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7BGU
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BU of 7bgu by Molmil
Mason-Pfizer Monkey Virus Protease mutant C7A/D26N/C106A in complex with peptidomimetic inhibitor
分子名称: Gag-Pro-Pol polyprotein, PENTAETHYLENE GLYCOL, peptidomimetic inhibitor
著者Wosicki, S, Gilski, M, Kazmierczyk, M, Jaskolski, M, Zabranska, H, Pichova, I.
登録日2021-01-08
公開日2021-12-15
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.433 Å)
主引用文献Crystal structures of inhibitor complexes of M-PMV protease with visible flap loops.
Protein Sci., 30, 2021
7BGT
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BU of 7bgt by Molmil
Mason-Pfizer Monkey Virus Protease mutant C7A/D26N/C106A in complex with peptidomimetic inhibitor
分子名称: ACETATE ION, Gag-Pro-Pol polyprotein, PENTAETHYLENE GLYCOL, ...
著者Wosicki, S, Gilski, M, Jaskolski, M, Zabranska, H, Pichova, I.
登録日2021-01-08
公開日2021-12-15
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Crystal structures of inhibitor complexes of M-PMV protease with visible flap loops.
Protein Sci., 30, 2021
6S1U
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BU of 6s1u by Molmil
Crystal structure of dimeric M-PMV protease C7A/D26N/C106A mutant in complex with inhibitor
分子名称: Gag-Pro-Pol polyprotein, PRO-0A1-VAL-PSA-ALA-MET-THR
著者Wosicki, S, Gilski, M, Jaskolski, M, Zabranska, H, Pichova, I.
登録日2019-06-19
公開日2019-10-16
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Comparison of a retroviral protease in monomeric and dimeric states.
Acta Crystallogr D Struct Biol, 75, 2019
6S1W
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BU of 6s1w by Molmil
Crystal structure of dimeric M-PMV protease D26N mutant
分子名称: Gag-Pro-Pol polyprotein
著者Wosicki, S, Gilski, M, Jaskolski, M, Zabranska, H, Pichova, I.
登録日2019-06-19
公開日2019-10-16
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献Comparison of a retroviral protease in monomeric and dimeric states.
Acta Crystallogr D Struct Biol, 75, 2019
6S1V
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BU of 6s1v by Molmil
Crystal structure of dimeric M-PMV protease D26N mutant in complex with inhibitor
分子名称: Gag-Pro-Pol polyprotein, PRO-0A1-VAL-PSA-ALA-MET-THR
著者Wosicki, S, Gilski, M, Jaskolski, M, Zabranska, H, Pichova, I.
登録日2019-06-19
公開日2019-10-16
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.64 Å)
主引用文献Comparison of a retroviral protease in monomeric and dimeric states.
Acta Crystallogr D Struct Biol, 75, 2019
3SQF
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BU of 3sqf by Molmil
Crystal structure of monomeric M-PMV retroviral protease
分子名称: Protease
著者Jaskolski, M, Kazmierczyk, M, Gilski, M, Krzywda, S, Pichova, I, Zabranska, H, Khatib, F, DiMaio, F, Cooper, S, Thompson, J, Popovic, Z, Baker, D, Group, Foldit Contenders
登録日2011-07-05
公開日2011-09-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.6324 Å)
主引用文献Crystal structure of a monomeric retroviral protease solved by protein folding game players.
Nat.Struct.Mol.Biol., 18, 2011
4O1G
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BU of 4o1g by Molmil
MTB adenosine kinase in complex with gamma-Thio-ATP
分子名称: Adenosine kinase, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, SODIUM ION
著者Dostal, J, Brynda, J, Hocek, M, Pichova, I.
登録日2013-12-15
公開日2014-11-26
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structural Basis for Inhibition of Mycobacterial and Human Adenosine Kinase by 7-Substituted 7-(Het)aryl-7-deazaadenine Ribonucleosides
J.Med.Chem., 57, 2014
4PVV
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BU of 4pvv by Molmil
Micobacterial Adenosine Kinase in complex with inhibitor
分子名称: 5-ethynyl-7-(beta-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine, Adenosine kinase
著者Pichova, I, Hocek, M, Dostal, J, Rezacova, P.
登録日2014-03-18
公開日2014-11-26
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Basis for Inhibition of Mycobacterial and Human Adenosine Kinase by 7-Substituted 7-(Het)aryl-7-deazaadenine Ribonucleosides
J.Med.Chem., 57, 2014
4O1L
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BU of 4o1l by Molmil
Human Adenosine Kinase in complex with inhibitor
分子名称: 5-ethynyl-7-(beta-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine, Adenosine kinase, MAGNESIUM ION
著者Brynda, J, Dostal, J, Pichova, I, Hodcek, M.
登録日2013-12-16
公開日2014-11-26
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Basis for Inhibition of Mycobacterial and Human Adenosine Kinase by 7-Substituted 7-(Het)aryl-7-deazaadenine Ribonucleosides
J.Med.Chem., 57, 2014
2D4M
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BU of 2d4m by Molmil
Crystal Structure of apo M-PMV dUTPase
分子名称: DU
著者Nemeth, V, Barabas, O, Vertessy, G.B.
登録日2005-10-20
公開日2006-11-21
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Flexible segments modulate co-folding of dUTPase and nucleocapsid proteins.
Nucleic Acids Res., 35, 2007
2D4L
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BU of 2d4l by Molmil
Crystal structure of truncated in C-terminal M-PMV dUTPase
分子名称: DU
著者Nemeth, V, Barabas, O, Vertessy, G.B.
登録日2005-10-20
公開日2006-11-07
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Flexible segments modulate co-folding of dUTPase and nucleocapsid proteins.
Nucleic Acids Res., 35, 2007
2D4N
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BU of 2d4n by Molmil
Crystal Structure of M-PMV dUTPase complexed with dUPNPP, substrate analogue
分子名称: 2'-DEOXYURIDINE 5'-ALPHA,BETA-IMIDO-TRIPHOSPHATE, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, DU, ...
著者Nemeth, V, Barabas, O, Vertessy, G.B.
登録日2005-10-20
公開日2006-11-21
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Flexible segments modulate co-folding of dUTPase and nucleocapsid proteins.
Nucleic Acids Res., 35, 2007

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件を2024-07-31に公開中

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