6DXJ
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![BU of 6dxj by Molmil](/molmil-images/mine/6dxj) | |
6DY5
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![BU of 6dy5 by Molmil](/molmil-images/mine/6dy5) | |
6DY9
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![BU of 6dy9 by Molmil](/molmil-images/mine/6dy9) | |
7JSA
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![BU of 7jsa by Molmil](/molmil-images/mine/7jsa) | |
7JSL
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![BU of 7jsl by Molmil](/molmil-images/mine/7jsl) | |
7V0B
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![BU of 7v0b by Molmil](/molmil-images/mine/7v0b) | |
7V0D
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![BU of 7v0d by Molmil](/molmil-images/mine/7v0d) | Crystal structure of halogenase CtcP from Kitasatospora aureofaciens | Descriptor: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ... | Authors: | Hou, C, Tsodikov, O.V. | Deposit date: | 2022-05-10 | Release date: | 2023-05-17 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Crystal structures and complex formation of halogenase CtcP and FAD reductase CtcQ from the chlortetracycline biosynthetic pathway To Be Published
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4I9G
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![BU of 4i9g by Molmil](/molmil-images/mine/4i9g) | Crystal structure of glycerol phosphate phosphatase Rv1692 from Mycobacterium tuberculosis in complex with magnesium | Descriptor: | Glycerol 3-phosphate phosphatase, MAGNESIUM ION | Authors: | Biswas, T, Larrouy-Maumus, G, de Carvalho, L.P, Tsodikov, O.V. | Deposit date: | 2012-12-05 | Release date: | 2013-07-10 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (3.25 Å) | Cite: | Discovery of a glycerol 3-phosphate phosphatase reveals glycerophospholipid polar head recycling in Mycobacterium tuberculosis. Proc.Natl.Acad.Sci.USA, 110, 2013
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4I9F
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![BU of 4i9f by Molmil](/molmil-images/mine/4i9f) | Crystal structure of glycerol phosphate phosphatase Rv1692 from Mycobacterium tuberculosis in complex with calcium | Descriptor: | CALCIUM ION, CHLORIDE ION, Glycerol 3-phosphate phosphatase | Authors: | Biswas, T, Larrouy-Maumus, G, de Carvalho, L.P, Tsodikov, O.V. | Deposit date: | 2012-12-05 | Release date: | 2013-07-10 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.21 Å) | Cite: | Discovery of a glycerol 3-phosphate phosphatase reveals glycerophospholipid polar head recycling in Mycobacterium tuberculosis. Proc.Natl.Acad.Sci.USA, 110, 2013
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4IJJ
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![BU of 4ijj by Molmil](/molmil-images/mine/4ijj) | Structure of transcription factor DksA2 from Pseudomonas aeruginosa | Descriptor: | Putative C4-type zinc finger protein, DksA/TraR family, SULFATE ION | Authors: | Biswas, T, Furman, R, Artsimovitch, I, Tsodikov, O.V. | Deposit date: | 2012-12-21 | Release date: | 2013-02-27 | Last modified: | 2013-03-27 | Method: | X-RAY DIFFRACTION (3.25 Å) | Cite: | DksA2, a zinc-independent structural analog of the transcription factor DksA. Febs Lett., 587, 2013
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9BDV
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![BU of 9bdv by Molmil](/molmil-images/mine/9bdv) | NF-kappaB RelA homo-dimer bound to TA-centric kappaB DNA | Descriptor: | DNA (5'-D(*AP*TP*CP*AP*CP*TP*GP*GP*AP*AP*AP*TP*TP*CP*CP*CP*AP*GP*T)-3'), DNA (5'-D(P*AP*CP*TP*GP*GP*GP*AP*AP*TP*TP*TP*CP*CP*AP*GP*TP*GP*AP*T)-3'), SULFATE ION, ... | Authors: | Biswas, T, Shahabi, S, Tsodikov, O.V. | Deposit date: | 2024-04-12 | Release date: | 2024-04-24 | Last modified: | 2024-06-12 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Transient interactions modulate the affinity of NF-kappa B transcription factors for DNA. Proc.Natl.Acad.Sci.USA, 121, 2024
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9BDW
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![BU of 9bdw by Molmil](/molmil-images/mine/9bdw) | NF-kappaB RelA homo-dimer bound to GC-centric kappaB DNA | Descriptor: | DNA (5'-D(P*AP*CP*TP*GP*GP*GP*AP*AP*GP*TP*TP*CP*CP*AP*GP*TP*GP*AP*T)-3'), DNA (5'-D(P*AP*TP*CP*AP*CP*TP*GP*GP*AP*AP*CP*TP*TP*CP*CP*CP*AP*GP*T)-3'), SULFATE ION, ... | Authors: | Biswas, T, Shahabi, S, Tsodikov, O.V, Huang, D, Ghosh, G. | Deposit date: | 2024-04-12 | Release date: | 2024-04-24 | Last modified: | 2024-06-12 | Method: | X-RAY DIFFRACTION (1.87 Å) | Cite: | Transient interactions modulate the affinity of NF-kappa B transcription factors for DNA. Proc.Natl.Acad.Sci.USA, 121, 2024
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9BDX
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![BU of 9bdx by Molmil](/molmil-images/mine/9bdx) | NF-kappaB RelA homo-dimer bound to CG-centric kappaB DNA | Descriptor: | DNA (5'-D(*AP*TP*CP*AP*CP*TP*GP*GP*AP*AP*GP*TP*TP*CP*CP*CP*AP*GP*T)-3'), DNA (5'-D(P*AP*CP*TP*GP*GP*GP*AP*AP*CP*TP*TP*CP*CP*AP*GP*TP*GP*AP*T)-3'), Transcription factor p65 | Authors: | Biswas, T, Shahabi, S, Tsodikov, O.V, Ghosh, G. | Deposit date: | 2024-04-12 | Release date: | 2024-04-24 | Last modified: | 2024-06-12 | Method: | X-RAY DIFFRACTION (3.6 Å) | Cite: | Transient interactions modulate the affinity of NF-kappa B transcription factors for DNA. Proc.Natl.Acad.Sci.USA, 121, 2024
