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7MIR
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BU of 7mir by Molmil
Cryo-EM structure of SidJ-SdeA-CaM reaction intermediate complex
Descriptor: ADENOSINE MONOPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ...
Authors:Osinski, A, Black, M.H, Pawlowski, K, Chen, Z, Li, Y, Tagliabracci, V.S.
Deposit date:2021-04-17
Release date:2021-08-18
Last modified:2024-05-29
Method:ELECTRON MICROSCOPY (2.5 Å)
Cite:Structural and mechanistic basis for protein glutamylation by the kinase fold.
Mol.Cell, 81, 2021
7MIS
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BU of 7mis by Molmil
Cryo-EM structure of SidJ-SdeC-CaM reaction intermediate complex
Descriptor: ADENOSINE MONOPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ...
Authors:Osinski, A, Black, M.H, Pawlowski, K, Chen, Z, Li, Y, Tagliabracci, V.S.
Deposit date:2021-04-17
Release date:2021-08-18
Last modified:2021-11-17
Method:ELECTRON MICROSCOPY (2.8 Å)
Cite:Structural and mechanistic basis for protein glutamylation by the kinase fold.
Mol.Cell, 81, 2021
7THM
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BU of 7thm by Molmil
SARS-CoV-2 nsp12/7/8 complex with a native N-terminus nsp9
Descriptor: MANGANESE (II) ION, Non-structural protein 7, Non-structural protein 8, ...
Authors:Osinski, A, Tagliabracci, V.S, Chen, Z, Li, Y.
Deposit date:2022-01-11
Release date:2022-03-16
Last modified:2024-01-17
Method:ELECTRON MICROSCOPY (3.18 Å)
Cite:The mechanism of RNA capping by SARS-CoV-2.
Nature, 609, 2022
6AR2
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BU of 6ar2 by Molmil
Structure of human SLMAP FHA domain in complex with pMST2
Descriptor: ASP-GLY-TPO-MET-LYS-ARG, Sarcolemmal membrane-associated protein
Authors:Osinski, A, Ni, L, Luo, X.
Deposit date:2017-08-21
Release date:2018-07-04
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:SAV1 promotes Hippo kinase activation through antagonizing the PP2A phosphatase STRIPAK.
Elife, 6, 2017
6OQQ
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BU of 6oqq by Molmil
Legionella pneumophila SidJ/Saccharomyces cerevisiae calmodulin complex
Descriptor: 1,2-ETHANEDIOL, ADENOSINE MONOPHOSPHATE, CALCIUM ION, ...
Authors:Tomchick, D.R, Tagliabracci, V.S, Black, M, Osinski, A.
Deposit date:2019-04-28
Release date:2019-05-15
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.102 Å)
Cite:Bacterial pseudokinase catalyzes protein polyglutamylation to inhibit the SidE-family ubiquitin ligases.
Science, 364, 2019
6AR0
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BU of 6ar0 by Molmil
Structure of human SLMAP FHA domain
Descriptor: Sarcolemmal membrane-associated protein
Authors:Ni, L, Luo, X.
Deposit date:2017-08-21
Release date:2018-07-04
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.08 Å)
Cite:SAV1 promotes Hippo kinase activation through antagonizing the PP2A phosphatase STRIPAK.
Elife, 6, 2017
6AO5
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BU of 6ao5 by Molmil
Crystal structure of human MST2 in complex with SAV1 SARAH domain
Descriptor: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Protein salvador homolog 1, ...
Authors:Tomchick, D.R, Luo, X, Ni, L.
Deposit date:2017-08-15
Release date:2017-11-08
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.955 Å)
Cite:SAV1 promotes Hippo kinase activation through antagonizing the PP2A phosphatase STRIPAK.
Elife, 6, 2017
7M7A
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BU of 7m7a by Molmil
Legionella pneumophila MavQ lipid kinase
Descriptor: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Phosphoinositide 3-kinase MavQ
Authors:Tomchick, D.R, Tagliabracci, V.S, Hsieh, T.S, Lopez, V.A.
Deposit date:2021-03-27
Release date:2021-04-28
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:Dynamic remodeling of host membranes by self-organizing bacterial effectors.
Science, 372, 2021
3LEA
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BU of 3lea by Molmil
Crystal structure of the catalytic domain of TACE with Isoindolinone-biphenyl-hydantoin inhibitor
Descriptor: 2-{[(4R)-2,5-dioxo-4-(4-pyridin-3-ylphenyl)imidazolidin-4-yl]methyl}-6-methoxy-1-oxo-1H-isoindolium, Disintegrin and metalloproteinase domain-containing protein 17, ISOPROPYL ALCOHOL, ...
Authors:Orth, P.
Deposit date:2010-01-14
Release date:2010-12-08
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2 Å)
Cite:Biaryl substituted hydantoin compounds as TACE inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
3LE9
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BU of 3le9 by Molmil
Crystal structure of the catalytic domain of TACE with Indazolinone-phenyl-hydantoin inhibitor
Descriptor: (5R)-5-[(5-methoxy-3-oxo-1,3-dihydro-2H-indazol-2-yl)methyl]-5-phenylimidazolidine-2,4-dione, Disintegrin and metalloproteinase domain-containing protein 17, ISOPROPYL ALCOHOL, ...
Authors:Orth, P.
Deposit date:2010-01-14
Release date:2010-12-08
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Biaryl substituted hydantoin compounds as TACE inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010

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数据于2024-07-17公开中

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