | Pathway and mechanism of tubulin folding mediated by TRiC/CCT along its ATPase cycle revealed using cryo-EM. Commun Biol, 6, 2023
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7X0S
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![BU of 7x0s by Molmil](/molmil-images/mine/7x0s) | Human TRiC-tubulin-S3 | Descriptor: | ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MAGNESIUM ION, ... | Authors: | Cong, Y, Liu, C.X. | Deposit date: | 2022-02-22 | Release date: | 2023-04-12 | Last modified: | 2024-06-26 | Method: | ELECTRON MICROSCOPY (3.1 Å) | Cite: | Pathway and mechanism of tubulin folding mediated by TRiC/CCT along its ATPase cycle revealed using cryo-EM. Commun Biol, 6, 2023
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7X0A
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![BU of 7x0a by Molmil](/molmil-images/mine/7x0a) | Cryo-EM structure of human TRiC-NPP state | Descriptor: | T-complex protein 1 subunit alpha, T-complex protein 1 subunit beta, T-complex protein 1 subunit delta, ... | Authors: | Cong, Y, Liu, C.X. | Deposit date: | 2022-02-21 | Release date: | 2023-04-12 | Last modified: | 2024-06-26 | Method: | ELECTRON MICROSCOPY (3.1 Å) | Cite: | Pathway and mechanism of tubulin folding mediated by TRiC/CCT along its ATPase cycle revealed using cryo-EM. Commun Biol, 6, 2023
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5WQE
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![BU of 5wqe by Molmil](/molmil-images/mine/5wqe) | |
7CJT
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![BU of 7cjt by Molmil](/molmil-images/mine/7cjt) | Crystal Structure of SETDB1 Tudor domain in complexed with (R,R)-59 | Descriptor: | 2-[[(3~{R},5~{R})-1-methyl-5-(4-phenylmethoxyphenyl)piperidin-3-yl]amino]-3-prop-2-enyl-5~{H}-pyrrolo[3,2-d]pyrimidin-4-one, Histone-lysine N-methyltransferase SETDB1 | Authors: | Guo, Y.P, Liang, X, Mao, X, Wu, C, Luyi, H, Yang, S. | Deposit date: | 2020-07-13 | Release date: | 2021-04-14 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (2.474 Å) | Cite: | Structure-Guided Discovery of a Potent and Selective Cell-Active Inhibitor of SETDB1 Tudor Domain. Angew.Chem.Int.Ed.Engl., 60, 2021
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7CAJ
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![BU of 7caj by Molmil](/molmil-images/mine/7caj) | Crystal structure of SETDB1 Tudor domain in complexed with Compound 2. | Descriptor: | 3-methyl-2-[[(3R,5R)-1-methyl-5-phenyl-piperidin-3-yl]amino]-5H-pyrrolo[3,2-d]pyrimidin-4-one, Histone-lysine N-methyltransferase SETDB1 | Authors: | Guo, Y.P, Liang, X, Xin, M, Luyi, H, Chengyong, W, Yang, S.Y. | Deposit date: | 2020-06-08 | Release date: | 2021-04-07 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (2.198 Å) | Cite: | Structure-Guided Discovery of a Potent and Selective Cell-Active Inhibitor of SETDB1 Tudor Domain. Angew.Chem.Int.Ed.Engl., 60, 2021
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7WVP
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![BU of 7wvp by Molmil](/molmil-images/mine/7wvp) | |
7WVQ
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![BU of 7wvq by Molmil](/molmil-images/mine/7wvq) | |
7CPC
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![BU of 7cpc by Molmil](/molmil-images/mine/7cpc) | |
7CPI
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![BU of 7cpi by Molmil](/molmil-images/mine/7cpi) | |
7CQO
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![BU of 7cqo by Molmil](/molmil-images/mine/7cqo) | Lysozyme grown in LCP soaked with selenourea for 6 min | Descriptor: | CHLORIDE ION, Lysozyme C, SODIUM ION, ... | Authors: | Luo, Z.P, Li, D.F. | Deposit date: | 2020-08-11 | Release date: | 2021-08-11 | Last modified: | 2022-08-31 | Method: | X-RAY DIFFRACTION (1.71 Å) | Cite: | Selenourea for experimental phasing of membrane protein crystals grown in lipid cubic phase Crystals, 12, 2022
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7CQM
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![BU of 7cqm by Molmil](/molmil-images/mine/7cqm) | PlsY grown in LCP soaked with selenourea for 22 min | Descriptor: | (2R)-2,3-dihydroxypropyl (7Z)-hexadec-7-enoate, Glycerol-3-phosphate acyltransferase, SULFATE ION, ... | Authors: | Luo, Z.P, Li, D.F. | Deposit date: | 2020-08-11 | Release date: | 2021-08-11 | Last modified: | 2024-05-29 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Selenourea for experimental phasing of membrane protein crystals grown in lipid cubic phase Crystals, 12, 2022
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8WRJ
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![BU of 8wrj by Molmil](/molmil-images/mine/8wrj) | glycosyltransferase UGT74AN3 | Descriptor: | 5-[(1R,2S,4R,6R,7R,10S,11S,14S,16R)-14-hydroxy-7,11-dimethyl-3-oxapentacyclo[8.8.0.02,4.02,7.011,16]octadecan-6-yl]pyran-2-one, Glycosyltransferase, URIDINE-5'-DIPHOSPHATE | Authors: | Huang, W, Long, F. | Deposit date: | 2023-10-15 | Release date: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Substrate Promiscuity, Crystal Structure, and Application of a Plant UDP-Glycosyltransferase UGT74AN3 Acs Catalysis, 14, 2024
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8WRK
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![BU of 8wrk by Molmil](/molmil-images/mine/8wrk) | glycosyltransferase UGT74AN3 | Descriptor: | Glycosyltransferase, PICEATANNOL, URIDINE-5'-DIPHOSPHATE | Authors: | Huang, W, Long, F. | Deposit date: | 2023-10-15 | Release date: | 2024-01-24 | Method: | X-RAY DIFFRACTION (2.03 Å) | Cite: | Substrate Promiscuity, Crystal Structure, and Application of a Plant UDP-Glycosyltransferase UGT74AN3 Acs Catalysis, 14, 2024
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6AH4
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![BU of 6ah4 by Molmil](/molmil-images/mine/6ah4) | Structure of human P2X3 receptor in complex with ATP and Ca2+ ion | Descriptor: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ADENOSINE-5'-TRIPHOSPHATE, ... | Authors: | Hattori, M. | Deposit date: | 2018-08-16 | Release date: | 2019-06-12 | Last modified: | 2020-12-23 | Method: | X-RAY DIFFRACTION (3.296 Å) | Cite: | Molecular mechanisms of human P2X3 receptor channel activation and modulation by divalent cation bound ATP. Elife, 8, 2019
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7E56
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![BU of 7e56 by Molmil](/molmil-images/mine/7e56) | |
7E3O
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![BU of 7e3o by Molmil](/molmil-images/mine/7e3o) | |
6B0T
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![BU of 6b0t by Molmil](/molmil-images/mine/6b0t) | |
6AYK
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![BU of 6ayk by Molmil](/molmil-images/mine/6ayk) | |