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3R1K
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![BU of 3r1k by Molmil](/molmil-images/mine/3r1k) | Crystal structure of acetyltransferase Eis from Mycobacterium tuberculosis H37Rv in complex with CoA and an acetamide moiety | Descriptor: | ACETAMIDE, COENZYME A, Enhanced intracellular survival protein | Authors: | Biswas, T, Chen, W, Garneau-Tsodikova, S, Tsodikov, O.V. | Deposit date: | 2011-03-10 | Release date: | 2011-06-01 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB. Proc.Natl.Acad.Sci.USA, 108, 2011
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3ITW
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![BU of 3itw by Molmil](/molmil-images/mine/3itw) | |
3K6Z
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![BU of 3k6z by Molmil](/molmil-images/mine/3k6z) | Crystal structure of Rv3671c protease, inactive form | Descriptor: | POSSIBLE MEMBRANE-ASSOCIATED SERINE PROTEASE | Authors: | Biswas, T, Small, J, Vandal, O, Ehrt, S, Tsodikov, O.V. | Deposit date: | 2009-10-10 | Release date: | 2010-10-13 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.75 Å) | Cite: | Structural insight into serine protease Rv3671c that Protects M. tuberculosis from oxidative and acidic stress. Structure, 18, 2010
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3I6B
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![BU of 3i6b by Molmil](/molmil-images/mine/3i6b) | |
3K6Y
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![BU of 3k6y by Molmil](/molmil-images/mine/3k6y) | Crystal structure of Rv3671c protease from M. tuberculosis, active form | Descriptor: | POSSIBLE MEMBRANE-ASSOCIATED SERINE PROTEASE | Authors: | Biswas, T, Small, J, Vandal, O, Ehrt, S, Tsodikov, O.V. | Deposit date: | 2009-10-10 | Release date: | 2010-10-13 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.3 Å) | Cite: | Structural insight into serine protease Rv3671c that Protects M. tuberculosis from oxidative and acidic stress. Structure, 18, 2010
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4RPA
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![BU of 4rpa by Molmil](/molmil-images/mine/4rpa) | |
4RV9
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![BU of 4rv9 by Molmil](/molmil-images/mine/4rv9) | Crystal structure of MtmC in complex with SAH | Descriptor: | ACETATE ION, CHLORIDE ION, D-mycarose 3-C-methyltransferase, ... | Authors: | Hou, C, Chen, J.-M, Rohr, J, Tsodikov, O.V. | Deposit date: | 2014-11-25 | Release date: | 2015-02-04 | Last modified: | 2023-12-06 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Structural Insight into MtmC, a Bifunctional Ketoreductase-Methyltransferase Involved in the Assembly of the Mithramycin Trisaccharide Chain. Biochemistry, 54, 2015
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5E8G
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![BU of 5e8g by Molmil](/molmil-images/mine/5e8g) | |
5EBV
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![BU of 5ebv by Molmil](/molmil-images/mine/5ebv) | Crystal structure of acetyltransferase Eis from Mycobacterium tuberculosis in complex with inhibitor 11c and CoA | Descriptor: | 5-(4-chlorophenyl)-~{N}-[3-(3,4-dihydro-1~{H}-isoquinolin-2-yl)propyl]-4-methyl-1,1-bis(oxidanylidene)-1,2-thiazol-3-amine, CHLORIDE ION, COENZYME A, ... | Authors: | Gajadeera, C.S, Hou, C, Garneau-Tsodikova, S, Tsodikov, O.V. | Deposit date: | 2015-10-19 | Release date: | 2016-03-30 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Potent Inhibitors of Acetyltransferase Eis Overcome Kanamycin Resistance in Mycobacterium tuberculosis. Acs Chem.Biol., 11, 2016
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5EC4
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![BU of 5ec4 by Molmil](/molmil-images/mine/5ec4) | Crystal structure of acetyltransferase Eis from Mycobacterium tuberculosis in complex with inhibitor 13g and CoA | Descriptor: | 5-(3-chlorophenyl)-4-methyl-~{N}-(3-morpholin-4-ylpropyl)-1,1-bis(oxidanylidene)-1,2-thiazol-3-amine, COENZYME A, Enhanced intracellular survival protein | Authors: | Gajadeera, C.S, Hou, C, Garneau-Tsodikova, S, Tsodikov, O.V. | Deposit date: | 2015-10-20 | Release date: | 2016-03-30 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (2.21 Å) | Cite: | Potent Inhibitors of Acetyltransferase Eis Overcome Kanamycin Resistance in Mycobacterium tuberculosis. Acs Chem.Biol., 11, 2016
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5DBJ
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![BU of 5dbj by Molmil](/molmil-images/mine/5dbj) | Crystal structure of halogenase PltA | Descriptor: | CHLORIDE ION, FADH2-dependent halogenase PltA, FLAVIN-ADENINE DINUCLEOTIDE | Authors: | Pang, A.H, Tsodikov, O.V. | Deposit date: | 2015-08-21 | Release date: | 2015-10-07 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (2.75 Å) | Cite: | Crystal structure of halogenase PltA from the pyoluteorin biosynthetic pathway. J.Struct.Biol., 192, 2015
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5E8I
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![BU of 5e8i by Molmil](/molmil-images/mine/5e8i) | |