5RDB
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![BU of 5rdb by Molmil](/molmil-images/mine/5rdb) | PanDDA analysis group deposition -- Endothiapepsin ground state model 33 | Descriptor: | ACETATE ION, DI(HYDROXYETHYL)ETHER, Endothiapepsin, ... | Authors: | Weiss, M.S, Wollenhaupt, J, Metz, A, Barthel, T, Lima, G.M.A, Heine, A, Mueller, U, Klebe, G. | Deposit date: | 2020-03-24 | Release date: | 2020-06-03 | Last modified: | 2020-06-17 | Method: | X-RAY DIFFRACTION (1.04 Å) | Cite: | F2X-Universal and F2X-Entry: Structurally Diverse Compound Libraries for Crystallographic Fragment Screening. Structure, 28, 2020
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5RDP
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![BU of 5rdp by Molmil](/molmil-images/mine/5rdp) | PanDDA analysis group deposition -- Endothiapepsin ground state model 41 | Descriptor: | Endothiapepsin | Authors: | Weiss, M.S, Wollenhaupt, J, Metz, A, Barthel, T, Lima, G.M.A, Heine, A, Mueller, U, Klebe, G. | Deposit date: | 2020-03-24 | Release date: | 2020-06-03 | Last modified: | 2020-06-17 | Method: | X-RAY DIFFRACTION (0.97 Å) | Cite: | F2X-Universal and F2X-Entry: Structurally Diverse Compound Libraries for Crystallographic Fragment Screening. Structure, 28, 2020
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5OG7
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![BU of 5og7 by Molmil](/molmil-images/mine/5og7) | Endothiapepsin in complex with hydrazide fragment | Descriptor: | 3-chloranyl-~{N}'-(4,5-dihydro-1~{H}-imidazol-3-ium-2-yl)propanehydrazide, DIMETHYL SULFOXIDE, Endothiapepsin | Authors: | Metz, A, Klauser, P.C, Heine, A, Klebe, G. | Deposit date: | 2017-07-12 | Release date: | 2018-08-08 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.823 Å) | Cite: | Endothiapepsin in complex with hydrazide fragment To Be Published
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5SW3
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![BU of 5sw3 by Molmil](/molmil-images/mine/5sw3) | Crystal Structure of TGT in complex with 3-Pyridinecarboxylic acid, 6-(dimethylamino) | Descriptor: | 6-(dimethylamino)pyridine-3-carboxylic acid, DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, ... | Authors: | Hassaan, E, Heine, A, Klebe, G. | Deposit date: | 2016-08-08 | Release date: | 2017-07-19 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.38 Å) | Cite: | Fragments as Novel Starting Points for tRNA-Guanine Transglycosylase Inhibitors Found by Alternative Screening Strategies. Chemmedchem, 15, 2020
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5UTJ
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![BU of 5utj by Molmil](/molmil-images/mine/5utj) | Crystal Structure of TGT in complex with 2,6-dioxy-8-azapurine, 2,6-dioxy-8-azapurine, 2,6-dioxy-8-azapurine | Descriptor: | 8-AZAXANTHINE, DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, ... | Authors: | Hassaan, E, Heine, A, Klebe, G. | Deposit date: | 2017-02-15 | Release date: | 2018-03-07 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.549 Å) | Cite: | Fragments as Novel Starting Points for tRNA-Guanine Transglycosylase Inhibitors Found by Alternative Screening Strategies. Chemmedchem, 15, 2020
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5V3C
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![BU of 5v3c by Molmil](/molmil-images/mine/5v3c) | Crystal structure of TGT in complex with 4-(aminomethane)cyclohexane-1-carboxylic acid | Descriptor: | DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, Queuine tRNA-ribosyltransferase, ... | Authors: | Hassaan, E, Heine, A, Klebe, G. | Deposit date: | 2017-03-07 | Release date: | 2018-05-16 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.419 Å) | Cite: | Fragments as Novel Starting Points for tRNA-Guanine Transglycosylase Inhibitors Found by Alternative Screening Strategies. Chemmedchem, 15, 2020
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5OYU
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![BU of 5oyu by Molmil](/molmil-images/mine/5oyu) | |
5OZ3
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5OZC
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5OYX
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5OZ7
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5OZI
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5OZT
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5P06
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![BU of 5p06 by Molmil](/molmil-images/mine/5p06) | |
5OZ6
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![BU of 5oz6 by Molmil](/molmil-images/mine/5oz6) | |
5OZH
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5OZB
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![BU of 5ozb by Molmil](/molmil-images/mine/5ozb) | |
5OZP
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![BU of 5ozp by Molmil](/molmil-images/mine/5ozp) | |
5P03
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![BU of 5p03 by Molmil](/molmil-images/mine/5p03) | |
5P0I
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5P0U
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5P19
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5P1P
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5P23
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5P2F
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![BU of 5p2f by Molmil](/molmil-images/mine/5p2f) | |