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Human PPAR gamma ligand binding domain in complex with a gammma selective synthetic partial agonist MEKT75
Descriptor:	N-(phenylsulfonyl)-4-propoxy-3-({[4-(pyrimidin-2-yl)benzoyl]amino}methyl)benzamide, Peroxisome proliferator-activated receptor gamma
Authors:	Oyama, T, Ohashi, M, Miyachi, H, Kusunoki, M.
Deposit date:	2013-11-19
Release date:	2014-11-19
Last modified:	2023-11-08
Method:	X-RAY DIFFRACTION (2.1 Å)
Cite:	Human PPRR gamma ligand binding domain in complex with a gammma selective synthetic partial agonist MEKT75 TO BE PUBLISHED

Human PPAR gamma ligand binding domain in complex with JKPL53
Descriptor:	(2S)-2-{4-butoxy-3-[({4-[(3S,5S,7S)-tricyclo[3.3.1.1~3,7~]dec-1-yl]benzoyl}amino)methyl]benzyl}butanoic acid, Peroxisome proliferator-activated receptor gamma
Authors:	Tomioka, D, Kuwabara, N, Hashimoto, H, Sato, M, Shimizu, T.
Deposit date:	2011-10-20
Release date:	2012-08-29
Last modified:	2023-11-08
Method:	X-RAY DIFFRACTION (2.61 Å)
Cite:	Peroxisome proliferator-activated receptors (PPARs) have multiple binding points that accommodate ligands in various conformations: phenylpropanoic acid-type PPAR ligands bind to PPAR in different conformations, depending on the subtype. J.Med.Chem., 55, 2012

Human PPAR GAMMA ligand binding domain in complex with JKPL35
Descriptor:	(2S)-2-[4-methoxy-3-({[4-(trifluoromethyl)benzoyl]amino}methyl)benzyl]pentanoic acid, Peroxisome proliferator-activated receptor gamma
Authors:	Tomioka, D, Kuwabara, N, Hashimoto, H, Sato, M, Shimizu, T.
Deposit date:	2011-10-20
Release date:	2012-08-29
Last modified:	2023-11-08
Method:	X-RAY DIFFRACTION (2.22 Å)
Cite:	Peroxisome proliferator-activated receptors (PPARs) have multiple binding points that accommodate ligands in various conformations: phenylpropanoic acid-type PPAR ligands bind to PPAR in different conformations, depending on the subtype. J.Med.Chem., 55, 2012